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Chemical Library Management in Drug Discovery - KIAS

Chemical Library Management in Drug Discovery - KIAS

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약물성 필터링(HTS팀)Lum<strong>in</strong>escent Cytochrome P450 AssayshERG channel membrane b<strong>in</strong>d<strong>in</strong>g assay- 일차 약물대사시스템 검색- 약물상호작용 검색2D61A2B62E13ACYP3A42C192C9Lightfirefly luciferase약물로 인한 심부정맥과 QT연장증후군 유발 가능성 예측화합물은행 대표화합물 3,000종에 대한 CYP 저해도 검색hERG 저해물질에 대한 전기생리학적결과와 막결합 결과의 상관석 분석

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