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KRONÄ°K HEPATÄ°T B TEDAVÄ°SÄ°NDE LAMÄ°VUDÄ°N VE ... - Klimik

KRONÄ°K HEPATÄ°T B TEDAVÄ°SÄ°NDE LAMÄ°VUDÄ°N VE ... - Klimik

KRONÄ°K HEPATÄ°T B TEDAVÄ°SÄ°NDE LAMÄ°VUDÄ°N VE ... - Klimik

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TELBİVUDİN-1<br />

• Hücresel kinazlar tarafından aktive<br />

edilir<br />

• Timidinin 1-nükleozid analoğu<br />

• Aktif trifosfat formu, kendi doğal<br />

substratı timidin 5’-trifosfat ile<br />

rekabet ederek HBV DNA polimeraz<br />

aktivitesini inhibe eder

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