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- Page 21 and 22: 21half-life (PBS, pH 7.4)Ref. 0600Q
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- Page 37 and 38: 37CYP3A inhibition (HLM, midazolam
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53cerepStandardprofilesADME-Tox pro
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55Drug developmentThe following CYP
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57❚ Non-KINASE enzyme profile Ref
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59Sample size❚ minimum compound a
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61applicationnotesIN VITRO ADMEAque
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63unnecessary. At Cerep we measure
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65by extrapolation from log D value
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67The analyte peak areas obtained f
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70 ADME-Tox & PK 2011 catalogP-gp
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