12/2010 - Državni zavod za intelektualno vlasništvo

3554 HR - Patenti - Hrvatski glasnik intelektualnog vlasništva 17, 2010, 12, 3477 – 3584Y je cijano, nitro, C 1 -C4-alkil, C 1 -C 4 -haloalkil, metoksi ili metiltio;p je 0 ili 1;R 1 je vodik, halogen, C 1 -C 4 -alkil ili C 1 -C 4 -haloalkil;R 2 je vodik, metil ili halogen;R 3 je vodik, metil ili etil;W je kisik ili sumpor.Patent sadrži još 11 patentnih zahtjeva.(51) MKP (10) HR P20100614 T1C07D 279/20 (2006.01)A61K 31/5415 (2006.01)A61P 25/28 (2006.01)(11) P20100614(46) 31.12.2010.(21) P20100614T (22) 12.11.2010.(86) PCT/GB20070 01103 28.03.2007.(96) EP 07732164.4 28.03.2007.(87) WO2007110627, 04.10.2007.(97) EP 2013191, 14.01.2009. 200903, En(97) EP 2013191, 18.08.2010. 201033, En(31) 786690 P (32) 29.03.2006.(33) US(54) SOLI 3,7-DIAMINO-10H-FENOTIAZINA I NJIHOVA UPORABA3,7-DIAMINO-10H-PHENOTHIAZINE SALTS AND THEIR USE(73) Wista Laboratories Ltd., 51 Ayer Rajah Crescent No. 07-01/02,139948 Singapore, SG(72) Claude Michel Wischik, WisTa Laboratories Ltd. Institute of MedicalSciences Forresterhill, Aberdeen AB25 2ZD, Scotland, GBJanet Elizabeth Rickard, WisTa Laboratories Ltd. Institute ofMedical Sciences Forresterhill, Aberdeen, AB25 2ZD, Scotland, GBCharles Robert Harrington, WisTa Laboratories Ltd. Institute ofMedical Sciences Forresterhill, Aberdeen, AB25 2ZD, Scotland, GBDavid Horsley, WisTa Laboratories Ltd. Institute of MedicalSciences Forresterhill, Aberdeen, AB25 2ZD, Scotland, GBJohn Mervyn David Storey, WisTa Laboratories Ltd. Department ofChemistry Meston Walk, Old Aberdeen, AB24 3UE, Scotland, GBColin Marshall, WisTa Laboratories Ltd. Department of ChemistryMeston Walk, Old Aberdeen, AB24 3UE, Scotland, GBJames Peter Sinclair, WisTa Laboratories Ltd. Department ofChemistry Meston Walk, Old Aberdeen, AB24 3UE, Scotland, GBThomas Craven Baddeley, WisTa Laboratories Ltd. Department ofChemistry Meston Walk, Old Aberdeen, AB24 3UE, Scotland, GB(74) CPZ - CENTAR ZA PATENTE d.d., Zagreb, HR(57) Spoj, naznačen time, da je odabran od spojeva sljedeće formule injihovih farmaceutski prihvatljivih soli, solvata i hidrata:PYRIMIDINE DERIVATIVES USED AS PI-3 KINASE INHIBITORS( 73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH(72) Matthew Burger, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USZhi-jie Ni, C/O NOVARTIS VACCINES AND DIAGNOSTICS INC.P.O. Box 8097, Emeryville, CA 94662-8097, USSabina Pecchi, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USGordana Atallah, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USSarah Bartulis, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USKelly Frazier, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USAaron Smith, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USJoelle Verhagen, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USYanchen Zhang, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USAllan Wagman, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USSimon Ng, C/O NOVARTIS VACCINES AND DIAGNOSTICS INC.P.O. Box 8097, Emeryville, CA 94662-8097, USKeith Pfister, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USDaniel Poon, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USAlicia Louie, C/O NOVARTIS VACCINES AND DIAGNOSTICS INC.P.O. Box 8097, Emeryville, CA 94662-8097, USTeresa Pick, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USPaul Barsanti, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USEdwin Iwanowicz, C/O NOVARTIS VACCINES ANDDIAGNOSTICS INC. P.O. Box 8097, Emeryville, CA 94662-8097,USWendy Fantl, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USThomas Hendrickson, C/O NOVARTIS VACCINES ANDDIAGNOSTICS INC. P.O. Box 8097, Emeryville, CA 94662-8097,USMark Knapp, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USHanne Meritt, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USCharles Voliva, C/O NOVARTIS VACCINES AND DIAGNOSTICSINC. P.O. Box 8097, Emeryville, CA 94662-8097, USMarion Wiesmann, C/O NOVARTIS VACCINES ANDDIAGNOSTICS INC. P.O. Box 8097, Emeryville, CA 94662-8097,USXiahua Xin, C/O NOVARTIS VACCINES AND DIAGNOSTICS INC.P.O. Box 8097, Emeryville, CA 94662-8097, US(74) CPZ - CENTAR ZA PATENTE d.d., Zagreb, HR(57) Spoj, naznačen time, da ima formulu I:gdje jesvaki od R 1 i R 9 neovisno odabran od -H, C 1-4 alkila, C 2-4 alkenila, ihalogeniranog C 1-4 alkila;svaki od R 3NA i R 3NB neovisno odabran od -H, C 1-4 alkila, C 2-4 alkenila, ihalogeniranog C 1-4 alkila;svaki od R 7NA i R 7NB neovisno odabran od -H, C 1-4 alkila, C 2-4 alkenila, ihalogeniranog C 1-4 alkila;svaki od HX 1 i HX 2 neovisno protična kiselina.Patent sadrži još 37 patentnih zahtjeva.(51) MKPC07D 401/04 (2006.01)(10) HR P20100603 T1C07D 401/14 (2006.01)C07D 405/12 (2006.01)C07D 405/14 (2006.01)C07D 417/12 (2006.01)A61K 31/506 (2006.01)A61P 35/00 (2006.01)(11) P20100603(46) 31.12.2010.(21) P20100603T (22) 09.11.2010.(86)(96)PCT/US20070 01708 22.01.2007.EP 07716906.8 22.01.2007.(87) WO2007084786, 26.07.2007.(97)(97)EP 1984350, 29.10.2008. 200844, EnEP 1984350, 18.08.2010. 201033, En(31) 760789 P (32) 20.01.2006.(33) US(54) DERIVATI PIRIMIDINA KOJI SE KORIS TE KAO INHIBITORI PI-3KINAZEili njegov stereoizomer, tautomer ili farmaceutski prihvatljiva sol, gdje Wje CR W ili N, gdje RWje odabran iz skupine koja sadrživodik,cijano,halogen,metil,trifluorometil,sulfonamid;R 1 je odabran iz skupine koja sadrživodik,cijano,nitro,halogen,supstituirani i nesupstituirani alkil,supstituirani i nesupstituirani alkenil,supstituirani i nesupstituirani alkinil,supstituirani i nesupstituirani aril,supstituirani i nesupstituirani heteroaril,ISSN 1847-3024