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European Patent Bulletin 2012/09 - European Patent Office

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(A61K) I.1(1)<br />

(88) 27.10.2011<br />

(30) 22.04.20<strong>09</strong> DE 1020<strong>09</strong>018474<br />

(54) PARTIKELFÖRMIGE PHARMAZEUTISCHE<br />

ZUSAMMENSETZUNG MIT EINEM OPIOID<br />

UND EINEM OPIOID- ANTAGONISTEN<br />

PARTICULATE PHARMACEUTICAL<br />

COMPOSITION HAVING AN OPIOID AND<br />

AN OPIOID ANTAGONIST<br />

COMPOSITION PHARMACEUTIQUE<br />

PARTICULAIRE CONTENANT UN OPIOÏDE<br />

ET UN ANTAGONISTE OPIOÏDE<br />

(71) Hermann, Lars Holger, Paulistrasse 69, 8834<br />

Schindellegi, CH<br />

(72) Hermann, Lars Holger, 8834 Schindellegi,<br />

CH<br />

(74) Winkler, Andreas Fritz Ernst, et al, Forrester<br />

& Boehmert Pettenkoferstrasse 20-22,<br />

80336 München, DE<br />

A61K 9/50 → (51) A61K 9/52<br />

(51) A61K 9/51 (11) 2 421 516 A1*<br />

A61K 31/192 A61K 31/496<br />

A01N 29/04 A61K 31/196<br />

A61K 31/5415 A01N 55/02<br />

A61K 31/405 B01J 2/00<br />

A01N 57/00 A61K 31/415<br />

A61K 31/137 A61K 31/421<br />

(25) En (26) En<br />

(21) 10766514.3 (22) 23.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) AU 2010/000465 23.04.2010<br />

(87) WO 2010/121321 2010/43 28.10.2010<br />

(30) 24.04.20<strong>09</strong> AU 20<strong>09</strong>901741<br />

24.04.20<strong>09</strong> US 172301 P<br />

(54) VERFAHREN ZUR VERBESSERUNG DES<br />

AUFLÖSUNGSPROFILS EINES BIOLO-<br />

GISCH AKTIVEN MATERIALS<br />

METHOD FOR IMPROVING THE DISSO-<br />

LUTION PROFILE OF A BIOLOGICALLY<br />

ACTIVE MATERIAL<br />

PROCÉDÉ D'AMÉLIORATION DU PROFIL<br />

DE DISSOLUTION D'UNE MATIÈRE<br />

BIOLOGIQUEMENT ACTIVE<br />

(71) Iceutica Pty Ltd., 52 Fairfield Street, Mouth<br />

Hawthorn, WA 6016, AU<br />

(72) DODD, Aaron, Centennial Park New South<br />

Wales 2021, AU<br />

MEISER, Felix, Mount Claremont Western<br />

Australia 6010, AU<br />

RUSSELL, Adrian, Rivervale Western<br />

Australia 6103, AU<br />

NORRET, Marck, Darlington Western<br />

Australia 6070, AU<br />

BOSCH, William, H., Bryn Mawr Pennsylvania<br />

19010, US<br />

CALLAHAN, Matt, Mount Hawthorn Western<br />

Australia 6016, AU<br />

(74) Coehn, Markus, et al, Fish & Richardson P.C.<br />

Mies-van-der-Rohe-Strasse 8, 80807 München,<br />

DE<br />

A61K 9/51 → (51) A61K 9/52<br />

A61K 9/51 → (51) A61K 31/196<br />

(51) A61K 9/52 (11) 2 421 517 A2*<br />

A61K 9/50 A61K 9/51<br />

A61K 47/30 A61M 35/00<br />

(25) En (26) En<br />

(21) 10767428.5 (22) 21.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/001191 21.04.2010<br />

(87) WO 2010/123563 2010/43 28.10.2010<br />

(88) 17.03.2011<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(30) 23.04.20<strong>09</strong> US 386853<br />

23.04.20<strong>09</strong> US 214452 P<br />

25.11.20<strong>09</strong> US 592536<br />

(54) SPENDEVORRICHTUNG MIT GESTEUER-<br />

TER AUSGABE<br />

CONTROLLED RELEASE DISPENSING<br />

DEVICE<br />

DISPOSITIF D'ADMINISTRATION À LIBÉ-<br />

RATION CONTRÔLÉE<br />

(71) Sustained Nano Systems Llc, 19 Shore Park<br />

Road, Great Neck, NY 11023, US<br />

(72) BARRY, Libin, Great Neck, NY 11023, US<br />

LIEBMANN, Jeffrey, M., Great Neck, NY<br />

11023, US<br />

CHEN, Weiliam, MT Sinai, NY 11766, US<br />

(74) Bottero, Carlo, et al, Barzano' & Zanardo<br />

Milano S.p.A. Via Borgonuovo, 10, <strong>2012</strong>1<br />

Milano, IT<br />

A61K 9/68 → (51) A61K 9/14<br />

A61K 9/70 → (51) A61N 1/30<br />

(51) A61K 9/72 (11) 2 421 518 A2*<br />

(25) En (26) En<br />

(21) 10714832.2 (22) 23.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) US 2010/032228 23.04.2010<br />

(87) WO 2010/124203 2010/43 28.10.2010<br />

(88) 15.12.2011<br />

(30) 24.04.20<strong>09</strong> US 172340 P<br />

(54) AGGLOMERAT-FORMULIERUNGEN MIT<br />

PHARMAZEUTISCHEN WIRKSTOFFEN<br />

MIT GEZIELTEN TEILCHENGRÖSSEN<br />

AGGLOMERATE FORMULATIONS<br />

INCLUDING ACTIVE PHARMACEUTICAL<br />

AGENTS WITH TARGETED PARTICLE<br />

SIZES<br />

PRÉPARATIONS D'AGGLOMÉRAT<br />

COMPRENANT DES AGENTS PHARMA-<br />

CEUTIQUES ACTIFS AYANT DES TAILLES<br />

DE PARTICULES CIBLÉES<br />

(71) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) PANDEY, Preetanshu, Springfield New<br />

Jersey 07081, US<br />

CHAMARTHY, Sai Prasanth, Springfield New<br />

Jersey 07081, US<br />

WYLIE, Jennifer, Lynn, Cranford New Jersey<br />

07016, US<br />

(74) Horgan, James Michael Frederic, Merck &<br />

Co., Inc. <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon EN11 9BU, GB<br />

A61K 9/72 → (51) A61K 9/16<br />

(51) A61K 31/00 (11) 2 421 519 A1*<br />

A61K 31/13 A61K 31/4468<br />

A61P 7/00 A61P 7/06<br />

(25) En (26) En<br />

(21) 10713975.0 (22) 18.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/055077 18.04.2010<br />

(87) WO 2010/121973 2010/43 28.10.2010<br />

(30) 23.04.20<strong>09</strong> EP <strong>09</strong>005683<br />

(54) NMDA-REZEPTOR-BLOCKER ZUR BE-<br />

HANDLUNG VON SICHELZELLANÄMIE<br />

BLOCKERS OF NMDA RECEPTOR FOR<br />

THE TREATMENT OF SICKLE CELL<br />

ANEMIA<br />

BLOQUEURS DE RÉCEPTEUR NMDA<br />

POUR LE TRAITEMENT D'UNE DRÉPA-<br />

NOCYTOSE<br />

(71) Universität Zürich, Rämistrasse 71, 8006<br />

Zürich, CH<br />

38<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>09</strong>/<strong>2012</strong>) 29.02.<strong>2012</strong><br />

(72) BOGDANOVA, Anna, Yulienva, CH-8051 Zürich,<br />

CH<br />

GASSMANN, Max, CH-8047 Zürich, CH<br />

GOEDE, Jeroen, CH-8620 Wetzikon, CH<br />

(74) Schmauder, Klaus Dieter, Schmauder &<br />

Partner AG <strong>Patent</strong>anwälte Zwängiweg 7,<br />

8038 Zürich, CH<br />

(51) A61K 31/00 (11) 2 421 520 A1*<br />

A61K 31/047 A61K 31/19<br />

A61K 31/70 A61K 31/715<br />

A61K 38/38 A61K 47/26<br />

A61K 47/48<br />

(25) En (26) En<br />

(21) 10717816.2 (22) 19.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

RS<br />

(86) IB 2010/051703 19.04.2010<br />

(87) WO 2010/122482 2010/43 28.10.2010<br />

(30) 20.04.20<strong>09</strong> IT RM20<strong>09</strong>0180<br />

(54) PHARMAZEUTISCHE ZUSAMMENSET-<br />

ZUNGEN ZUR BEHANDLUNG VON NA-<br />

SENPOLYPEN<br />

PHARMACEUTICAL COMPOSITIONS FOR<br />

THE TREATMENT OF NASAL POLYPOSIS<br />

COMPOSITIONS PHARMACEUTIQUES<br />

POUR LE TRAITEMENT D'UNE POLY-<br />

POSE NASALE<br />

(71) D.M.G. Italia Srl, Via Laurentina Km 26,700,<br />

00040 Pomezia (RM), IT<br />

(72) MERCURI, Luigi, I-00040 Pomezia RM, IT<br />

(74) Sarpi, Maurizio, Studio Ferrario S.r.l. Via<br />

Collina, 36, 00187 Roma, IT<br />

A61K 31/047 → (51) A61K 31/00<br />

A61K 31/122 → (51) A61K 9/14<br />

A61K 31/13 → (51) A61K 9/00<br />

A61K 31/13 → (51) A61K 31/00<br />

A61K 31/137 → (51) A61K 9/51<br />

(51) A61K 31/155 (11) 2 421 521 A1*<br />

A61K 31/433 A61K 9/00<br />

A61P 17/10 A61P 17/00<br />

(25) En (26) En<br />

(21) 10715466.8 (22) 23.04.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) US 2010/032186 23.04.2010<br />

(87) WO 2010/124175 2010/43 28.10.2010<br />

(30) 24.04.20<strong>09</strong> US 172526 P<br />

(54) STABILE TOPISCHE ZUSAMMENSETZUN-<br />

GEN FÜR 1,2,4-THIADIAZOL-DERIVATE<br />

STABLE TOPICAL COMPOSITIONS FOR<br />

1,2,4-THIADIAZOLE DERIVATIVES<br />

COMPOSITIONS TOPIQUES STABLES<br />

POUR DES DÉRIVÉS DE 1,2,4-THIADIA-<br />

ZOLE<br />

(71) Janssen Pharmaceuticals, Inc., 1125<br />

Trenton-Harbourton Road, Titusville, NJ<br />

08560, US<br />

(72) CUI, Chengji, Pennington NJ 08534, US<br />

NG, Shirley, Mei-King, Bridgewater NJ<br />

08807, US<br />

WONG, George, Belle Mead NJ 08502, US<br />

YUSUF, Mohammed, Hatfield NJ 19440, US<br />

ZHANG, Fa, Belle Mead NJ 08502, US<br />

(74) Kirsch, Susan Edith, Carpmaels & Ransford<br />

One Southampton Row, London WC1B 5HA,<br />

GB

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