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ELS-tíðindi - júní 2001

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50 <strong>ELS</strong> <strong>tíðindi</strong> 6/01<br />

(21) 5840<br />

(22) 5.2.<strong>2001</strong><br />

(41) 5.2.<strong>2001</strong><br />

(51) C07D 263/32; C07D 277/24; A61K<br />

31/421; A61K 31/426; C07D 413/12;<br />

C07D 417/12; A61K 31/422; A61K<br />

31/427<br />

(54) Setnar oxazól og þíazól afleiður sem<br />

hPPAR gamma og hPPAR alfa<br />

hvatar.<br />

(71) Glaxo Group Limited, Glaxo<br />

Wellcome House, Berkeley Avenue,<br />

Greenford, Middlesex, UB6 ONN,<br />

Bretlandi.<br />

(72) Jon Loren Collins, Research Triangle<br />

Park; Timothy Mark Willson, Research<br />

Triangle Park; Jeffrey Alan Oplinger,<br />

Research Triangle Park; Milana<br />

Duzube, Chapel Hill; North Carolina,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 7.8.98, GB, 9817118.4<br />

(85) 5.2.<strong>2001</strong><br />

(86) 5.8.99, PCT/EP99/05666<br />

(21) 5843<br />

(22) 9.2.<strong>2001</strong><br />

(41) 9.2.<strong>2001</strong><br />

(51) C07D 473/06; A61K 31/522<br />

(54) Fenýl janþín (yanthine) afleiður.<br />

(71) Glaxo Group Limited, Glaxo<br />

Wellcome House, Berkeley Avenue,<br />

Greenford, Middlesex, UB6 0NN,<br />

Bretlandi.<br />

(72) Susan Mary Daluge; Cynthia Holder<br />

Jurgensen; Michael Tolar Martin;<br />

Martin Howard Osterhout; Research<br />

Triangle Park, North Carolina,<br />

Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 13.8.98, GB, 9817623.3<br />

(85) 9.2.<strong>2001</strong><br />

(86) 11.8.99, PCT/EP99/05814<br />

(21) 5848<br />

(22) 16.2.<strong>2001</strong><br />

(41) 16.2.<strong>2001</strong><br />

(51) A61K 38/00<br />

(54) Aðferð til að stilla T-frumur sem eru<br />

svarar og samsetningu þeirra.<br />

(71) Biogen, Inc., 14 Cambridge Center,<br />

Cambridge, Massachusetts 02142,<br />

Bandaríkjunum.<br />

(72) Daniel Magilavy, Cambridge,<br />

Massachusetts, Bandaríkjunum.<br />

(74) PATICE, Ólafur Ragnarsson, hrl.,<br />

Skeifunni 7, 108 Reykjavík.<br />

(30) 31.8.98, US, 60/098,456<br />

(85) 16.2.<strong>2001</strong><br />

(86) 31.8.99, PCT/US99/20026<br />

(21) 5849<br />

(22) 16.2.<strong>2001</strong><br />

(41) 16.2.<strong>2001</strong><br />

(51) C07D 213/42; C07D 239/42; C07D<br />

295/22; C07D 213/74; C07D 417/12;<br />

C07D 401/12; C07D 215/12; C07D<br />

333/20; C07D 241/12; A61K 31/44;<br />

A61K 31/495<br />

(54) Arýlpíperazín og notkun þeirra sem<br />

málmprótínasa bælandi miðlar<br />

(MMP).<br />

(71) AstraZeneca AB, S-151 85 Södertälje,<br />

Svíþjóð.<br />

(72) Bernard Christophe Barlaam,<br />

Wilmington, Delaware, Bandaríkjunum;<br />

Nicholas John Newcombe,<br />

Macclesfield, Cheshire, Bretlandi;<br />

Howard Tucker, Macclesfield,<br />

Cheshire, Bretlandi; David Waterson,<br />

Macclesfield, Cheshire, Bretlandi.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 31.8.98, EP, 98402144.4<br />

4.6.99, EP, 99401351.4<br />

(85) 16.2.<strong>2001</strong><br />

(86) 25.8.99, PCT/GB99/02801<br />

(21) 5850<br />

(22) 16.2.<strong>2001</strong><br />

(41) 16.2.<strong>2001</strong><br />

(51) A23L 1/30; A23L 1/302; A61K 31/385<br />

(54) Andoxunar samsetning sem<br />

samanstendur af asetýl L-karnitíni og<br />

alfa-lípósýru.<br />

(71) Sigma-Tau Healthscience S.P.A.,<br />

Via Treviso, 4, I-00040 Pomezia,<br />

Ítalíu.<br />

(72) Claudio Cavazza, Roma, Ítalíu.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 1.9.98, IT, RM98A000566<br />

(85) 16.2.<strong>2001</strong><br />

(86) 19.8.99, PCT/IT99/00268<br />

(21) 5852<br />

(22) 20.2.<strong>2001</strong><br />

(41) 20.2.<strong>2001</strong><br />

(51) A61K 31/505; A61P 25/16<br />

(54) Lyfjamiðlar til meðhöndlunar á<br />

parkinsonsveiki ADHD og smákirtilsæxlum.<br />

(71) Pfizer Products Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Elisa Rose Jackson, Norwich;<br />

Stafford McLean, Stonington; Stevin<br />

Howard Zorn, North Stonington;<br />

Connecticut, Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 21.9.98, US, 60/101,191<br />

12.10.98, US, 60/103,868<br />

(85) 20.2.<strong>2001</strong><br />

(86) 3.9.99, PCT/IB99/01503<br />

(21) 5856<br />

(22) 23.2.<strong>2001</strong><br />

(41) 23.2.<strong>2001</strong><br />

(51) A61K 38/17; A61K 39/395<br />

(54) Aðferðir þar sem integrín-mótlyf eru<br />

notuð til að meðhöndla margföld<br />

mergæxli og uppsog í bein af völdum<br />

mergæxla.<br />

(71) Board of Regents, the University<br />

of Texas system, 201 West 71st<br />

Street, Austin, Texas 78701,<br />

Bandaríkjunum.<br />

(72) Gregory R. Mundy; Toshiyuki<br />

Yoneda; San Antonio, Texas,<br />

Bandaríkjunum.<br />

(74) PATICE, Ólafur Ragnarsson, hrl.,<br />

Skeifunni 7, 108 Reykjavík.<br />

(30) 14.9.98, US, 60/100,182<br />

(85) 23.2.<strong>2001</strong><br />

(86) 13.9.99, PCT/US99/21170<br />

(21) 5857<br />

(22) 23.2.<strong>2001</strong><br />

(41) 23.2.<strong>2001</strong><br />

(51) A22C 25/16<br />

(54) Aðferð til flökunar á fiski og<br />

flökunarvél til notkunar við flökunina.<br />

(71) Arne K. Nordstrand, N-6050<br />

Valderøy, Noregi.<br />

(72) Arne K. Nordstrand, Valderøy,<br />

Noregi.<br />

(74) PATICE, Ólafur Ragnarsson, hrl.,<br />

Skeifunni 7, 108 Reykjavík.<br />

(30) 24.8.98, NO, 19983885<br />

(85) 23.2.<strong>2001</strong><br />

(86) 23.8.99, PCT/NO99/00263<br />

(21) 5858<br />

(22) 23.2.<strong>2001</strong><br />

(41) 23.2.<strong>2001</strong><br />

(51) C07D 215/42; A61K 31/47; C07D<br />

221/16; C07D 215/46; C07D 417/12;<br />

C07D 413/12<br />

(54) 4-amínó setinn-2-setinn-1, 2, 3, 4tetrahýdrókínólín<br />

sem CETP latar.<br />

(71) Pfizer Products Inc., Eastern Point<br />

Road, Groton, Connecticut 06340,<br />

Bandaríkjunum.<br />

(72) Michael Paul DeNinno, Gales Ferry;<br />

George Tetteh Magnus-Aryitey,<br />

Ledyard; Roger Benjamin Ruggeri,<br />

Waterford; Ronald Thure Wester,<br />

Ledyard; Connecticut, Bandaríkjunum.<br />

(74) Faktor einkaleyfaskrifstofa, ehf.,<br />

Pósthólf 678, 121 Reykjavík.<br />

(30) 17.9.98, US, 60/100,927<br />

(85) 23.2.<strong>2001</strong><br />

(86) 10.9.99, PCT/IB99/01534

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