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DRUGS REPORTS

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Drugs Off-Patent Reports<br />

Drugs Off-Patent<br />

Reports<br />

ISSN 0793694X<br />

Year of Expiration - 2007<br />

Drug OFF<br />

Generic Patent Patent Exclusivity Patent & Earliest 1999<br />

Patent<br />

Name Holder Expiry Expiry Exclusivity Generic 2001 1<br />

Marketer<br />

Trade Generic NAME Patent # DATE CODES DATE USD$<br />

(Mil)<br />

QUET-<br />

IAPINE<br />

Sibutramin<br />

e HCl<br />

Propulsid<br />

Kytril<br />

Seroquel Astra -<br />

Zen<br />

03/20/07<br />

4-879-288<br />

MERIDIA KNOLL 5/29/07<br />

Cisapride<br />

Risperdal Risperi -<br />

Zytrec<br />

Tabs/Syrup<br />

Fosamax<br />

done<br />

Cetirazine<br />

HCl<br />

JNJ-<br />

Allendronate<br />

Na<br />

Janssen<br />

4-929-629<br />

10/9/07<br />

4-962-115<br />

S-K-B 12/29/07<br />

4-886-808<br />

Monohydrate<br />

JNJ-<br />

Granisetron<br />

Janssen<br />

12/29/07<br />

4-804-663<br />

5-158-952<br />

Pfizer 06/25/07<br />

4-525-358<br />

Merck<br />

Co.<br />

08/06/07<br />

4-621-077<br />

5-849-726<br />

9/26/02 -<br />

NCE<br />

11/22/02 -<br />

NCE<br />

07/29/98 U-79<br />

NCE<br />

12/29/98 NCE<br />

10/17/00<br />

Aerobid Flunisolide Forrest 06/12/07<br />

4-933-168 M/D/YY<br />

LOTREL<br />

NORVASC<br />

Camptosar<br />

Amlodipine<br />

Besylate<br />

Amlodipine<br />

Besylate<br />

irinotecan<br />

HCL<br />

(oncology)<br />

Novartis 3/25/07<br />

4-879-303<br />

Pfizer 3/25/07<br />

Pharmacia<br />

Effexor XR Venlafaxine AHP-<br />

Wyeth<br />

Suprane Desflurane BOC<br />

Ohmeda<br />

* US 2000 SALES<br />

4-879-303<br />

08/20/07<br />

4-604-463<br />

12/13/07<br />

4-535-186<br />

2/2/07<br />

4-762-856<br />

U-89<br />

U-90<br />

D-37<br />

NCE<br />

03/20/07 105<br />

112<br />

05/29/07 155<br />

165<br />

10/09/07 500<br />

560<br />

12/29/07 269<br />

299<br />

12/29/07<br />

[10/29/09]<br />

690<br />

733<br />

12/08/0O NCE 06/25/07 525<br />

601<br />

09/29/07 U-114<br />

NCE<br />

08/06/07<br />

[06/06/15]<br />

505<br />

756<br />

- 06/12/07 220<br />

245<br />

07/31/97 NC 03/25/07 166<br />

187<br />

07/31/97 NCE 03/25/07 1205<br />

1270<br />

06/14/01 NCE 08/20/07 293<br />

299<br />

[116]*<br />

10/20/00 NDF 12/13/07 210<br />

233<br />

9/18/97 U-67<br />

NCE<br />

02/02/07<br />

80<br />

89<br />

Drugs Off-Patent Reports 18 Over USD$ 100 million

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