ELS-tíðindi - júní 2001
ELS-tíðindi - júní 2001
ELS-tíðindi - júní 2001
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50 <strong>ELS</strong> <strong>tíðindi</strong> 6/01<br />
(21) 5840<br />
(22) 5.2.<strong>2001</strong><br />
(41) 5.2.<strong>2001</strong><br />
(51) C07D 263/32; C07D 277/24; A61K<br />
31/421; A61K 31/426; C07D 413/12;<br />
C07D 417/12; A61K 31/422; A61K<br />
31/427<br />
(54) Setnar oxazól og þíazól afleiður sem<br />
hPPAR gamma og hPPAR alfa<br />
hvatar.<br />
(71) Glaxo Group Limited, Glaxo<br />
Wellcome House, Berkeley Avenue,<br />
Greenford, Middlesex, UB6 ONN,<br />
Bretlandi.<br />
(72) Jon Loren Collins, Research Triangle<br />
Park; Timothy Mark Willson, Research<br />
Triangle Park; Jeffrey Alan Oplinger,<br />
Research Triangle Park; Milana<br />
Duzube, Chapel Hill; North Carolina,<br />
Bandaríkjunum.<br />
(74) Faktor einkaleyfaskrifstofa, ehf.,<br />
Pósthólf 678, 121 Reykjavík.<br />
(30) 7.8.98, GB, 9817118.4<br />
(85) 5.2.<strong>2001</strong><br />
(86) 5.8.99, PCT/EP99/05666<br />
(21) 5843<br />
(22) 9.2.<strong>2001</strong><br />
(41) 9.2.<strong>2001</strong><br />
(51) C07D 473/06; A61K 31/522<br />
(54) Fenýl janþín (yanthine) afleiður.<br />
(71) Glaxo Group Limited, Glaxo<br />
Wellcome House, Berkeley Avenue,<br />
Greenford, Middlesex, UB6 0NN,<br />
Bretlandi.<br />
(72) Susan Mary Daluge; Cynthia Holder<br />
Jurgensen; Michael Tolar Martin;<br />
Martin Howard Osterhout; Research<br />
Triangle Park, North Carolina,<br />
Bandaríkjunum.<br />
(74) Faktor einkaleyfaskrifstofa, ehf.,<br />
Pósthólf 678, 121 Reykjavík.<br />
(30) 13.8.98, GB, 9817623.3<br />
(85) 9.2.<strong>2001</strong><br />
(86) 11.8.99, PCT/EP99/05814<br />
(21) 5848<br />
(22) 16.2.<strong>2001</strong><br />
(41) 16.2.<strong>2001</strong><br />
(51) A61K 38/00<br />
(54) Aðferð til að stilla T-frumur sem eru<br />
svarar og samsetningu þeirra.<br />
(71) Biogen, Inc., 14 Cambridge Center,<br />
Cambridge, Massachusetts 02142,<br />
Bandaríkjunum.<br />
(72) Daniel Magilavy, Cambridge,<br />
Massachusetts, Bandaríkjunum.<br />
(74) PATICE, Ólafur Ragnarsson, hrl.,<br />
Skeifunni 7, 108 Reykjavík.<br />
(30) 31.8.98, US, 60/098,456<br />
(85) 16.2.<strong>2001</strong><br />
(86) 31.8.99, PCT/US99/20026<br />
(21) 5849<br />
(22) 16.2.<strong>2001</strong><br />
(41) 16.2.<strong>2001</strong><br />
(51) C07D 213/42; C07D 239/42; C07D<br />
295/22; C07D 213/74; C07D 417/12;<br />
C07D 401/12; C07D 215/12; C07D<br />
333/20; C07D 241/12; A61K 31/44;<br />
A61K 31/495<br />
(54) Arýlpíperazín og notkun þeirra sem<br />
málmprótínasa bælandi miðlar<br />
(MMP).<br />
(71) AstraZeneca AB, S-151 85 Södertälje,<br />
Svíþjóð.<br />
(72) Bernard Christophe Barlaam,<br />
Wilmington, Delaware, Bandaríkjunum;<br />
Nicholas John Newcombe,<br />
Macclesfield, Cheshire, Bretlandi;<br />
Howard Tucker, Macclesfield,<br />
Cheshire, Bretlandi; David Waterson,<br />
Macclesfield, Cheshire, Bretlandi.<br />
(74) Faktor einkaleyfaskrifstofa, ehf.,<br />
Pósthólf 678, 121 Reykjavík.<br />
(30) 31.8.98, EP, 98402144.4<br />
4.6.99, EP, 99401351.4<br />
(85) 16.2.<strong>2001</strong><br />
(86) 25.8.99, PCT/GB99/02801<br />
(21) 5850<br />
(22) 16.2.<strong>2001</strong><br />
(41) 16.2.<strong>2001</strong><br />
(51) A23L 1/30; A23L 1/302; A61K 31/385<br />
(54) Andoxunar samsetning sem<br />
samanstendur af asetýl L-karnitíni og<br />
alfa-lípósýru.<br />
(71) Sigma-Tau Healthscience S.P.A.,<br />
Via Treviso, 4, I-00040 Pomezia,<br />
Ítalíu.<br />
(72) Claudio Cavazza, Roma, Ítalíu.<br />
(74) Faktor einkaleyfaskrifstofa, ehf.,<br />
Pósthólf 678, 121 Reykjavík.<br />
(30) 1.9.98, IT, RM98A000566<br />
(85) 16.2.<strong>2001</strong><br />
(86) 19.8.99, PCT/IT99/00268<br />
(21) 5852<br />
(22) 20.2.<strong>2001</strong><br />
(41) 20.2.<strong>2001</strong><br />
(51) A61K 31/505; A61P 25/16<br />
(54) Lyfjamiðlar til meðhöndlunar á<br />
parkinsonsveiki ADHD og smákirtilsæxlum.<br />
(71) Pfizer Products Inc., Eastern Point<br />
Road, Groton, Connecticut 06340,<br />
Bandaríkjunum.<br />
(72) Elisa Rose Jackson, Norwich;<br />
Stafford McLean, Stonington; Stevin<br />
Howard Zorn, North Stonington;<br />
Connecticut, Bandaríkjunum.<br />
(74) Faktor einkaleyfaskrifstofa, ehf.,<br />
Pósthólf 678, 121 Reykjavík.<br />
(30) 21.9.98, US, 60/101,191<br />
12.10.98, US, 60/103,868<br />
(85) 20.2.<strong>2001</strong><br />
(86) 3.9.99, PCT/IB99/01503<br />
(21) 5856<br />
(22) 23.2.<strong>2001</strong><br />
(41) 23.2.<strong>2001</strong><br />
(51) A61K 38/17; A61K 39/395<br />
(54) Aðferðir þar sem integrín-mótlyf eru<br />
notuð til að meðhöndla margföld<br />
mergæxli og uppsog í bein af völdum<br />
mergæxla.<br />
(71) Board of Regents, the University<br />
of Texas system, 201 West 71st<br />
Street, Austin, Texas 78701,<br />
Bandaríkjunum.<br />
(72) Gregory R. Mundy; Toshiyuki<br />
Yoneda; San Antonio, Texas,<br />
Bandaríkjunum.<br />
(74) PATICE, Ólafur Ragnarsson, hrl.,<br />
Skeifunni 7, 108 Reykjavík.<br />
(30) 14.9.98, US, 60/100,182<br />
(85) 23.2.<strong>2001</strong><br />
(86) 13.9.99, PCT/US99/21170<br />
(21) 5857<br />
(22) 23.2.<strong>2001</strong><br />
(41) 23.2.<strong>2001</strong><br />
(51) A22C 25/16<br />
(54) Aðferð til flökunar á fiski og<br />
flökunarvél til notkunar við flökunina.<br />
(71) Arne K. Nordstrand, N-6050<br />
Valderøy, Noregi.<br />
(72) Arne K. Nordstrand, Valderøy,<br />
Noregi.<br />
(74) PATICE, Ólafur Ragnarsson, hrl.,<br />
Skeifunni 7, 108 Reykjavík.<br />
(30) 24.8.98, NO, 19983885<br />
(85) 23.2.<strong>2001</strong><br />
(86) 23.8.99, PCT/NO99/00263<br />
(21) 5858<br />
(22) 23.2.<strong>2001</strong><br />
(41) 23.2.<strong>2001</strong><br />
(51) C07D 215/42; A61K 31/47; C07D<br />
221/16; C07D 215/46; C07D 417/12;<br />
C07D 413/12<br />
(54) 4-amínó setinn-2-setinn-1, 2, 3, 4tetrahýdrókínólín<br />
sem CETP latar.<br />
(71) Pfizer Products Inc., Eastern Point<br />
Road, Groton, Connecticut 06340,<br />
Bandaríkjunum.<br />
(72) Michael Paul DeNinno, Gales Ferry;<br />
George Tetteh Magnus-Aryitey,<br />
Ledyard; Roger Benjamin Ruggeri,<br />
Waterford; Ronald Thure Wester,<br />
Ledyard; Connecticut, Bandaríkjunum.<br />
(74) Faktor einkaleyfaskrifstofa, ehf.,<br />
Pósthólf 678, 121 Reykjavík.<br />
(30) 17.9.98, US, 60/100,927<br />
(85) 23.2.<strong>2001</strong><br />
(86) 10.9.99, PCT/IB99/01534