section 1 - World Intellectual Property Organization

23/1998
11 Jun/juin 1998 PCT Gazette - Section I - Gazette du PCT 10051
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH HU ID
IL IS JP KE KG KP KR KZ LC LK LR LS LT
LU LV MD MG MK MN MW MX NO NZ PL PT
RO RU SD SE SG SI SK SL TJ TM TR TT UA
UG US UZ VN YU ZW; AP (GH KE LS MW SD
SZ UG ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH DE DK ES FI FR GB GR
IE IT LU MC NL PT SE); OA (BF BJ CF CG CI
CM GA GN ML MR NE SN TD TG).
(11) WO 98/24803 (13) A1
(21) PCT/EP97/06829
(22) 8 Dec/déc 1997 (08.12.1997)
(25) de (26) de
(31) 196 52 408.3 (32) 6 Dec/déc 1996 (33) DE
(06.12.1996)
(43) 11 Jun/juin 1998 (11.06.1998)
(51) 6 C07J 53/00, A61K 31/565
(54) STEROID ESTERS, METHOD FOR THE MANU-
FACTURE THEREOF AND THEIR PHARMA-
CEUTICAL USE
ESTERS STEROIDES, LEUR PROCEDE DE
PREPARATION ET LEUR UTILISATION PHAR-
MACEUTIQUE
(71) SCHERING AKTIENGESELLSCHAFT
[DE/DE]; Müllerstrasse 178, D–13353 Berlin
(DE).
(72) KLAR, Ulrich; Isegrimsteig 8a, D–13503 Berlin
(DE). CLEVE, Arwed; Konstanzer Strasse
8, D–10707 Berlin (DE). SCHWEDE, Wolfgang;
Klosterheider Weg 35, D–13467 Berlin
(DE). NEEF, Günter; Markgraf–Albrecht–Strasse
4, D–10711 Berlin (DE). OTTOW, Eckhard;
Moltkestrasse 48, D–12203 Berlin (DE). CHWA-
LISZ, Kristof; Lobber Steig 7a, D–13503 Berlin
(DE). SCHNEIDER, Martin; Schluchseestrasse
6a, D–13469 Berlin (DE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DK EE ES FI GB GE GH HU IL IS JP
KE KG KP KR KZ LC LK LR LS LT LU LV MD
MG MK MN MW MX NO NZ PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT UA UG UZ VN
YU ZW; AP (GH KE LS MW SD SZ UG ZW);
EA (AM AZ BY KG KZ MD RU TJ TM); EP (AT
BE CH DE DK ES FI FR GB GR IE IT LU MC
NL PT SE); OA (BF BJ CF CG CI CM GA GN
ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/24804
(21) PCT/US97/22355
(13) A2
(22) 5 Dec/déc 1997 (05.12.1997)
(25) en (26) en
(31) 60/032,129 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 60/041,938 (32) 4 Apr/avr 1997
(04.04.1997)
(33) US
(31) 60/050,796 (32) 26 Jun/juin 1997
(26.06.1997)
(33) US
(43) 11 Jun/juin 1998 (11.06.1998)
(51) 6 C07K 5/02
(54) INHIBITORS OF INTERLEUKIN–1 CONVER-
TING ENZYME
INHIBITEUR DE L’ENZYME DE CONVER-
SION DE L’INTERLEUKINE 1
(71) VERTEX PHARMACEUTICALS INCORPO-
RATED [US/US]; 130 Waverly Street, Cambridge,
MA 02139–4242 (US).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) GOLEC, Julian, M., C. [GB/GB]; 8 Manor
Farm, Chapel Road, Ashbury, Swindon, Wiltshire
SN6 8LS (GB). LAUFFER, David, J. [US/US];
254 Taylor Road, Stow, MA 01775 (US). LIVING-
STON, David, J. [US/US]; 20 Madison Avenue,
Newtonville, MA 02160 (US). MULLICAN, Michael,
D. [US/US]; 110 Parker Road, Needham,
MA 02194 (US). NYCE, Philip, L. [US/US]; 18
Prospect Street, Millbury, MA 01527 (US). RO-
BIDOUX, Andrea, L., C. [US/US]; 180 Salem
Street, Andover, MA 01810 (US). WANNAMA-
KER, Marion, W. [US/US]; 375 Harvard Road,
Stow, MA 01775 (US).
(74) HALEY, James, F., Jr.; Fish & Neave, 1251
Avenue of the Americas, New York, NY 10020
(US) et al. / etc.
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH HU ID
IL IS JP KE KG KP KR KZ LC LK LR LS LT
LU LV MD MG MK MN MW MX NO NZ PL PT
RO RU SD SE SG SI SK SL TJ TM TR TT UA
UG US UZ VN YU ZW; AP (GH KE LS MW SD
SZ UG ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH DE DK ES FI FR GB GR
IE IT LU MC NL PT SE); OA (BF BJ CF CG CI
CM GA GN ML MR NE SN TD TG).
(11) WO 98/24805
(21) PCT/US97/22289
(13) A1
(22) 5 Dec/déc 1997 (05.12.1997)
(25) en (26) en
(31) 60/032,792 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 60/042,660 (32) 4 Apr/avr 1997
(04.04.1997)
(33) US
(31) 60/053,001 (32) 26 Jun/juin 1997
(26.06.1997)
(33) US
(43) 11 Jun/juin 1998 (11.06.1998)
(51) 6 C07K 5/023, A61K 38/06
(54) INHIBITORS OF INTERLEUKIN–1 CONVER-
TING ENZYME
INHIBITEURS DE L’ENZYME DE CONVER-
SION DE L’INTERLEUKINE–1
(71) VERTEX PHARMACEUTICALS INCORPO-
RATED [US/US]; 130 Waverly Street, Cambridge,
MA 02139–4242 (US).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) GOLEC, Julian, M., C. [GB/GB]; 8 Manor
Farm, Chapel Road, Ashbury, Swindon, Wiltshire
SN6 8LS (GB). LAUFFER, David, J. [US/US];
254 Taylor Road, Stow, MA 01775 (US). LIVING-
STON, David, J. [US/US]; 20 Madison Avenue,
Newtonville, MA 02160 (US). MULLICAN, Michael,
D. [US/US]; 110 Parker Road, Needham,
MA 02194 (US). MURCKO, Mark, A. [US/US];
520 Marshall Street, Holliston, MA 01746 (US).
NYCE, Philip, L. [US/US]; 18 Prospect Street,
Millbury, MA 01527 (US). ROBIDOUX, Andrea,
L., C. [US/US]; 180 Salem Street, Andover,
MA 01810 (US). WANNAMAKER, Marion,
W. [US/US]; 375 Harvard Road, Stow, MA 01775
(US).
(74) HALEY, James, F., Jr.; Fish & Neave, 1251
Avenue of the Americas, New York, NY 10020
(US) et al. / etc.
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH HU ID
IL IS JP KE KG KP KR KZ LC LK LR LS LT
LU LV MD MG MK MN MW MX NO NZ PL PT
RO RU SD SE SG SI SK SL TJ TM TR TT UA
UG US UZ VN YU ZW; AP (GH KE LS MW SD
SZ UG ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH DE DK ES FI FR GB GR
IE IT LU MC NL PT SE); OA (BF BJ CF CG CI
CM GA GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/24806
(21) PCT/US97/21636
(13) A2
(22) 5 Dec/déc 1997 (05.12.1997)
(25) en (26) en
(31) 08/761,190 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 08/762,381 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 08/771,317 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 08/760,916 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 08/761,313 (32) 6 Dec/déc 1996
(06.12.1996)
(33) US
(31) 08/985,201 (32) 4 Dec/déc 1997
(04.12.1997)
(33) US
(31) 08/984,881 (32) 4 Dec/déc 1997
(04.12.1997)
(33) US
(31) 08/985,056 (32) 4 Dec/déc 1997
(04.12.1997)
(33) US
(31) 08/984,884 (32) 4 Dec/déc 1997
(04.12.1997)
(33) US
(31) 08/985,298 (32) 4 Dec/déc 1997
(04.12.1997)
(33) US
(43) 11 Jun/juin 1998 (11.06.1998)
(51) 6 C07K 5/062, 5/078, C07D 413/12, 413/14,
271/10, 417/12
(54) SERINE PROTEASE INHIBITORS
INHIBITEURS DE LA SERINE PROTEASE
(71) CORTECH, INC. [US/US]; 6850 North Broadway,
Denver, CO 80221 (US).
(71, 72) GYORKOS, Albert [US/US]; 11795 Decatur
Drive, Westminster, CO 80234 (US). SPRUCE,
Lyle, W. [US/US]; 948 Camino del Sol, Chula
Vista, CA 91910 (US).
(74) BURKE, John, E. et al. / etc.; Cushman Darby &
Cushman, Intellectual Property Group of Pillbury
Madison & Sutro, 1100 New York Avenue, N.W.,
Washington, DC 20005 (US).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH HU ID
IL IS JP KE KG KP KR KZ LC LK LR LS LT LU
LV MD MG MK MN MW MX NO NZ PL PT RO
RU SD SE SG SI SK SL TJ TM TR TT UA UG
UZ VN YU ZW; AP (GH KE LS MW SD SZ UG
ZW); EA (AM AZ BY KG KZ MD RU TJ TM);
EP (AT BE CH DE DK ES FI FR GB GR IE IT
LU MC NL PT SE); OA (BF BJ CF CG CI CM
GA GN ML MR NE SN TD TG).
(11) WO 98/24807
(21) PCT/US97/22251
(13) A2
(22) 4 Dec/déc 1997 (04.12.1997)
(25) en (26) en
(31) 60/032,358 (32) 4 Dec/déc 1996
(04.12.1996)
(33) US
(31) 08/760,672 (32) 4 Dec/déc 1996
(04.12.1996)
(33) US
(31) 08/855,204 (32) 13 May/mai 1997
(13.05.1997)
(33) US
(43) 11 Jun/juin 1998 (11.06.1998)
(51) 6 C07K 7/00
(54) SOMATOSTATIN ANTAGONISTS
ANTAGONISTES DE LA SOMATOSTATINE