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DRUGS REPORTS

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Drugs Off-Patent Reports<br />

Drugs Off-Patent<br />

Reports<br />

ISSN 0793694X<br />

Year of Expiration - 2000<br />

Drug OFF<br />

Generic Patent Patent Exclusivity Patent & Earliest 1999<br />

Patent<br />

Name Holder Expiry Expiry Exclusivity Generic 2001 1<br />

Marketer<br />

Trade Generic NAME Patent # DATE CODES DATE USD$<br />

(Mil)<br />

2/22/00<br />

Vasotec Enalaprilat Merck &<br />

Co.<br />

Hismanal Astemizole JNJ-<br />

Janssen<br />

Buspar Buspirone<br />

HCl<br />

Lotrisone<br />

Betamethaz<br />

one Diprop<br />

2/22/00<br />

4-374-829<br />

4/3/00<br />

4-219-559<br />

B-M-S 5/22/00<br />

4-182-763<br />

Schering 10/06/00<br />

4-298-604<br />

Gluco<br />

phage<br />

Ultram<br />

ZIAC<br />

CEFTIN<br />

Atrovent<br />

Cardura<br />

ZOLADEX<br />

Pepcid Famotidine Merck<br />

& Co.<br />

10/15/00<br />

4-283-408<br />

Pepcid Famotidine Merck 10/15/00<br />

AC<br />

& Co. 4-283-408 04/28/98<br />

Glucotril Glipizide Pfizer<br />

XL<br />

Pratt --<br />

Intal Cormolyn Rhone- 9/20/00<br />

sodium Poulenc- 4-405-598<br />

Sevoflurane<br />

Metformin<br />

HCl<br />

Tramadol<br />

Hcl<br />

Bisoprolol<br />

fumerate<br />

Cefuroxime<br />

acetil<br />

Ipratropium<br />

Br<br />

Doxazosin<br />

mesylate<br />

Goserelin<br />

Acetate<br />

Rorer<br />

BM<br />

Squibb<br />

J/J - Mc<br />

Neil<br />

3/03/00<br />

-<br />

P<br />

AHP 3/24/00<br />

Lederle 4-258-062 7/31/97<br />

GW 5/12/00 M/D/YY<br />

4-267-320<br />

B 5/24/00<br />

Ingelheim 4-385-048 10/20/98<br />

Pfizer 10/18/00<br />

4-188-390 2/6/98<br />

Zeneca 4/22/99<br />

4-100-274<br />

ULTANE Abbott 12/26/04<br />

4-250-334<br />

Terazosin Hytrin Abbott 2/17/00<br />

4-251-532<br />

Neurontin Gabapentin WLA<br />

P Davis<br />

01/16/00<br />

5-084-479<br />

--<br />

Expired<br />

02/22/00<br />

M/D/YY<br />

Expired<br />

--<br />

04/03/00<br />

5/22/00 U-13 Expired<br />

05/22/00<br />

M/D/YY<br />

Expired<br />

--<br />

10/06/00<br />

M/D/YY<br />

Expired<br />

--<br />

10/15/00<br />

NS Expired<br />

10/15/00<br />

11/25/00 NDF Expired<br />

11/25/00<br />

M/D/YY<br />

Expired<br />

--<br />

09/20/00<br />

M/D/YY NCE Expired<br />

3/03/00<br />

M/D/YY NCE Expired<br />

03/03/00<br />

U-63<br />

NCE<br />

--<br />

NDF<br />

U-119<br />

NCE<br />

1-96<br />

6/27/00 --<br />

I-191<br />

6/7/00<br />

NCE<br />

725<br />

860<br />

28<br />

33<br />

540<br />

611<br />

201<br />

233<br />

1350<br />

1487<br />

125<br />

138<br />

179<br />

199<br />

89<br />

98<br />

1110<br />

1302.<br />

453<br />

501.<br />

03/24/00 173<br />

198<br />

Expired<br />

05/12/00<br />

Expired<br />

05/24/00<br />

Expired<br />

10/18/00<br />

Expired<br />

06/27/00<br />

Expired<br />

06/07/00<br />

M/D/YY -- Expired<br />

02/17/00<br />

12/30/98 U-106<br />

(Epilepsy)<br />

Expired<br />

01/16/00<br />

425<br />

485.<br />

306<br />

346<br />

330<br />

401<br />

219<br />

244<br />

114<br />

134<br />

425<br />

598.<br />

500<br />

590<br />

NA = Not Applicable ODE = Orphan Drug Exclusivity NS = New Strength<br />

NCE = New Chemical Entity NE = New Active Salt or Ester NP= New Drug Product<br />

NDF = New Dosage Form NC = New Combination 2001 1 USA + EU Sales<br />

U = Code for Therapeutic Use still I = Code for specific Indication D = New Dosing Schedule<br />

Drugs Off-Patent Reports 10 Over USD$ 100 million

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