Inflammation - Institutleder til klinisk medicin
Inflammation - Institutleder til klinisk medicin
Inflammation - Institutleder til klinisk medicin
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Antihistaminer - virkningsmekanisme<br />
PIP 2<br />
IP 3<br />
PKC<br />
PLC<br />
DAG<br />
G q<br />
H 1<br />
- antihistamin ÷<br />
H 1 -receptor<br />
Ca 2+<br />
Antihistaminer - farmakodynamik<br />
Kompetitive antagonister (astemizol non-kompetitiv)<br />
Heterogen gruppe<br />
terfenadin<br />
astemizol<br />
cetirizin<br />
- prodrug<br />
- aktive metabolitter<br />
- metaboliseres ikke