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<strong>Extemporaneous</strong> Formulations <strong>for</strong> Pediatric, Geriatric, and Special Needs<br />

Patients<br />

Jew, Rita K. PharmD<br />

ISBN-13: <strong>9781585282456</strong><br />

<strong>Table</strong> <strong>of</strong> <strong>Contents</strong><br />

TABLE OF CONTENTS<br />

Part I: Elixir/Solution/Suspension/Syrup<br />

Acetazolamide Suspension 25 mg/ml ........................................................ 1<br />

Allopurinol Suspension 20 mg/ml ............................................................... 2<br />

Amiodarone Suspension 5 mg/ml ............................................................... 3<br />

Amitriptyline Syrup 1 mg/ml ....................................................................... 4<br />

Amlodipine Suspension 1 mg/ml ................................................................ 5<br />

Amphetamine and Dextroamphetamine (Adderall) Suspension 1 mg/ml ... 6<br />

Atenolol Syrup 2 mg/ml—Formulation 1 .................................................... 7<br />

Atenolol Syrup 2 mg/ml—Formulation 2 .................................................... 8<br />

Azathioprine Suspension 50 mg/ml ............................................................ 9<br />

Bacl<strong>of</strong>en Suspension 10 mg/ml ................................................................ 10<br />

Bacl<strong>of</strong>en Syrup 5 mg/ml ............................................................................11<br />

Bethanechol Solution 1 mg/ml ................................................................. 12<br />

Bethanechol Suspension 5 mg/ml ............................................................ 13<br />

Busulfan Syrup 2 mg/ml ........................................................................... 14<br />

Captopril Solution 1 mg/ml—Formulation 1 .............................................. 15<br />

Captopril Suspension 0.75 mg/ml ............................................................. 16<br />

Captopril Suspension 1 mg/ml—Formulation 2 ........................................ 17<br />

Carvedilol Suspension 0.1 mg/ml ............................................................. 18<br />

Carvedilol Suspension 1.67 mg/ml ........................................................... 19<br />

Chloroquine Phosphate Suspension 15 mg/ml ......................................... 20<br />

Chloroquine Phosphate Syrup 16.7 mg/ml ............................................... 21<br />

Clonazepam Suspension 0.1 mg/ml ......................................................... 22<br />

Clonidine Syrup 0.1 mg/ml ....................................................................... 23<br />

Clopidogrel Suspension 5 mg/ml .............................................................. 24<br />

Cyclophosphamide Elixir 2 mg/ml ............................................................ 25<br />

Dantrolene Syrup 5 mg/ml ........................................................................ 26<br />

Dapsone Suspension 2 mg/ml—Formulation 1 ........................................ 27<br />

Dapsone Syrup 2 mg/ml—Formulation 2 .................................................. 28<br />

Diltiazem Suspension 12 mg/ml ............................................................... 29<br />

Dipyridamole Suspension 10 mg/ml ......................................................... 30<br />

Disopyramide Syrup 1 mg/ml ................................................................... 31<br />

Disopyramide Syrup 10 mg/ml ................................................................. 32<br />

Dolasetron Suspension 10 mg/ml ............................................................. 33<br />

Preface to the First Edition ............................................................................... VIII<br />

Preface to the Second Edition .......................................................................... X<br />

Introduction ...................................................................................................... XI<br />

Enalapril Suspension 1 mg/ml .................................................................. 34<br />

Ethacrynic Acid Solution 1 mg/ml ............................................................ 35<br />

Etoposide Solution 10 mg/ml .................................................................... 36<br />

Flecainide Acetate Suspension 20 mg/ml ................................................ 37<br />

Flecainide Acetate Syrup 5 mg/ml ........................................................... 38<br />

Flucytosine Suspension 10 mg/ml ........................................................... 39<br />

Flucytosine Suspension 50 mg/ml ........................................................... 40<br />

Ganciclovir Syrup 100 mg/ml .................................................................... 41<br />

Hydralazine Suspension 4 mg/ml ............................................................. 42<br />

Hydrocortisone Suspension 1 mg/ml ........................................................ 43<br />

Hydrocortisone Suspension 2 mg/ml ........................................................ 44<br />

Hydroxyurea Syrup 100 mg/ml ................................................................. 45<br />

Hypromellose Suspension 10 mg/ml ........................................................ 46<br />

Isradipine Syrup 1 mg/ml .......................................................................... 47<br />

Ketoconazole Suspension 20 mg/ml ........................................................ 48<br />

Labetalol Suspension 40 mg/ml ............................................................... 49<br />

Labetalol Syrup 10 mg/ml ......................................................................... 50<br />

Lamotrigine Suspension 1 mg/ml ............................................................. 51<br />

Lansoprazole Solution 3 mg/ml ................................................................ 52<br />

Levodopa 5 mg/ml and Carbidopa 1.25 mg/ml Suspension ..................... 53


Levothyroxine Solution 25 mcg/ml ............................................................ 54<br />

Lisinopril Suspension 1 mg/ml—Formulation 1 ........................................ 55<br />

Lisinopril Syrup 1 mg/ml—Formulation 2 ................................................. 56<br />

Lisinopril Syrup 2 mg/ml ........................................................................... 57<br />

Losartan Suspension 2.5 mg/ml ............................................................... 58<br />

Mercaptopurine Syrup 50 mg/ml .............................................................. 59<br />

Methylcellulose Suspension 10 mg/ml ..................................................... 60<br />

Methyldopa Syrup 50 mg/ml ..................................................................... 61<br />

Metolazone Suspension 1 mg/ml ............................................................. 62<br />

Metoprolol Tartrate Suspension 10 mg/ml ................................................ 63<br />

Metronidazole Suspension 10 mg/ml ....................................................... 64<br />

Metronidazole Suspension 50 mg/ml ....................................................... 65<br />

Metronidazole Syrup 5 mg/ml ................................................................... 66<br />

Mexiletine Solution 10 mg/ml ................................................................... 67<br />

Moxifloxacin Suspension 20 mg/ml .......................................................... 68<br />

Naratriptan Suspension 0.5 mg/ml ........................................................... 69<br />

Nifedipine Solution 10 mg/ml .................................................................... 70<br />

Nifedipine Suspension 1 mg/ml ................................................................ 71<br />

Norfloxacin Suspension 20 mg/ml ............................................................ 72<br />

Omeprazole Solution 2 mg/ml .................................................................. 73<br />

Pantoprazole Solution 2 mg/ml—Formulation 1 ....................................... 74<br />

Pantoprazole Solution 2 mg/ml—Formulation 2 ....................................... 75<br />

Pentoxifylline Solution 20 mg/ml .............................................................. 76<br />

Phenoxybenzamine Solution 2 mg/ml ...................................................... 77<br />

Potassium Perchlorate Solution 13.3 mg/ml ............................................ 78<br />

Propylthiouracil Suspension 5 mg/ml ....................................................... 79<br />

Pyrazinamide Suspension 10 mg/ml ........................................................ 80<br />

Pyrazinamide Syrup 100 mg/ml ............................................................... 81<br />

Pyrimethamine Suspension 2 mg/ml ........................................................ 82<br />

Quinidine Sulfate Suspension 10 mg/ml .................................................. 83<br />

Rifabutin Suspension 20 mg/ml ................................................................ 84<br />

Rifampin Suspension 25 mg/ml ................................................................ 85<br />

Rifampin Syrup 10 mg/ml ......................................................................... 86<br />

Sildenafil Suspension 2.5 mg/ml .............................................................. 87<br />

Sotalol Suspension 5 mg/ml ..................................................................... 88<br />

Spironolactone 5 mg/ml and Hydrochlorothiazide 5 mg/ml Suspension .. 89<br />

Spironolactone Suspension 25 mg/ml ...................................................... 90<br />

Spironolactone Syrup 2.5 mg/ml .............................................................. 91<br />

Spironolactone Syrup 5 mg/ml ................................................................. 92<br />

Spironolactone Syrup 10 mg/ml ................................................................ 93<br />

Sulfasalazine Suspension 100 mg/ml ....................................................... 94<br />

Sumatriptan Suspension 5 mg/ml ............................................................ 95<br />

Tacrolimus Suspension 0.5 mg/ml ........................................................... 96<br />

Tacrolimus Suspension 1 mg/ml .............................................................. 97<br />

Temozolomide Suspension 10 mg/ml ....................................................... 98<br />

Terbinafine Suspension 25 mg/ml ............................................................. 99<br />

Terbutaline Syrup 1 mg/ml ...................................................................... 100<br />

Tetracycline Suspension 25 mg/ml ......................................................... 101<br />

Tiagabine Suspension 1 mg/ml .............................................................. 102<br />

Topiramate Suspension 6 mg/ml ............................................................ 103<br />

Tramadol 7.5 mg/ml and Acetaminophen 65 mg/ml Suspension ........... 104<br />

Tramadol Suspension 5 mg/ml ............................................................... 105<br />

Ursodiol Suspension 25 mg/ml ............................................................... 106<br />

Ursodiol Suspension 50 mg/ml ............................................................... 107<br />

Ursodiol Syrup 60 mg/ml ........................................................................ 108<br />

Valacyclovir Suspension 50 mg/ml ......................................................... 109<br />

Verapamil Suspension 50 mg/ml ............................................................. 110<br />

Zonisamide Syrup 10 mg/ml .................................................................... 111<br />

Bacitracin Ophthalmic Solution 9,600 units/ml ....................................... 113<br />

Cefazolin Ophthalmic Solution 33 mg/ml ................................................ 114<br />

Cid<strong>of</strong>ovir Intravitreous Solution 0.2 mg/ml ................................................ 115<br />

Cid<strong>of</strong>ovir Intravitreous Solution 8.1 mg/ml ................................................ 116<br />

Fumagillin Ophthalmic Solution 70 mcg/ml ............................................. 117<br />

Ganciclovir Intravitreous Solution 20 mg/ml ............................................. 118<br />

Part II: Ointment/Ophthalmic Solution<br />

Gentamicin Ophthalmic Solution 13.6 mg/ml (Fortified) ......................... 119<br />

LET (Lidocaine 4%/Racepinephrine 0.225%/Tetracaine 0.5%) Solution 120<br />

Tobramycin Ophthalmic Solution 13.6 mg/ml (Fortified) ........................ 121<br />

Tobramycin Ophthalmic Solution 15 mg/ml ............................................ 122<br />

Vancomycin Ophthalmic Solution 31 mg/ml .......................................... 123<br />

Alprazolam Suspension 1 mg/ml ............................................................ 125


Caffeine Citrate Solution 10 mg/ml ......................................................... 126<br />

Caffeine Citrate Solution 20 mg/ml—Formulation 1 ................................ 127<br />

Caffeine Citrate Syrup 20 mg/ml —Formulation 2 .................................. 128<br />

Carbamazepine Syrup 40 mg/ml ............................................................ 129<br />

Cimetidine Syrup 60 mg/ml .................................................................... 130<br />

Cipr<strong>of</strong>loxacin Suspension 50 mg/ml ....................................................... 131<br />

Famotidine Suspension 8 mg/ml—Formulation 1 ................................... 132<br />

Famotidine Syrup 8 mg/ml—Formulation 2 ............................................ 133<br />

Fluconazole Solution 1 mg/ml ................................................................ 134<br />

Fluoxetine Syrup 1 mg/ml ....................................................................... 135<br />

Fluoxetine Syrup 2 mg/ml ....................................................................... 136<br />

Gabapentin Suspension 100 mg/ml ........................................................ 137<br />

Granisetron Hydrochloride Suspension 0.05 mg/ml ............................... 138<br />

Granisetron Hydrochloride Syrup 0.2 mg/ml .......................................... 139<br />

Indomethacin Syrup 2 mg/ml .................................................................. 140<br />

Itraconazole Suspension 20 mg/ml ........................................................ 141<br />

Itraconazole Syrup 40 mg/ml .................................................................. 142<br />

Lev<strong>of</strong>loxacin Suspension 50 mg/ml ........................................................ 143<br />

Midazolam Gelatin 1 mg/ml .................................................................... 144<br />

Midazolam Gelatin 2 mg/ml .................................................................... 145<br />

Midazolam Syrup 2.5 mg/ml ................................................................... 146<br />

Mycophenolate M<strong>of</strong>etil Suspension 50 mg/ml ........................................ 147<br />

Mycophenolate M<strong>of</strong>etil Syrup 100 mg/ml ............................................... 148<br />

Nizatidine Solution 2.5 mg/ml ................................................................. 149<br />

Ondansetron Suspension 0.8 mg/ml ...................................................... 150<br />

Oseltamivir Syrup 15 mg/ml .................................................................... 151<br />

Phenobarbital Suspension 10 mg/ml ...................................................... 152<br />

Prednisolone Disodium Phosphate Solution 10 mg/ml .......................... 153<br />

Prednisone Syrup 0.5 mg/ml .................................................................. 154<br />

Propranolol Syrup 1 mg/ml ..................................................................... 155<br />

Ranitidine Syrup 15 mg/ml ..................................................................... 156<br />

Tacrolimus Cream 0.1% .......................................................................... 157<br />

Part III: Commercially Available Products<br />

Use extemporaneously prepared <strong>for</strong>mulation only when commercial product is unavailable or a more<br />

dilute or more concentrated product is desired.<br />

Theophylline Suspension 5 mg/ml .......................................................... 158<br />

Trimethoprim Syrup 10 mg/ml ................................................................. 159<br />

Valganciclovir Suspension 30 mg/ml ...................................................... 160<br />

Valganciclovir Suspension 60 mg/ml ...................................................... 161<br />

Zidovudine Syrup 10 mg/ml ..................................................................... 162<br />

Appendix A: ASHP Technical Assistance Bulletin on Compounding Nonsterile Products<br />

in Pharmacies ............................................................................................................. 165<br />

Appendix B: ASHP Guidelines on Pharmacy-Prepared Ophthalmic Products ................................ 175

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