PCT/2001/3 : PCT Gazette, Weekly Issue No. 3, 2001 - WIPO

03/2001
18 Jan/jan 2001 PCT Gazette - Section I - Gazette du PCT 939
MZ NO NZ PL PT RO RU SD SE SG SI SK
SL TJ TM TR TT TZ UA UG UZ VN YU ZA
ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 209/88, 303/36, 307/91, 333/76,
301/24, C07C 303/40, 311/08, 311/13,
A61K 31/403, A61P 3/06, 3/10
(11) WO 01/04092 (13) A1
(21) PCT/JP00/04015
(22) 20 Jun/juin 2000 (20.06.2000)
(25) ja (26) ja
(30) 11/195519 9 Jul/juil 1999 JP
(09.07.1999)
(43) 18 Jan/jan 2001 (18.01.2001)
(54) PROCESS FOR THE PREPARATION
OF TRICYCLIC AMINO ALCOHOL
DERIVATIVES
PROCEDE DE PREPARATION DE DE-
RIVES D’ALCOOLS AMINES TRICY-
CLIQUES
(71) ASAHI KASEI KOGYO KABUSHIKI
KAISHA [JP/JP]; 2-6, Dojimahama
1-chome, Kita-ku, Osaka-shi, Osaka
530-8205 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) MIYOSHI, Shiro [JP/JP]; 843-8,
Gokanjima, Fuji-shi, Shizuoka 416-0946
(JP). MATSUBARA, Koki [JP/JP]; Asahi
Kasei Taishi-ryo 226, 140-1, Nakamaru,
Fuji-shi, Shizuoka 416-0933 (JP).
(74) HIRAKI, Yusuke; Toranomon No.5 Mori
Building Third Floor, 17-1, Toranomon
1-chome, Minato-ku, Tokyo 105-0001 (JP).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 211/00
(11) WO 01/04093
(21) PCT/GB00/02698
(13) A2
(22) 13 Jul/juil 2000 (13.07.2000)
(25) en (26) en
(30) 9916392.5 13 Jul/juil 1999
(13.07.1999)
GB
(43) 18 Jan/jan 2001 (18.01.2001)
(54) NOVEL PROCESS
NOUVEAU PROCEDE
(71) SMITHKLINE BEECHAM PLC
[GB/GB]; New Horizons Court, Brentford,
Middlesex TW8 9EP (GB).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) JONES, David, Alan [GB/GB];
SmithKline Beecham Pharmaceuticals, Old
Powder Mills, Near Leigh, Tonbridge, Kent
TN11 9AN (GB).
(74) WEST, Vivien; SmithKline Beecham, Corporate
Intellectual Property, Two New Horizons
Court, Brentford, Middlesex TW8 9EP
(GB).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 221/16
(11) WO 01/04094
(21) PCT/JP00/04525
(13) A1
(22) 6 Jul/juil 2000 (06.07.2000)
(25) ja (26) ja
(30) 11/195430 9 Jul/juil 1999
(09.07.1999)
JP
(43) 18 Jan/jan 2001 (18.01.2001)
(54) PROCESSES FOR THE PREPARATION
OF IPIDACRINE OR IPIDACRINE HY-
DROCHLORIDE HYDRATE
PROCEDES DE PREPARATION D’IPI-
DACRINE OU D’HYDROCHLORURE
D’IPIDACRINE HYDRATE
(71) NIKKEN CHEMICALS CO., LTD.
[JP/JP]; 4-14, Tsukiji 5-chome, Chuo-ku,
Tokyo 104-0045 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) OMORI, Hiromasa [JP/JP]; Omiya
Research Laboratory, Nikken Chemicals
Co., Ltd., 346, Kitabukuro-cho 1-chome,
Omiya-shi, Saitama 330-0835 (JP).
(74) ISHIDA, Takashi et al. / etc.; A. Aoki,
Ishida & Associates, Toranomon 37 Mori
Bldg., 5-1, Toranomon 3-chome, Minato-ku,
Tokyo 105-8423 (JP).
(81) CA RU US.
(84) EP (AT BE CH CY DE DK ES FI FR GB GR
IE IT LU MC NL PT SE).
(51) 7 C07D 231/00
(11) WO 01/04095
(21) PCT/EP00/05857
(13) A2
(22) 23 Jun/juin 2000 (23.06.2000)
(25) de (26) de
(30) 199 31 881.6 9 Jul/juil 1999
(09.07.1999)
DE
(43) 18 Jan/jan 2001 (18.01.2001)
(54) e-α’-SUBSTITUTED N-ALKYL-3-
ALKENYLBENZOYL-PYRA-
ZOL-DERIVATIVES
DERIVES DE N-ALKYL-3-ALCENYL-
BENZOYLPYRAZOLES A SUBSTITU-
TION $G(A)-α’
(71) BASF AKTIENGESELLSCHAFT
[DE/DE]; D-67056 Ludwigshafen (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) NEIDLEIN, Ulf [DE/DE]; Brahmsstr.
3, D-68165 Mannheim (DE). GÖTZ, Norbert
[DE/DE]; Schöfferstr. 25, D-67547
Worms (DE). BAUMANN, Ernest [DE/DE];
Falkenstr. 6a, D-67373 Dudenhofen (DE).
VON DEYN, Wolfgang [DE/DE]; An der
Bleiche 24, D-67435 Neustadt (DE). KUDIS,
Steffen [DE/DE]; Spelzenstr. 10, D-68167
Mannheim (DE). GÖTZ, Roland [DE/DE];
Langebrücker Str. 25, D-68809 Neulussheim
(DE). LANGEMANN, Klaus [DE/DE];
Goldbergstr. 18, D-67551 Worms (DE).
MAYER, Guido [DE/DE]; Gutleuthausstr.
8, D-67433 Neustadt (DE). MISSLITZ, Ulf
[DE/DE]; Mandelring 74, D-67433 Neustadt
(DE). WITSCHEL, Matthias [DE/DE];
Wittelsbachstr. 81, D-67061 Ludwigshafen
(DE). OTTEN, Martina [DE/DE]; Gunterstr.
28, D-67069 Ludwigshafen (DE).
WESTPHALEN, Karl-Otto [DE/DE]; Zum
Pfauenturm 17, D-67346 Speyer (DE). WAL-
TER, Helmut [DE/DE]; Grünstadter Str. 82,
D-67283 Obrigheim (DE).
(74) BASF AKTIENGESELLSCHAFT;
D-67056 Ludwigshafen (DE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 231/00
(11) WO 01/04096
(21) PCT/EP00/05860
(13) A2
(22) 23 Jun/juin 2000 (23.06.2000)
(25) de (26) de
(30) 199 31 863.8 9 Jul/juil 1999
(09.07.1999)
DE
(43) 18 Jan/jan 2001 (18.01.2001)
(54) N-CYCLOALKYL-3-ALKENYLBEN-
ZOYL-PYRAZOLE DERIVATIVES
DERIVES DE N-CYCLOALKYL-3-AL-
CENYLBENZOYLPYRAZOLES
(71) BASF AKTIENGESELLSCHAFT
[DE/DE]; D-67056 Ludwigshafen (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) NEIDLEIN, Ulf [DE/DE];
Brahmsstrasse 3, D-68165 Mannheim (DE).
GÖTZ, Norbert [DE/DE]; Schöfferstrasse
25, D-67547 Worms (DE). BAUMANN,
Ernst [DE/DE]; Falkenstrasse 6a,
D-67373 Dudenhofen (DE). VON DEYN,
Wolfgang [DE/DE]; An der Bleiche
24, D-67435 Neustadt (DE). KUDIS,
Steffen [DE/DE]; Spelzenstrasse 10,
D-68167 Mannheim (DE). GÖTZ, Roland