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DRUGS REPORTS

oFF-Patents - iagim

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Drug OFF<br />

Generic Patent<br />

Patent<br />

Name Holder<br />

Marketer<br />

Drugs Off-Patent Reports<br />

Drugs Off-Patent<br />

Reports<br />

ISSN 0793694X<br />

Year of Expiration - 2013<br />

Patent<br />

Expiry<br />

+<br />

Exclusivity<br />

Expiry<br />

Patent &<br />

Exclusivit<br />

y<br />

Earliest<br />

Generic<br />

1999<br />

2001 1<br />

Trade Generic NAME Patent # DATE CODES DATE USD$<br />

(Mil)<br />

Wellbutrin Bupropion Cerenex 08/12/13 M/D/YY -<br />

08/12/13<br />

155<br />

HCl<br />

4-507-323<br />

310<br />

ZYBAN Bupropion Cerenex 08/12/13 05/14/00<br />

08/12/13<br />

200<br />

HCl<br />

5-731-000<br />

NP<br />

289<br />

ALLEGRA<br />

ALLEGRA<br />

D<br />

Fexofenadine<br />

HCl<br />

Fexofenadine<br />

HCl<br />

Hoechst<br />

Marion<br />

Roussel<br />

Hoechst<br />

Marion<br />

Roussel<br />

Zoloft Sertraline Pfizer<br />

Roerig<br />

Imitrex<br />

DDAVP<br />

Sumatriptan<br />

Succinate<br />

Desmopressin<br />

Acetate<br />

Cerenex<br />

Glaxo<br />

Rhone<br />

Poulenc<br />

Rorer<br />

Accolate Zafirlukast Astra<br />

Zeneca<br />

CRIXIVAN<br />

Indinavir<br />

Sulfate<br />

Merck<br />

Co<br />

11/26/13<br />

5-578-610<br />

11/26/13<br />

5-578-610<br />

8/13/12<br />

5-249-699 08/07/00<br />

09/10/13<br />

5-554-639<br />

9/10/08<br />

5-407-398<br />

5-763-407<br />

01/06/13<br />

5-482-963<br />

05/07/13<br />

5-413-999<br />

ASACOL Mesalamine P&G 07/30/13<br />

5-541-171<br />

REZULIN Troglitazone Warner-L 09/13/13<br />

5-478-852<br />

Magnevist<br />

Viracept<br />

Gadapentetate<br />

Di-meglumine<br />

Nelfinavir<br />

Mesalate<br />

Berlex 10/01/13<br />

5-560-903<br />

Agguron 10/07/13<br />

5-484-926<br />

07/25/01 U-138<br />

NCE<br />

12/24/00 U-138<br />

NC<br />

8/26/00<br />

11/26/13<br />

11/26/13<br />

360<br />

420<br />

105<br />

140<br />

NCE 08/13/12 1629<br />

1780<br />

NDF<br />

U-72<br />

09/10/13 898<br />

990<br />

M/D/YY [09/10/08]<br />

12/23/13<br />

170<br />

210<br />

- - 01/09/13 146<br />

159<br />

3/13/01 U-132<br />

NCE<br />

8/18/00 U-141<br />

I-203<br />

01/29/02 U-163<br />

NCE<br />

- -<br />

-<br />

03/14/02 -<br />

NCE<br />

05/07/13 335<br />

356<br />

07/30/13 163<br />

183<br />

09/13/13 855<br />

930<br />

10/1/13 128<br />

155<br />

10/07/13 399<br />

410<br />

NA = Not Applicable ODE = Orphan Drug Exclusivity NS = New Strength<br />

NCE = New Chemical Entity NE = New Active Salt or Ester NP = New Drug Product<br />

NDF = New Dosage Form NC = New Combination 2001 1 USA + EU Sales<br />

U = Code for Therapeutic Use still I = Code for specific Indication D = New Dosing Schedule<br />

under Patent Protection<br />

under Exclusivity Protection<br />

Drugs Off-Patent Reports 22 Over USD$ 100 million

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