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European Patent Bulletin 2012/30 - European Patent Office

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(A01N) I.1(1)<br />

(51) A01N 43/00 (11) 2 477 492 A1*<br />

A61K 31/55<br />

(25) En (26) En<br />

(21) 10817928.4 (22) 17.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/049358 17.09.2010<br />

(87) WO 2011/035174 2011/12 24.03.2011<br />

(<strong>30</strong>) 17.09.2009 US 243378 P<br />

(54) SUBSTITUIERTE HETEROARYLAMIN-<br />

CARBOXAMID-ANALOGA ALS NEGATIVE<br />

ALLOSTERISCHE MGLUR5-MODULATO-<br />

REN SOWIE VERFAHREN ZU IHRER HER-<br />

STELLUNG UND VERWENDUNG<br />

SUBSTITUTED HETEROARYLAMINE<br />

CARBOXAMIDE ANALOGS AS MGLUR5<br />

NEGATIVE ALLOSTERIC MODULATORS<br />

AND METHODS OF MAKING AND USING<br />

THE SAME<br />

ANALOGUES D'HÉTÉROARYLAMINE<br />

CARBOXAMIDE SUBSTITUÉ UTILISÉS<br />

COMME MODULATEURS ALLOSTÉRI-<br />

QUES NÉGATIFS DE MGLUR5, LEURS<br />

PROCÉDÉS DE PRÉPARATION ET D'UTI-<br />

LISATION<br />

(71) Vanderbilt University, <strong>Office</strong> Of Technology<br />

Transfer <strong>30</strong>5 Kirkland Hall, Nashville,<br />

Tennessee 37240, US<br />

(72) CONN, P. Jeffrey, Brentwood, TN 37027, US<br />

LINDSLEY, Craig W., Brentwood, TN 37027,<br />

US<br />

EMMITTE, Kyle A., Spring Hill, TN 37174,<br />

US<br />

WEAVER, Charles David, Franklin, TN 37067,<br />

US<br />

RODRIGUEZ, Alice, L., Nashville, TN 37209,<br />

US<br />

FELTS, Andrew S., Nashville, TN 37204, US<br />

JONES, Carrie K., Nashville, TN 37221, US<br />

BATES, Brittney S., Nashville, TN 37215, US<br />

(74) Warner, James Alexander, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

(51) A01N 43/14 (11) 2 477 493 A1*<br />

(25) En (26) En<br />

(21) 10817824.5 (22) 16.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/049113 16.09.2010<br />

(87) WO 2011/035019 2011/12 24.03.2011<br />

(<strong>30</strong>) 16.09.2009 US 243104 P<br />

(54) NEUE TRIZYKLISCHE PROTEINKINASE-<br />

MODULATOREN<br />

NOVEL TRICYCLIC PROTEIN KINASE<br />

MODULATORS<br />

MODULATEURS TRICYCLIQUES INÉDITS<br />

DES PROTÉINES KINASES<br />

(71) Cylene Pharmaceuticals, Inc., 5820 Nancy<br />

Ridge Drive, Suite 200, San Diego, CA<br />

92121, US<br />

(72) HADDACH, Mustapha, San Diego California<br />

92127, US<br />

PIERRE, Fabrice, La Jolla California 92037,<br />

US<br />

(74) Keen, Celia Mary, J A Kemp 14 South Square<br />

Gray's Inn, London WC1R 5JJ, GB<br />

(51) A01N 43/16 (11) 2 477 494 A1*<br />

A61K 31/35<br />

(25) En (26) En<br />

(21) 10817681.9 (22) 09.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/048227 09.09.2010<br />

(87) WO 2011/034772 2011/12 24.03.2011<br />

(<strong>30</strong>) 16.09.2009 US 24<strong>30</strong>36 P<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) NA/K-ATPASE-LIGANDEN, OUABAIN-AN-<br />

TAGONISTEN, ASSAYS DAMIT UND VER-<br />

WENDUNGEN DAVON<br />

NA/K-ATPASE LIGANDS, OUABAIN<br />

ANTAGONISTS, ASSAYS AND USES<br />

THEREOF<br />

LIGANDS DE NA/K-ATPASE, ANTAGO-<br />

NISTES OUABAÏNES, LEURS ESSAIS ET<br />

LEURS UTILISATIONS<br />

(71) The University of Toledo, A University<br />

Instrumentality of the State of Ohio 2801 W.<br />

Bancroft Street, Toledo, OH 43606, US<br />

(72) XIE, Zi-jian, Saline MI 48176, US<br />

SHAPIRO, Joseph, I., Toledo OH 43617, US<br />

SI, Shuyi, Beijing 100052, CN<br />

ZHANG, Zhongbing, Beijing 102600, CN<br />

(74) Turner, Craig Robert, A.A. Thornton & Co.<br />

235 High Holborn, London WC1V 7LE, GB<br />

A01N 43/<strong>30</strong> → (51) A01N 35/06<br />

A01N 43/40 → (51) A01N 25/00<br />

A01N 43/40 → (51) A01N 25/<strong>30</strong><br />

A01N 43/40 → (51) A01N 35/06<br />

A01N 43/40 → (51) A01N 43/90<br />

(51) A01N 43/42 (11) 2 477 495 A1*<br />

A61K 31/44<br />

(25) En (26) En<br />

(21) 10817825.2 (22) 16.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/049116 16.09.2010<br />

(87) WO 2011/035022 2011/12 24.03.2011<br />

(<strong>30</strong>) 16.09.2009 US 243107 P<br />

(54) TRIZYKLISCHE VERBINDUNGEN UND<br />

PHARMAZEUTISCHE VERWENDUNGEN<br />

DAVON<br />

TRICYCLIC COMPOUNDS AND PHARMA-<br />

CEUTICAL USES THEREOF<br />

COMPOSÉS TRICYCLIQUES ET LEURS<br />

UTILISATIONS PHARMACEUTIQUES<br />

(71) Cylene Pharmaceuticals, Inc., 5820 Nancy<br />

Ridge Drive, Suite 200, San Diego, CA<br />

92121, US<br />

(72) HADDACH, Mustapha, San Diego California<br />

92127, US<br />

PIERRE, Fabrice, La Jolla California 92037,<br />

US<br />

(74) Keen, Celia Mary, J A Kemp 14 South Square<br />

Gray's Inn, London WC1R 5JJ, GB<br />

A01N 43/50 → (51) A01N 43/90<br />

A01N 43/54 → (51) A01N 25/00<br />

A01N 43/54 → (51) A01N 35/06<br />

A01N 43/54 → (51) A01N 43/90<br />

A01N 43/56 → (51) A01N 25/00<br />

A01N 43/56 → (51) A01N 43/90<br />

(51) A01N 43/58 (11) 2 477 496 A1*<br />

A61K 31/50 A61K 31/495<br />

(25) En (26) En<br />

(21) 10817865.8 (22) 17.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/049199 17.09.2010<br />

(87) WO 2011/035077 2011/12 24.03.2011<br />

(<strong>30</strong>) 18.09.2009 US 243549 P<br />

20<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>30</strong>/<strong>2012</strong>) 25.07.<strong>2012</strong><br />

(54) NEUARTIGE VERBINDUNGEN UND IHRE<br />

THERAPEUTISCHE VERWENDUNG ZUR<br />

PROTEINKINASEHEMMUNG<br />

NOVEL COMPOUNDS AND THERAPEUTIC<br />

USE THEREOF FOR PROTEIN KINASE<br />

INHIBITION<br />

NOUVEAUX COMPOSÉS ET LEUR UTILI-<br />

SATION THÉRAPEUTIQUE POUR UNE<br />

INHIBITION DE PROTÉINE KINASE<br />

(71) Wu, Zhanggui, 190 Longwood St. Apt. 58,<br />

Brookline, Massachusetts 02446, US<br />

(72) Wu, Zhanggui, Brookline, Massachusetts<br />

02446, US<br />

(74) Krauss, Jan, Boehmert & Boehmert Pettenkoferstrasse<br />

20-22, 80336 München, DE<br />

A01N 43/653 → (51) A01N 25/00<br />

A01N 43/653 → (51) A01N 43/90<br />

A01N 43/88 → (51) A01N 43/90<br />

(51) A01N 43/90 (11) 2 477 497 A2*<br />

A01N 47/38 A01N 47/24<br />

A01N 47/12 A01N 45/02<br />

A01N 43/88 A01N 43/653<br />

A01N 43/56 A01N 43/54<br />

A01N 43/50 A01N 43/40<br />

A01N 37/50 A01N 37/36<br />

A01N 37/24 A01N 37/20<br />

(25) En (26) En<br />

(21) 10752727.7 (22) 02.09.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/005395 02.09.2010<br />

(87) WO 2011/029551 2011/11 17.03.2011<br />

(88) 18.08.2011<br />

(<strong>30</strong>) 14.09.2009 EP 09170209<br />

14.09.2009 US 242076 P<br />

17.09.2009 EP 09176213<br />

(54) SYNERGISTISCHE FUNGIZIDKOMBINA-<br />

TIONEN MIT EINEM DITHIINO-TETRA-<br />

CARBOXAMID-FUNGIZID<br />

SYNERGISTIC FUNGICIDAL COMBI-<br />

NATIONS CONTAINING A DITHIINO-<br />

TETRACARBOXAMIDE FUNGICIDE<br />

COMBINAISONS FONGICIDES SYNERGI-<br />

QUES CONTENANT UN FUNGICIDE DU<br />

TYPE DITHIINO-CARBOXAMIDE<br />

(71) Bayer CropScience AG, Alfred-Nobel-Straße<br />

50, 40789 Monheim, DE<br />

(72) SEITZ, Thomas, 40764 Langenfeld, DE<br />

WACHENDORFF-NEUMANN, Ulrike, 56566<br />

Neuwied, DE<br />

DAHMEN, Peter, 41470 Neuss, DE<br />

A01N 45/02 → (51) A01N 43/90<br />

A01N 47/02 → (51) A01N 25/00<br />

A01N 47/12 → (51) A01N 43/90<br />

A01N 47/24 → (51) A01N 25/00<br />

A01N 47/24 → (51) A01N 43/90<br />

A01N 47/38 → (51) A01N 43/90<br />

A01N 47/40 → (51) A01N 25/<strong>30</strong><br />

A01N 51/00 → (51) A01N 25/00<br />

A01N 51/00 → (51) A01N 25/<strong>30</strong><br />

A01N 55/00 → (51) A01N 25/10<br />

(51) A01N 57/00 (11) 2 477 498 A1*<br />

C07C 403/00<br />

(25) En (26) En

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