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Fragment based drug design

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Tradiční <strong>design</strong> léčiv<br />

• Tradiční recepty a náhodné objevy<br />

• Kombinatorní chemie, přírodní sloučeniny<br />

• Screening (ultra high-throuput screening,<br />

HTS), "hit" → "lead compound"<br />

• Knihovny sloučenin - řádově milion<br />

sloučenin<br />

ve farmceutických společnostech

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