PCT/1998/22 - World Intellectual Property Organization
PCT/1998/22 - World Intellectual Property Organization
PCT/1998/22 - World Intellectual Property Organization
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<strong>22</strong>/<strong>1998</strong><br />
4 Jun/juin <strong>1998</strong> <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 9807<br />
(74) SPIEGEL, Allen, J. et al. / etc.; Pfizer Inc., 235<br />
East 42nd Street, New York, NY 10017 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE HU ID IL<br />
IS JP KE KG KP KR KZ LC LK LR LS LT LU<br />
LV MD MG MK MN MW MX NO NZ PL PT RO<br />
RU SD SE SG SI SK TJ TM TR TT UA UG UZ<br />
VN YU; AP (GH KE LS MW SD SZ UG ZW);<br />
EA (AM AZ BY KG KZ MD RU TJ TM); EP (AT<br />
BE CH DE DK ES FI FR GB GR IE IT LU MC<br />
NL PT SE); OA (BF BJ CF CG CI CM GA GN<br />
ML MR NE SN TD TG).<br />
(11) WO 98/23604 (13) A1<br />
(21) <strong>PCT</strong>/JP97/04280<br />
(<strong>22</strong>) 21 Nov/nov 1997 (21.11.1997)<br />
(25) ja (26) ja<br />
(31) 8/334559 (32) 28 Nov/nov 1996 (33) JP<br />
(28.11.1996)<br />
(31) 9/286169 (32) 1 Oct/oct 1997 (33) JP<br />
(01.10.1997)<br />
(43) 4 Jun/juin <strong>1998</strong> (04.06.<strong>1998</strong>)<br />
(51) 6 C07D 317/34, A61K 47/26, C09K 3/00<br />
(54) SUGAR COMPOUNDS, GELLING AGENTS,<br />
GELLING AGENT COMPOSITIONS, PRO-<br />
CESSES FOR THE PREPARATION OF THEM,<br />
AND GEL COMPOSITIONS<br />
COMPOSITIONS DE SUCRE, AGENTS GELI-<br />
FIANTS, COMPOSITIONS D’AGENT GELI-<br />
FIANT, LEURS PROCEDES DE PREPARATION<br />
ET COMPOSITIONS DE GEL<br />
(71) NEW JAPAN CHEMICAL CO., LTD. [JP/JP];<br />
13, Yoshijima Yagura–cho, Fushimi–ku, Kyoto–shi,<br />
Kyoto 612 (JP).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) KOBAYASHI, Toshiaki [JP/JP]; 11–16, Suzaku<br />
5–chome, Nara–shi, Nara 631 (JP). ANDO,<br />
Kenshi [JP/JP]; Yuniraifu Ujikohata 605, 19–184,<br />
Kumakoji, Kohata, Uji–shi, Kyoto 611 (JP).<br />
NOMOTO, Harutomo [JP/JP]; Yasui Manshon<br />
B101, 366–1, Hizume–cho, Yodo, Fushimi–ku,<br />
Kyoto–shi, Kyoto 613 (JP).<br />
(74) SAEGUSA, Eiji et al. / etc.; Kitahama TNK Building,<br />
1–7–1, Dosho–machi, Chuo–ku, Osaka–shi,<br />
Osaka 541 (JP).<br />
(81) BR CA CN ID JP KR MX NO US; EP (AT BE<br />
CH DE DK ES FI FR GB GR IE IT LU MC NL<br />
PT SE).<br />
(11) WO 98/23605 (13) A1<br />
(21) <strong>PCT</strong>/EP97/06368<br />
(<strong>22</strong>) 14 Nov/nov 1997 (14.11.1997)<br />
(25) de (26) de<br />
(31) 196 49 093.6 (32) 27 Nov/nov 1996 (33) DE<br />
(27.11.1996)<br />
(43) 4 Jun/juin <strong>1998</strong> (04.06.<strong>1998</strong>)<br />
(51) 6 C07D 333/38, 413/12, A01N 43/10, 43/80<br />
(54) MICROBICIDAL AGENTS BASED ON<br />
THIOPHENE–2–CARBOXYLIC ACID DE-<br />
RIVATIVES<br />
MICROBICIDES A BASE DE DERIVES<br />
D’ACIDE THIOPHENE–2–CARBOXYLIQUE<br />
(71) BAYER AKTIENGESELLSCHAFT [DE/DE];<br />
D–51368 Leverkusen (DE).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) FISCHER, Reiner [DE/DE];<br />
Nelly–Schachs–Strasse 23, D–40789 Monheim<br />
(DE). LUI, Norbert [DE/DE]; Roggendorfstrasse<br />
55, D–51061 Köln (DE). DUTZMANN, Stefan<br />
[DE/DE]; Weißenstein 95, D–40764 Langenfeld<br />
(DE). HÄNSSLER, Gerd [DE/DE]; Am<br />
Arenzberg 85a, D–51381 Leverkusen (DE).<br />
(74) BAYER AKTIENGESELLSCHAFT; D–51368<br />
Leverkusen (DE).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH HU IL<br />
IS JP KE KG KP KR KZ LC LK LR LS LT LU<br />
LV MD MG MK MN MW MX NO NZ PL PT<br />
RO RU SD SE SG SI SK TJ TM TR TT UA UG<br />
US UZ VN YU; AP (GH KE LS MW SD SZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ TM);<br />
EP (AT BE CH DE DK ES FI FR GB GR IE IT<br />
LU MC NL PT SE); OA (BF BJ CF CG CI CM<br />
GA GN ML MR NE SN TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/23606 (13) A1<br />
(21) <strong>PCT</strong>/JP97/04281<br />
(<strong>22</strong>) 25 Nov/nov 1997 (25.11.1997)<br />
(25) ja (26) ja<br />
(31) 8/332941 (32) 27 Nov/nov 1996 (33) JP<br />
(27.11.1996)<br />
(31) 9/270394 (32) 16 Sep/sep 1997 (33) JP<br />
(16.09.1997)<br />
(43) 4 Jun/juin <strong>1998</strong> (04.06.<strong>1998</strong>)<br />
(51) 6 C07D 339/04, 339/08, 341/00, A61K 31/38<br />
(54) CYCLIC DITHIO DERIVATIVES, REME-<br />
DIES FOR DIABETIC KIDNEY DISEASES,<br />
HYPOGLYCEMIC AGENTS, HYPOLIPIDEMIC<br />
AGENTS, AND LENITIVES FOR DIGESTIVE<br />
DISORDERS<br />
DERIVES DITHIO CYCLIQUES, REMEDES<br />
CONTRE DES MALADIES RENALES DIA-<br />
BETIQUES, AGENTS HYPOGLYCEMIQUES,<br />
AGENTS HYPOLIPIDEMIQUES ET AGENTS<br />
LENITIFS CONTRE LES TROUBLES DIGES-<br />
TIFS<br />
(71) FUJI KAGAKU KOGYO KABUSHIKI KAI-<br />
SHA [JP/JP]; 55, Yokohoonji, Kamiichimachi, Nakaniikawa–gun,<br />
Toyama 930–03 (JP).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) KUROBE, Hiroshi [JP/JP]; Fuji Kagaku Kogyo<br />
Kabushiki Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP).<br />
NUNOZAWA, Tetsuji [JP/JP]; Fuji Kagaku Kogyo<br />
Kabushiki Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP). SU-<br />
GAWARA, Tomokazu [JP/JP]; Fuji Kagaku Kogyo<br />
Kabushiki Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP).<br />
KAWAI, Shinji [JP/JP]; Fuji Kagaku Kogyo Kabushiki<br />
Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP). KAWA-<br />
BATA, Hironori [JP/JP]; Fuji Kagaku Kogyo Kabushiki<br />
Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP). MATSU-<br />
TANI, Yoshihide [JP/JP]; Fuji Kagaku Kogyo Kabushiki<br />
Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP). TAKA-<br />
HASHI, Jiro [JP/JP]; Fuji Kagaku Kogyo Kabushiki<br />
Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP). MORI-<br />
GUCHI, Koei [JP/JP]; Fuji Kagaku Kogyo Kabushiki<br />
Kaisha, 55, Yokohoonji, Kamiichimachi,<br />
Nakaniikawa–gun, Toyama 930–03 (JP). ENDO,<br />
Takeshi [JP/JP]; Fuji Kagaku Kogyo Kabushiki<br />
Kaisha, 55, Yokohoonji, Kamiichimachi, Nakaniikawa–gun,<br />
Toyama 930–03 (JP).<br />
(74) KUZUWA, Kiyoshi et al. / etc.; Kuzuwa &<br />
Partner, Sogo Kojimachi Dai–ichi Building, 2,<br />
Kojimachi 3–chome, Chiyoda–ku, Tokyo 102 (JP).<br />
(81) CA CN JP KR US; EP (AT BE CH DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE).<br />
(11) WO 98/23607 (13) A1<br />
(21) <strong>PCT</strong>/JP97/04287<br />
(<strong>22</strong>) 25 Nov/nov 1997 (25.11.1997)<br />
(25) ja (26) ja<br />
(31) 8/328010 (32) 25 Nov/nov 1996 (33) JP<br />
(25.11.1996)<br />
(31) 9/323972 (32) 11 Nov/nov 1997 (33) JP<br />
(11.11.1997)<br />
(43) 4 Jun/juin <strong>1998</strong> (04.06.<strong>1998</strong>)<br />
(51) 6 C07D 401/12, 401/14, 211/90, 471/04, A61K<br />
31/445, 31/495, 31/535<br />
(54) 1,4–DIHYDROPYRIDINE DERIVATIVES<br />
DERIVES DE 1,4–DIHYDROPYRIDINE<br />
(71) NIKKEN CHEMICALS CO., LTD. [JP/JP];<br />
4–14, Tsukiji 5–chome, Chuo–ku, Tokyo 104 (JP).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) TASAKA, Shigeyuki [JP/JP]; Omiya Research<br />
Laboratory, Nikken Chemicals Co., Ltd., 346, Kitabukurocho<br />
1–chome, Omiya–shi, Saitama 330<br />
(JP). TANABE, Hirokazu [JP/JP]; Omiya Research<br />
Laboratory, Nikken Chemicals Co., Ltd.,<br />
346, Kitabukurocho 1–chome, Omiya–shi, Saitama<br />
330 (JP). OMORI, Hiromasa [JP/JP]; Omiya Research<br />
Laboratory, Nikken Chemicals Co., Ltd.,<br />
346, Kitabukurocho 1–chome, Omiya–shi, Saitama<br />
330 (JP). KIUE, Akira [JP/JP]; Omiya Research<br />
Laboratory, Nikken Chemicals Co., Ltd., 346, Kitabukurocho<br />
1–chome, Omiya–shi, Saitama 330 (JP).<br />
(74) ISHIDA, Takashi et al. / etc.; A. Aoki &<br />
Associates, Toranomon 37 Mori Building, 5–1,<br />
Toranomon 3–chome, Minato–ku, Tokyo 105 (JP).<br />
(81) CA US; EP (AT BE CH DE DK ES FI FR GB GR<br />
IE IT LU MC NL PT SE).<br />
(11) WO 98/23608 (13) A1<br />
(21) <strong>PCT</strong>/US97/21596<br />
(<strong>22</strong>) 26 Nov/nov 1997 (26.11.1997)<br />
(25) en (26) en<br />
(31) 60/033,208 (32) 27 Nov/nov 1996 (33) US<br />
(27.11.1996)<br />
(43) 4 Jun/juin <strong>1998</strong> (04.06.<strong>1998</strong>)<br />
(51) 6 C07D 401/12, A61K 31/395, C07D 215/56,<br />
413/14<br />
(54) NOVEL INTEGRIN RECEPTOR ANTAGONISTS<br />
NOUVEAUX ANTAGONISTES DES RECEP-<br />
TEURS DE L’INTEGRINE<br />
(71) THE DU PONT MERCK PHARMACEUTICAL<br />
COMPANY [US/US]; 1007 Market Street, Wilmington,<br />
DE 19898 (US).<br />
(72) WITYAK, John; 127 Kelton Road, West Grove,<br />
PA 19390 (US). TOBIN, Aleksandra, Ewa; 498<br />
Lewisville Road, Lincoln University, PA 19352<br />
(US).<br />
(74) LARSEN, Scott, K.; The Du Pont Merck Pharmaceutical<br />
Company, Legal/Patent Records Center,<br />
1007 Market Street, Wilmington, DE 19898 (US).<br />
(81) AU CA IL JP MX NZ; EP (AT BE CH DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE).<br />
Published / Publiée : (c)<br />
(11) WO 98/23609 (13) A1<br />
(21) <strong>PCT</strong>/US97/20551<br />
(<strong>22</strong>) 21 Nov/nov 1997 (21.11.1997)<br />
(25) en (26) en<br />
(31) 60/031,740 (32) 25 Nov/nov 1996<br />
(25.11.1996)<br />
(43) 4 Jun/juin <strong>1998</strong> (04.06.<strong>1998</strong>)<br />
(33) US