Final Programme - iuphar

FC11 G protein-coupled 7TM receptors:
From molecular to physiological function
Thu 036 The conserved Trp IV:10 (4.50) together with Ser/Asn II:05 (2.45) are crucial for 7TM receptors
activation and might be a putative cholesterol binding site
Jacek Mokrosinski, (Denmark), R Nygaard, MS Engelstoft, L Valentin-Hansen, B Holst, TW Schwartz
Thu 037 Screening and characterization of GPCR C-terminal tail interactions with the PSD-95 PDZ domains
Thor Møller, (Denmark), P Jacky, A Bach, K Strømgaard, T Schwartz, K Martinez
Thu 038 Novel pathway of smooth muscle contraction by UTP in rat aortic myocyte
Hiromitsu Morita, (Japan), M Sugihara, M Matsuda, S Kajioka, Y Ito, K Abe, M Hirata
Thu 039 β3-adrenoceptors substitute the role M2 muscarinic receptors in the heart of stressed mice
Jaromir Myslivecek, (Czech Republic), M Novakova, V Farar, R Kvetnansky
Thu 040 Presynaptic BK channels activated by IP3-induced Ca 2+ release are involved in prostanoid TP
receptor-mediated inhibition of noradrenaline release from the rat gastric sympathetic nerves
Kumiko Nakamura, (Japan), K Yokotani
Thu 041 Mutational analysis of an M4 muscarinic acetylcholine receptor allosteric site
Vindhya Nawaratne, (Australia), K Leach, CC Felder, PM Sexton, A Christopoulos
Thu 042 The involvement of nitric oxide in the local antinociceptive effects of JWH-015 and expression of
cannabinoid-2, μ- and δ-opioid receptors during chronic inflammatory pain in mice
R Negrete, J Martín-Campos, A Hervera, S Leánez, Olga Pol (Spain)
Thu 043 Pharmacological evaluation of new bivalent ligands aimed to interact with orthosteric and allosteric
sites of mAChRs
Marta Nesi, (Italy)
Thu 044 Conditional mutant mouse with enhanced Gα-i2 signalling due to loss of regulator of G protein signalling
(RGS) regulation
Richard Neubig, (USA), X Huang, S Wade, R Charbeneau
Thu 045 Pertussis toxin inhibits EP4 and IP receptor-mediated cAMP production in adult rat dorsal root ganglion
cells
Kai-Yu Ng, (PR China), Y-H Wong, H Wise
Thu 046 Identification of Adrenergic Receptor Interacting Protein (ARIP), as a novel receptor-interacting protein
that modulates α1A- and α1L-adrenoceptor expression
Atsushi Nishimune, (Japan), F Suzuki, H Yoshiki, S Morishima, I Muramatsu
Thu 047 G protein-coupled estrogen receptor 1 function in vivo and in vitro
B Olde, C Sandén, S Broselid, U Mårtensson, Fredrik Leeb-Lundberg, (Sweden)
Thu 048 The expression of cardiac and lymphocytic GRKs in human cardiovascular diseases correlated to the
expression levels of β-ARs
Eduardo Oliver, (Spain), F Monto, D Vicente, J Agüero, EE Rovira, L Almenar, P D'Ocon
Thu 049 Conditional functional selectivity of β2-adrenoceptor ligands in stimulating adenylyl cyclase and ERK
phosphorylation in HEK 293 cells
Gülnihal Özcan, (Turkey), A Kaya, O Onaran, Ö Ugur
Thu 050 The three α1-AR subtypes show different spatio-temporal patterns of ERK1/2 phosphorylation and
internalization
Miguel Perez-Aso, (Spain), V Segura, M-A Noguera, P D'Ocon
Thursday 22 July ■ 13:00 - 14:00 ■ Poster Area 283