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Pitfalls in Oncologische Pijnbehandeling

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Werk<strong>in</strong>gsmechanisme Opioïden<br />

µ δ κ<br />

Agonisten Oxycodon +++ + +<br />

Hydromorfon +++ + +<br />

Morf<strong>in</strong>e +++ + +<br />

Methadon +++ - -<br />

Fentanyl +++ + -<br />

Partiële Agonist Buprenorf<strong>in</strong>e (+++) - ++<br />

Antagonisten Naloxone +++ + ++<br />

+ aff<strong>in</strong>iteit en <strong>in</strong>tr<strong>in</strong>sieke activiteit<br />

+ aff<strong>in</strong>iteit en geen <strong>in</strong>tr<strong>in</strong>sieke activiteit<br />

- geen of zwakke aff<strong>in</strong>iteit<br />

Naltrexone +++ + +++

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