synthesis and catalytic functionalization of biologically active indoles

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11 “Selective Reduction and Functionalization of Diethyl 1-alkyl-1Hindole-2,3-dicarboxylates” A. Sayyed, K. Alex, A. Tillack, N. Schwarz, A. Spannenberg, D. Michalik, M. Beller, Tetrahedron 2008, 64, 4590-4595. Posterbeiträge 1 N. Schwarz, A. Pews-Davtyan, K. Alex, A. Tillack, M. Beller, Catalytic Synthesis of 3-Silyloxyindoles and Palladium-catalyzed C-O Coupling of Electron- Rich Indoles, XXIII International Conference on Organometallic Chemistry, 13-18.07.2008, Rennes, Frankreich 23 rd ICOMC Poster Prize for recognition of innovative work in the field of catalysis 2 N. Schwarz, A. Tillack, K. Alex, I. Sayyed, M. Beller, A novel Palladium Catalyst for the Amination of Electron-rich Indole Derivatives, 10. Frühjahrssymposium, 27.-29.03.2008, Rostock 3 N. Schwarz, K. Alex, A. Tillack, V. Khedkar, M. Beller, Synthesis of New Indole Derivatives via Hydroamination, School Medicinal Chemistry, 25.- 27.09.2006, Regensburg 4 N. Schwarz, K. Alex, A. Tillack, V. Khedkar, M. Beller, Synthesis of New Indole Derivatives via Hydroamination, 1 st European Chemistry Congress, 28.-31.08.2006, Budapest, Ungarn 5 N. Schwarz, K. Alex, A. Tillack, V. Khedkar, M. Beller, Eine neue Methode für die Synthese von Tryptaminen und Tryptopholen mittels katalytischer Hydrohydrazinierung von Alkinen, XXIX. Jahrestreffen Deutscher Katalytiker, 15.-17.03.2006, Weimar Vortrag N. Schwarz, Synthesis of New Indole Derivatives-Development of 5-HT6 Receptor Ligands, 4 th Symposium of the Research Training Group 1213 (RTG), New Methods for Sustainability in Catalysis and Technique, 17.07.2008, Rostock
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Leibniz-Institut für Katalyse e. V
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Für meine Eltern Siegfried und Ker
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Mein besonderer Dank gilt Dr. Anneg
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Table of Contents Preface .........
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List of Abbreviations Ac Acetyl aq
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Preface The search for drugs is an
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1 Palladium-catalyzed Coupling Reac
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3 Publications 3.1 Titanium-Catalyz
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1092 N. Schwarz et al. LETTER Table
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1094 N. Schwarz et al. LETTER 2,6-d
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3 Publications 84 3.2 Zinc-Promoted
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Table 2: Reaction of N-methyl-N-phe
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Am. Chem. Soc. 2002, 124, 15168 - 1
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A novel palladium catalyst for the
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Table 2. Reaction of different amin
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3 Publications 94 Experimental Data
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3 Publications 96 (q); 115.3 (d, J
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3 Publications 98 3.4 Palladium-Cat
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PAPER Coupling Reactions of Electro
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PAPER Coupling Reactions of Electro
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Page 119 and 120: 3 Publications 108 3.5 Synthesis of
Page 121 and 122: Scheme 2 Ti-catalyzed synthesis of
Page 123 and 124: mixture was used for the synthesis
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Page 127 and 128: FULL PAPER DOI: 10.1002/ejoc.200800
Page 129 and 130: Synthesis of Potential 5-HT 6 Recep
Page 139 and 140: FULL PAPER DOI: 10.1002/ejoc.200700
Page 141 and 142: Synthesis of Indole-2,3-dicarboxyla
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Page 151 and 152: DOI: 10.1002/cssc.200700160 General
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Page 155 and 156: Zn-Catalyzed Hydroamination of Term
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Page 161 and 162: 3 Publications 150 3.11 First Synth
Page 163 and 164: 4608 K. Alex et al. / Tetrahedron L
Page 165: Publikationen 1 Titanium-Catalyzed
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