全文 [3.9MB] - 放射線医学総合研究所
全文 [3.9MB] - 放射線医学総合研究所
全文 [3.9MB] - 放射線医学総合研究所
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放 射 線 医 学 総 合 研 究 所 平 成 23 年 度 資 料 集<br />
2. Toshimitsu Okamura, Tatsuya Kikuchi, Mika Nodaira, Kenichi Odaka, Kiyoshi Fukushi, Toshiaki Irie:<br />
Effects of Halogenation on Tyrosine Phosphorylation and Peptide Binding to the Src Homology 2 Domain<br />
of Lymphocyte-Specific Protein Tyrosine Kinase, Biological & Pharmaceutical Bulletin, 35(3), 433-437,<br />
2012<br />
3. Tatsuya Kikuchi, Maki Okada, Nobuki Nengaki, Kenji Furutsuka*, Hidekatsu Wakizaka, Toshimitsu<br />
Okamura, Ming-Rong Zhang, Koichi Kato: Efficient synthesis and chiral separation of 11C-labeled<br />
ibuprofen assisted by DMSO for imaging of in vivo behavior of the individual isomers by positron emission<br />
tomography, Bioorganic & Medicinal Chemistry, 19(10), 3265-3273, 2011<br />
4. Katsushi Kumata, Masanao Ogawa*, Makoto Takei*, Masayuki Fujinaga, Yuichirou Yoshida*, Nobuki<br />
Nengaki, Toshimitsu Fukumura, Kazutoshi Suzuki, Ming-Rong Zhang: Radiosynthesis of [13N]dantrolene<br />
a positron emission tomography probe for breast cancer resistant protein using no-carrier-added<br />
[13N]ammonia, Bioorganic & Medicinal Chemistry, 20(1), 305-310, 2012<br />
5. Tomoteru Yamasaki, Masayuki Fujinaga, Yuichiro Yoshida, Katsushi Kumata, Joji Yui, Kazunori<br />
Kawamura, Akiko Hatori, Toshimitsu Fukumura, Ming-Rong Zhang: Radiosynthesis and preliminary<br />
evaluation of 4-[18F]fluoro-N-[4-[6-(isopropylamino) pyrimidin-4-yl]-13-thiazol-2-yl]-N-methylbenzamide<br />
as a new positron emission tomography ligand for metabotropic glutamate receptor subtype 1, Bioorganic<br />
& Medicinal Chemistry Letters, 21(10), 2998-3001, 2011<br />
6. Chiharu Asakawa, Masanao Ogawa*, Katsushi Kumata, Masayuki Fujinaga, Tomoteru Yamasaki, Lin Xie,<br />
Joji Yui, Kazunori Kawamura, Toshimitsu Fukumura, Ming-Rong Zhang: Radiosynthesis of three<br />
[11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumors,<br />
Bioorganic & Medicinal Chemistry Letters, 21(23), 7017-7020, 2011<br />
7. Chiharu Asakawa, Masanao Ogawa, Katsushi Kumata, Masayuki Fujinaga, Koichi Kato, Tomoteru<br />
Yamasaki, Joji Yui, Kazunori Kawamura, Akiko Hatori, Toshimitsu Fukumura, Ming-Rong Zhang:<br />
[11C]Sorafenib: Radiosynthesis and preliminary PET study of brain uptake in P-gp/Bcrp knockout mice,<br />
Bioorganic & Medicinal Chemistry Letters, 21(8), 2220-2223, 2011<br />
8. Koichi Kato, Atsushi Tsuji, Tsuneo Saga, Ming-Rong Zhang: An efficient and expedient method for the<br />
synthesis of 11C-labeled a-aminoisobutyric acid: A tumor imaging agent potentially useful for cancer<br />
diagnosis, Bioorganic & Medicinal Chemistry Letters, 21(8), 2437-2440, 2011<br />
9. Atsushi Wakai, Kazuki Tsuchida, Toshimitsu Fukumura, Kazutoshi Suzuki: Isotopic effect in the (2+1)<br />
REMPI spectra of 13C-substituted methyl iodide for UV selective dissociation, Chemical Physics Letters,<br />
516(1/3), 23-28, 2011<br />
10. Tomoteru Yamasaki, Masayuki Fujinaga, Jun Maeda, Kazunori Kawamura, Joji Yui, Akiko Hatori,<br />
Yuichirou Yoshida*, Yuji Nagai, Masaki Tokunaga, Makoto Higuchi, Tetsuya Suhara, Toshimitsu<br />
Fukumura, Ming-Rong Zhang: Imaging for metabotropic glutamate receptor subtype 1 in rat and monkey<br />
brains using PET with [18F]FITM, European Journal of Nuclear Medicine and Molecular Imaging, 39(4),<br />
632-641, 2012<br />
11. Francisco Lazaro, Guerra Gomez, Yuuki Takada, Rie Hosoi, Sotaro Momosaki, Kazuhiko Yanamoto,<br />
Koutarou Nagatsu, Hisashi Suzuki, Ming-Rong Zhang, Osamu Inoue, Yasushi Arano, Toshimitsu<br />
Fukumura: Production and purification of the positron emitter zinc-63, Journal of Labelled Compounds &<br />
Radiopharmaceuticals, 55(1), 5-9, 2012<br />
12. Katsushi Kumata, Joji Yui, Akiko Hatori, Masayuki Fujinaga, Kazuhiko Yanamoto, Tomoteru Yamasaki,<br />
Kazunori Kawamura, Hidekatsu Wakizaka, Nobuki Nengaki, Yuichirou Yoshida*, Masanao Ogawa*,<br />
Toshimitsu Fukumura, Ming-Rong Zhang: Synthesis and Evaluation of Novel Carbon-11 Labeled<br />
Oxopurine Analogues for Positron Emission Tomography Imaging of Translocator Protein (18 kDa) in<br />
Peripheral Organs, Journal of Medicinal Chemistry, 54(17), 6040-6049, 2011<br />
13. Masayuki Fujinaga, Jun Maeda, Joji Yui, Akiko Hatori, Tomoteru Yamasaki, Kazunori Kawamura,<br />
Katsushi Kumata, Yuichirou Yoshida*, Yuji Nagai, Makoto Higuchi, Tetsuya Suhara, Toshimitsu<br />
Fukumura, Ming-Rong Zhang: Characterization of 1-(2-[18F]fluoro-3-pyridyl)-4-(2-isopropyl-1-oxo-<br />
36 独 立 行 政 法 人 放 射 線 医 学 総 合 研 究 所 National Institute of Radiological Sciences