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PDF (4,3 MB) - Úrad priemyselného vlastníctva SR

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VESTNÍK ÚRADU PRIEMYSELNÉHO VLASTNÍCTVA <strong>SR</strong> 3 - 2008 - SK (preklady patentov)<br />

8 (51) C07D 295/00, C07D 213/00, C07D 333/00,<br />

A61K 31/495, A61P 25/00, A61P 3/00, A61P 1/00<br />

(11) E 2774<br />

(96) 06290494.1, 29.3.2006<br />

(97) 1707564, 12.9.2007<br />

(24) 12.9.2007<br />

(31) 0503071<br />

(32) 30.3.2005<br />

(33) FR<br />

(73) Les Laboratoires Servier, Courbevoie Cedex, FR;<br />

(72) De Nanteuil Guillaume, Suresnes, FR; Portevin<br />

Bernard, Elancourt, FR; Gloanec Philippe, Marly-Le-Roi,<br />

FR; Millan Mark, Le Pecq, FR; Ortuno<br />

Jean-Claude, Bois d'Arcy, FR; Mannoury La<br />

Cour Clotilde, Paris, FR; Gobert Alain, Rueil-<br />

Malmaison, FR;<br />

(74) ROTT, RŮŽIČKA & GUTTMANN, v. o. s.,<br />

Bratislava, SK;<br />

(54) Indalyn-piperazínové deriváty, spôsob ich prípravy<br />

a farmaceutické kompozície s ich obsahom<br />

8 (51) C07D 305/00<br />

(11) E 2754<br />

(96) 04016493.1, 13.7.2004<br />

(97) 1616868, 12.9.2007<br />

(24) 12.9.2007<br />

(73) INDENA S.p.A., Milano, IT;<br />

(72) Gabetta Bruno, Milano, IT; Zini Gianfranco, Milano,<br />

IT;<br />

(74) Majlingová Marta, Ing., Bratislava, SK;<br />

(54) Spôsob získavania paklitaxelu z Taxus rastlín<br />

8 (51) C07D 309/00<br />

(11) E 2764<br />

(96) 05740374.3, 21.4.2005<br />

(97) 1758875, 3.10.2007<br />

(24) 3.10.2007<br />

(31) 04090157, 565849 P<br />

(32) 22.4.2004, 28.4.2004<br />

(33) EP, US<br />

(73) Bayer Schering Pharma Aktiengesellschaft, Berlin,<br />

DE;<br />

(72) PLATZEK Johannes, Berlin, DE; PETROV Orlin,<br />

Berlin, DE; WILLUHN Marc, c/o Zimmer, Düsseldorf,<br />

DE; GRASKE Klaus-Dieter, Berlin, DE;<br />

SKUBALLA Werner, Berlin, DE;<br />

(74) Čechvalová Dagmar, Bratislava, SK;<br />

(86) PCT/EP2005/004492<br />

(87) WO 2005/101950<br />

(54) Chirálne deriváty heptínu na prípravu epotilónov<br />

a spôsob ich prípravy<br />

8 (51) C07D 333/00, C07D 409/00, A61K 31/4427,<br />

A61P 29/00<br />

(11) E 2737<br />

(96) 04701632.4, 13.1.2004<br />

(97) 1583756, 3.10.2007<br />

(24) 3.10.2007<br />

(31) 0300091<br />

(32) 15.1.2003<br />

(33) SE<br />

(73) AstraZeneca AB, Södertälje, SE;<br />

(72) MORLEY Andrew David, AstraZeneca R & D<br />

Alderley, Macclesfield, Cheshire, GB; POYSER<br />

Jeffrey P., AstraZeneca R & D Alderley, Macclesfield,<br />

Cheshire, GB;<br />

(74) Čechvalová Dagmar, Bratislava, SK;<br />

(86) PCT/GB2004/000106<br />

(87) WO 2004/063185<br />

(54) Tiofénové karboxamidy ako inhibítory enzýmu<br />

IKK-2<br />

8 (51) C07D 401/00, C07D 403/00, C07D 407/00,<br />

C07D 409/00, C07D 413/00, A61K 31/4196,<br />

A61K 31/4245, A61P 3/00<br />

(11) E 2830<br />

(96) 03814074.5, 16.12.2003<br />

(97) 1581515, 10.10.2007<br />

(24) 10.10.2007<br />

(31) 435074 P, 458592 P, 503410 P<br />

(32) 20.12.2002, 28.3.2003, 16.9.2003<br />

(33) US, US, US<br />

(73) Merck & Co., Inc., Rahway, New Jersey, US;<br />

(72) WADDELL Sherman T., Rahway, NJ, US; SAN-<br />

TORELLI Gina M., Rahway, NJ, US; MALETIC<br />

Milana M., Rahway, NJ, US; LEEMAN Aaron<br />

H., Rahway, NJ, US; GU Xin, Rahway, NJ, US;<br />

GRAHAM Donald W., Rahway, NJ, US; BAL-<br />

KOVEC James M., Rahway, NJ, US; ASTER<br />

Susan D., Rahway, NJ, US;<br />

(74) Majlingová Marta, Ing., Bratislava, SK;<br />

(86) PCT/US2003/040127<br />

(87) WO 2004/058741<br />

(54) Triazolové deriváty ako inhibítory 11-beta-<br />

-hydroxysteroid dehydrogenázy-1<br />

8 (51) C07D 403/00, C07D 401/00, C07D 417/00,<br />

A61K 31/427, A61P 3/00<br />

(11) E 2846<br />

(96) 03750648.2, 26.9.2003<br />

(97) 1549638, 3.10.2007<br />

(24) 3.10.2007<br />

(31) 415737 P<br />

(32) 3.10.2002<br />

(33) US<br />

(73) F. HOFFMANN-LA ROCHE AG, Basel, CH;<br />

(72) CORBETT Wendy Lea, Randolph, US;<br />

(74) Bušová Eva, JUDr., Bratislava, SK;<br />

(86) PCT/EP2003/010776<br />

(87) WO 2004/031179<br />

(54) Indol-2-karboxamidy ako aktivátory glukokinázy<br />

(GK)<br />

8 (51) C07D 405/00, A61K 31/445<br />

(11) E 2760<br />

(96) 04736513.5, 10.6.2004<br />

(97) 1638959, 19.9.2007<br />

(24) 19.9.2007<br />

(31) PCT/EP03/50237<br />

(32) 19.6.2003<br />

(33) WO<br />

(73) Janssen Pharmaceutica N.V., Beerse, BE;<br />

(72) BOSMANS Jean-Paul René Marie André, Beerse,<br />

BE; GIJSEN Henricus Jacobus Maria, Beerse,<br />

BE; MEVELLEC Laurence Anne, Issy-les-Moulineaux<br />

Cedex 9, FR;

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