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European Patent Bulletin 2012/14 - European Patent Office

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(A61K) I.1(1)<br />

(30) 27.05.2009 US 181550 P<br />

(54) KOMBINATIONSTHERAPIE ZUR BEHAND-<br />

LUNG VON MULTIPLEM MYELOM MIT<br />

CEP-18770 UND BORTEZOMIB ODER<br />

MEPHALAN<br />

COMBINATION THERAPY FOR THE<br />

TREATMENT OF MULTIPLE MYELOMA<br />

USING CEP-18770 TOGETHER WITH<br />

BORTEZOMIB OR MEPHALAN<br />

THÉRAPIE D'ASSOCIATION POUR LE<br />

TRAITEMENT DU MYÉLOME MULTIPLE<br />

EN UTILISANT CEP-18770 CONJOINTE-<br />

MENT AVEC LE BORTÉZOMIB OU LE<br />

MELPHALAN<br />

(71) Cephalon, Inc., 41 Moores Road P.O. Box<br />

4011, Frazer, PA 19355, US<br />

(72) BERENSON, James, R., Beverly Hills CA<br />

90210, US<br />

(74) Hallybone, Huw George, Carpmaels &<br />

Ransford One Southampton Row, GB-<br />

London WC1B 5HA, GB<br />

(51) A61K 31/198 (11) 2 435 039 A2*<br />

A61K 31/202 A61P 35/00<br />

A61P 3/<strong>14</strong><br />

(25) En (26) En<br />

(21) 10726616.5 (22) 27.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) NL 2010/050319 27.05.2010<br />

(87) WO 2010/137979 2010/48 02.12.2010<br />

(88) <strong>14</strong>.04.2011<br />

(30) 27.05.2009 PCT/NL2009/050297<br />

(54) KOMBINATION EINER LEUCINQUELLE<br />

UND EINER UNGESÄTTIGTEN OMEGA-3-<br />

FETTSÄURENQUELLE FÜR DIE BEHAND-<br />

LUNG VON HYPERKALZÄMIE<br />

COMBINATION OF A LEUCINE SOURCE<br />

AND AN OMEGA-3 UNSATURATED FATTY<br />

ACID SOURCE FOR USE IN THE<br />

TREATMENT OF HYPERCALCAEMIA<br />

COMBINAISON D'UNE SOURCE DE<br />

LEUCINE ET D' UNE SOURCE D'ACIDE<br />

GRAS INSATURÉ OMEGA-3& xA; POUR<br />

LE TRAITEMENT DE L'HYPERCALCÉMIE<br />

(71) N.V. Nutricia, Eerste Stationsstraat 186,<br />

2712 HM Zoetermeer, NL<br />

(72) VAN NORREN, Klaske, NL-6871 LP Renkum,<br />

NL<br />

FABER, Joyce, NL-7471 RC Goor, NL<br />

VAN HELVOORT, Adrianus Lambertus Bertholdus,<br />

NL-6703 ED Wageningen, NL<br />

HAGEMAN, Robert Johan Joseph, NL-6705<br />

CT Wageningen, NL<br />

(74) Jansen, Cornelis Marinus, et al, VEREE-<br />

NIGDE Johan de Wittlaan 7, 2517 JR Den<br />

Haag, NL<br />

(51) A61K 31/20 (11) 2 435 040 A2*<br />

A61K 31/17<br />

(25) En (26) En<br />

(21) 10781280.2 (22) 28.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/036584 28.05.2010<br />

(87) WO 2010/138820 2010/48 02.12.2010<br />

(88) 27.01.2011<br />

(30) 28.05.2009 US 181920 P<br />

(54) N,N-DIARYLHARNSÄURE-VERBINDUN-<br />

GEN UND N,N'-DIARYLTHIOHARNSÄU-<br />

RE-VERBINDUNGEN ALS TRANSLATI-<br />

ONSSTARTHEMMER<br />

N,N-DIARYLUREA COMPOUNDS AND<br />

N,N'-DIARYLTHIOUREA COMPOUNDS AS<br />

INHIBITORS OF TRANSLATION<br />

INITIATION<br />

COMPOSÉS DE N,N'-DIARYLURÉE ET DE<br />

N,N'-DIARYLTHIOURÉE UTILISÉS EN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

TANT QU'INHIBITEURS DE L'INITIATION<br />

DE LA TRADUCTION<br />

(71) President and Fellows of Harvard College, 17<br />

Quincy Street, Cambridge, MA 02138, US<br />

(72) AKTAS, Huseyin, Newton, MA 02465, US<br />

HALPERIN, Jose, A., Brookline, MA 02446,<br />

US<br />

CHOREV, Michael, Chestnut Hill, MA 02467,<br />

US<br />

(74) Tetaz, Franck Claude Edouard, et al, Cabinet<br />

Regimbeau 139, rue Vendôme, F-69477<br />

Lyon Cedex 06, FR<br />

A61K 31/202 → (51) A61K 31/198<br />

A61K 31/21 → (51) C07D 213/82<br />

(51) A61K 31/282 (11) 2 435 041 A1*<br />

A61K 31/337 A61K 31/4745<br />

A61K 31/513 A61K 31/519<br />

A61K 31/704 A61K 31/7068<br />

A61K 33/24 A61K 45/06<br />

A61K 31/4412 A61K 31/4965<br />

A61K 31/506<br />

(25) En (26) En<br />

(21) 10723967.5 (22) 21.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/057027 21.05.2010<br />

(87) WO 2010/136394 2010/48 02.12.2010<br />

(30) 26.05.2009 EP 09161111<br />

(54) THERAPEUTISCHE KOMBINATION AUS<br />

EINEM PLK1-HEMMER UND EINEM AN-<br />

TINEOPLASTIKUM<br />

THERAPEUTIC COMBINATION<br />

COMPRISING A PLK1 INHIBITOR AND AN<br />

ANTINEOPLASTIC AGENT<br />

COMBINAISON THÉRAPEUTIQUE<br />

COMPRENANT UN INHIBITEUR DE PLK1<br />

ET UN AGENT ANTINÉOPLASIQUE<br />

(71) Nerviano Medical Sciences S.r.l., 11 Viale<br />

Pasteur, 10 P.O. Box 11, 200<strong>14</strong> Nerviano<br />

(MI), IT<br />

(72) VALSASINA, Barbara, I-20131 Milan, IT<br />

BERIA, Italo, I-200<strong>14</strong> Nerviano (MI), IT<br />

CIAVOLELLA, Antonella, I-22020 Bizzarone<br />

(CO), IT<br />

BALLINARI, Dario, I-20097 San Donato Milanese<br />

(MI), IT<br />

PESENTI, Enrico, I-20015 Parabiago (MI), IT<br />

MOLL, Juergen, I-22070 Appiano Gentile<br />

(CO), IT<br />

A61K 31/33 → (51) C07D 211/16<br />

A61K 31/335 → (51) A01N 43/26<br />

A61K 31/337 → (51) A61K 31/282<br />

A61K 31/343 → (51) A61K 31/135<br />

A61K 31/343 → (51) C07C 205/43<br />

A61K 31/35 → (51) C07D 311/78<br />

A61K 31/352 → (51) C07D 311/78<br />

A61K 31/353 → (51) A23L 1/30<br />

A61K 31/353 → (51) C08J 3/075<br />

A61K 31/375 → (51) A23L 1/30<br />

A61K 31/40 → (51) A01N 43/36<br />

A61K 31/40 → (51) A61K 9/12<br />

40<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>14</strong>/<strong>2012</strong>) 04.04.<strong>2012</strong><br />

(51) A61K 31/403 (11) 2 435 042 A1*<br />

A61K 9/50 A61K 9/16<br />

A61K 9/00<br />

(25) Fr (26) Fr<br />

(21) 10728845.8 (22) 28.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) FR 2010/051039 28.05.2010<br />

(87) WO 2010/136740 2010/48 02.12.2010<br />

(30) 29.05.2009 FR 0953607<br />

29.05.2009 US 182533 P<br />

(54) VERFAHREN ZUR HERSTELLUNG VON<br />

HOHLEN TEILCHEN UND SEINE VER-<br />

WENDUNG<br />

METHOD FOR PREPARING HOLLOW<br />

PARTICLES, AND USES THEREOF<br />

PROCEDE DE PREPARATION DE PARTI-<br />

CULES CREUSES ET LEURS APPLICA-<br />

TIONS<br />

(71) Flamel Technologies, 33 avenue du Docteur<br />

Georges Lévy, 69200 Vénissieux, FR<br />

(72) CASTAN, Catherine, F-69530 Orlienas, FR<br />

CAISSE, Philippe, F-69720 St Bonnet De<br />

Mure, FR<br />

(74) Cabinet Plasseraud, 235 Cours Lafayette,<br />

69006 Lyon, FR<br />

(51) A61K 31/4045 (11) 2 435 043 A1*<br />

A61P 25/16 A61P 25/28<br />

A61P 9/10<br />

(25) En (26) En<br />

(21) 10724371.9 (22) 27.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/057364 27.05.2010<br />

(87) WO 2010/136546 2010/48 02.12.2010<br />

(30) 27.05.2009 EP 09161292<br />

(54) 3-ALKYL-5-FLUORINDOLDERIVATE ALS<br />

MYELOPEROXIDASEHEMMER<br />

3-ALKYL-5-FLUOROINDOLE DERI-<br />

VATIVES AS MYELOPEROXIDASE INHI-<br />

BITORS<br />

DÉRIVÉS DE 3-ALKYL-5-FLUOROINDOLE<br />

EN TANT QU'INHIBITEURS DE PEROXY-<br />

DASE LEUCOCYTAIRE<br />

(71) Université Libre de Bruxelles, Avenue F.D.<br />

Roosevelt, C.P. 50, 1050 Bruxelles, BE<br />

(72) SOUBHYE, Jalal, B-1000 Bruxelles, BE<br />

DUFRASNE, François, B-1180 Bruxelles, BE<br />

VAN ANTWERPEN, Pierre, B-1090 Bruxelles,<br />

BE<br />

(74) Pecher, Nicolas, Pecher Consultants SPRL<br />

Centre Monnet - Avenue Jean Monnet, 1,<br />

1348 Louvain-la-Neuve, BE<br />

A61K 31/4164 → (51) C07D 233/64<br />

A61K 31/4178 → (51) C07D 413/10<br />

A61K 31/4184 → (51) C07D 401/<strong>14</strong><br />

A61K 31/4184 → (51) C07D 403/<strong>14</strong><br />

A61K 31/4245 → (51) A61K 45/06<br />

A61K 31/433 → (51) C07D 513/04<br />

A61K 31/435 → (51) C07D 213/82<br />

(51) A61K 31/437 (11) 2 435 044 A1*<br />

A61K 31/15 A61P 25/20<br />

(25) En (26) En<br />

(21) 10727910.1 (22) 25.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) IB 2010/052308 25.05.2010

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