hrvatski glasnik intelektualnog vlasništva 05/2005 - Državni zavod ...

1980 HR - Patenti. - Hrvatski glasnik intelektualnog vlasništva 12, 2005, 5, 1897 – 2089
(31) 100 40 174.0 (32) 17. 08.2000. (33) DE
(54) UPOTREBA TRIAZINTRION SULFONA ZA SUZBIJANJE
KOKCIDIOZA
USE OF TRIAZINETRIONE SULFONES FOR COMBATING
COCCIDIOSIS
(71) Bayer Aktiengesellschaft, 51368 Leverkusen, DE
(72) Gisela Greif, Marienhöhe 15, 53424 Remagen, DE
Iris Heep, Grüner Weg 7a, 50859 Köln, DE
Hans-Christian Mundt, Lessingstrasse 30, 40699 Erkrath, DE
(74) CPZ - CENTAR ZA PATENTE d.d., ZAGREB, HR
(57) Izum se odnosi na upotrebu posebnih derivata triazintriona za
suzbijanje kokcidioza kod životinja, posebno svinja.
(51) Int.Cl. C 07 D 265/02 7 (10) HR P20030148 A2
C 07 D 307/88
C 07 D 413/12
A 61 K 31/536
A 61 K 31/365
A 61 P 29/00
(21) P20030148A (22) 28. 02.2003.
(43) 31. 10.2005.
(86) PCT/EP01/08501; 23. 07.2001.
(87) WO02/10143; 07. 02.2002.
(31) 100 38 639.3 (32) 28. 07.2000. (33) DE
(54) NESTEROIDNE SUPSTANCE, ANTIUPALNOG DJELOVANJA
NON STEROIDAL INFLAMMATION INHIBITORS
(71) Schering Aktiengesellschaft, Müllerstrasse 178, 13353 Berlin, DE
(72) Stefan Jaroch, Schlueterstr. 65, 10625 Berlin, DE
Manfred Lehmann, Lutherstrasse 13, 12305 Berlin, DE
Norbert Schmees, Horber Str. 3, 13469 Berlin, DE
Bernd Buchmann, Erdmannstrasse 44, 16540 Hohen Neuendorf,
DE
Hartmut Rehwinkel, Glasower Str. 41, 12051 Berlin, DE
Peter Droescher, Lessingstrasse 7, 99425 Weimar, DE
Werner Skuballa, Mattersburger Weg 12, 13465 Berlin, DE
Konrad Krolikiewicz, Ehrenpreisweg 33, 12357 Berlin, DE
Hartwig Hennekes, Handjerystr. 16, 12159 Berlin, DE
Heike Schaecke, Gartenstr. 105, 10115 Berlin, DE
Arndt Schottelius, Schlossstr. 32, 14059 Berlin, DE
(74) Dragutin Sikirić, Zagreb, HR
(57) Predočeni izum se odnosi na spojeve opće formule (I),
kao nesteroidne supstance antiupalnog djelovanja, kao i postupke za
njihovo spravljanje i odabrane spojeve.
(51) Int.Cl. C 07 D 277/06 7 (10) HR P20031014 A2
A 61 K 31/425
C 07 D 417/12
C 07 D 403/12
C 07 D 207/16
A 61 P 31/18
(21) P20031014A (22) 08. 12.2003.
(43) 31. 10.2005.
(86) PCT/US02/18548; 11. 06.2002.
(87) WO02/100845; 19. 12.2002.
(31) 60/297,460 (32) 11. 06.2001. (33) US
60/297,729 12. 06.2001. US
(54) INHIBITORI HIV PROTEAZA, SPOJEVI KOJI SADRŽE ISTE,
NJIHOVA FARMACEUTSKA UPORABA I MATERIJALI ZA
NJIHOVU SINTEZU
HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING
THE SAME, THEIR PHARMACEUTICAL USES AND MATERIALS
FOR THEIR SYNTHESIS
(71) Agouron Pharmaceuticals Inc., 10350 North Torrey Pines Road, La
Jolla, CA 92037, US
(72) Stacie S. Canon-Koch, 5940 La Jolla Messa Drive, La Jolla, CA
92137, US
Therese N. Alexander, 6557 Thornwood Street, San Diego, CA
92111, US
Mark Barvian, 1225 Olivia Avenue, Ann Arbor, MI 48104, US
Gary Bolton, 4800 Hillway Ct., Ann Arbor, MI 48105, US
Fredrick E. Boyer, 482 Pleasant Ridge Drive, Canton Township, MI
48188, US
Benjamin J. Burke, 5761 Campanile Way, San Diego, CA 92115,
US
Tod Holler, 2381 Placid Way, Ann Arbor, MI 48105, US
Tanya M. Jewell, 12604 Torrey Bluff Dr. #400, San Diego, CA
92130, US
Vara Prasad Josyula, 3129 Fawn Meadow Court, Ann Arbor, MI
48105, US
David, J. Kucera, 14099 Recuerdo Drive, Del Mar, CA 92014, US
Maria, A. Linton, 11320 Red Cedar Drive, San Diego, CA 92131,
US
Jeff Machak, 12980 Easton Court, Shelby Township, MI 48315, US
Lennert J. Mitchell, 520 N. Woodlawn Avenue, Chula Vista, CA
91910, US
Sean T. Murphy, 7716 Dover Drive, Ypsilanti, MI 48197, US
Siegfried H. Reich, 311 Glenmont Drive, Solana Beach, CA 92075,
US
Donald J. Skalitzky, 4269 Taos Drive, San Diego, CA 92117, US
John H. Tatlock, 13153 Dressage Lane, San Diego, CA 92130, US
Michael D. Varney, 738 Barbara Avenue, Solana Beach, CA 92075,
US
Scott C. Virgil, 3950 Mahaila Avenue, Apt. S23, San Diego, CA
92122, US
Stephen E. Webber, 3531 Millikan Avenue, San Diego, CA 92122,
US
Stephen T. Worland, 727 Hoska Drive, Del Mar, CA 92014, US
Michael Melnick, 3613 Weeburn Court, Ann Arbor, MI 48108, US
(74) Hraste & Partneri odvjetničko društvo, Zagreb, HR
(57)
Dokazano je da spojevi formule (I) u kojoj su varijable formule kao što je
ovdje definirano, povoljno inhibiraju ili blokiraju biološku aktivnost HIV
proteaze. Ovi spojevi, baš kao i farmaceutski pripravci koji sadrže ove
spojeve, su korisni u liječenju pacijenata ili domaćina zaraženih HIV
virusom. Opisuju se i intermedijeri i sintetski postupci za pripremu
ovakvih spojeva.
(51) Int.Cl. C 07 D 277/06 7 (10) HR P20031015 A2
A 61 K 31/426
C 07 D 401/12
C 07 D 417/12
C 07 D 207/16
C 07 D 265/06
C 07 D 211/60
A 61 P 31/18
(21) P20031015A (22) 08. 12.2003.
(43) 31. 10.2005.
(86) PCT/US02/18717; 11. 06.2002.
(87) WO02/100844; 19. 12.2002.
(31) 60/297,460 (32) 11. 06.2001. (33) US
60/297,729 12. 06.2001. US
(54) INHIBITORI HIV PROTEAZE, SMJESE KOJE IH SADRŽE,
NJIHOVE FARMACEUTSKE PRIMJENE I MATERIJALI ZA
NJIHOVU SINTEZU
HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING
THE SAME, THEIR PHARMACEUTICAL USES AND MATERIALS
FOR THEIR SYNTHESIS
(71) Agouron Pharmaceuticals Inc., 10350 North Torrey Pines Road, La
Jolla, CA 92037, US
(72) Stacie S. Canon-Koch, 5940 La Jolla Messa Drive, La Jolla, CA
92137, US
Therese N. Alexander, 6557 Thornwood Street, San Diego, CA
92111, US
Mark Barvian, 1225 Olivia Avenue, Ann Arbor, MI 48104, US
Gary Bolton, 4800 Hillway Ct., Ann Arbor, MI 48105, US
Fredrick E. Boyer, 482 Pleasant Ridge Drive, Canton Township, MI
48188, US
Benjamin J. Burke, 5761 Campanile Way, San Diego, CA 92115,
US
Tod Holler, 2381 Placid Way, Ann Arbor, MI 48105, US
Tanya M. Jewell, 12604 Torrey Bluff Dr. #400, San Diego, CA
92130, US
Vara Prasad Josyula, 3129 Fawn Meadow Court, Ann Arbor, MI
48105, US
David, J. Kucera, 14099 Recuerdo Drive, Del Mar, CA 92014, US
Maria, A. Linton, 11320 Red Cedar Drive, San Diego, CA 92131,
US
Jeff Machak, 12980 Easton Court, Shelby Township, MI 48315, US
Lennert J. Mitchell, 520 N. Woodlawn Avenue, Chula Vista, CA
91910, US
Sean T. Murphy, 7716 Dover Drive, Ypsilanti, MI 48197, US
Siegfried H. Reich, 311 Glenmont Drive, Solana Beach, CA 92075,
US
Donald J. Skalitzky, 4269 Taos Drive, San Diego, CA 92117, US
John H. Tatlock, 13153 Dressage Lane, San Diego, CA 92130, US
Michael D. Varney, 738 Barbara Avenue, Solana Beach, CA 92075,
US
ISSN 1331-2030