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HIV associated CNS disease in the era of HAART - Virology Education

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Antiretroviral Treatment<br />

<strong>CNS</strong> Penetration-Effectiveness Scores<br />

1 0.5 0<br />

NRTIs Abacavir Emtricitab<strong>in</strong>e Didanos<strong>in</strong>e<br />

Zidovud<strong>in</strong>e Lamivud<strong>in</strong>e Ten<strong>of</strong>ovir<br />

Stavud<strong>in</strong>e Zalcitab<strong>in</strong>e<br />

NNRTIs Delavird<strong>in</strong>e<br />

Nevirap<strong>in</strong>e<br />

Efavirenz<br />

PIs Amprenavir-r Amprenavir Nelf<strong>in</strong>avir<br />

Ind<strong>in</strong>avir-r Atazanavir Ritonavir<br />

Lop<strong>in</strong>avir/r Atazanavir-r Saqu<strong>in</strong>avir<br />

Ind<strong>in</strong>avir Saqu<strong>in</strong>avir-r<br />

Tipranavir-r<br />

Fusion<br />

Inhibitors<br />

Enfuvirtide<br />

Letendre S, et al. 13th CROI, Denver, 2006, Abstract #74; Letendre S, et al. Arch Neurol. 2008;65:65-70.<br />

Presented at <strong>the</strong> 5th INTEREST workshop – 10 – 13 May 2010, Dar-es-Salaam, Tanzania<br />

1.0

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