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Fragment based drug design

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Screening<br />

Screening fragmentů proti proteinovým objektům<br />

(targets)<br />

Používají se následující techniky:<br />

(i) rtg. krystalografie (proteinová krystalografie)<br />

(ii) NMR spektroskopie (Water LOGSY)<br />

(iii) Isotermální titrační kalorimetrie<br />

(iv) Surface plasmon resonance<br />

(v) Nekovalentní hmotnostní spektroskopie (MS)

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