PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO

21/2001
8694 PCT Gazette - Section I - Gazette du PCT 25 May/mai 2001
PROCEDE DE FABRICATION, ET
UTILISATION EN TANT QUE MEDI-
CAMENT
(71) BOEHRINGER INGELHEIM PHARMA
KG [DE/DE]; 55216 Ingelheim am Rhein
(DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) ANDERSKEWITZ, Ralf [DE/DE];
Stromberger Strasse 36c, 55411 Bingen
(DE). BRAUN, Christine [DE/CH]; Via
Fabrizia, 22, CH-6512 Giubiasco (CH).
HAMM, Rainer [DE/DE]; In der Bitz 20,
55218 Ingelheim am Rhein (DE). DISSE,
Bernd [DE/DE]; Liebermannstrasse 7, 55127
Mainz (DE). JENNEWEIN, Hans, Michael
[DE/DE]; Idsteiner Strasse 14, 65193 Wiesbaden
(DE). SPECK, Georg [DE/DE]; In
der Bitz 10, 55218 Ingelheim (DE).
(74) LAUDIEN, Dieter; Boehringer Ingelheim
GmbH, 55216 Ingelheim am Rhein (DE).
(81) AE AU BG BR CA CN CZ EE HU ID IL IN
JP KR LT LV MX NO NZ PL RO SG SI SK
UA US UZ VN YU ZA.
(84) EA (AM AZ BY KG KZ MD RU TJ TM); EP
(ATBECHCYDEDKESFIFRGBGRIE
IT LU MC NL PT SE TR).
(51) 7 C07C 217/60, 217/62, 217/72, C07D
209/14, 213/61, A61K 31/135, 31/44, 31/415
(11) WO 01/36375
(21) PCT/JP00/08007
(13) A1
(22) 13 Nov/nov 2000 (13.11.2000)
(25) en (26) en
(30) PQ 4076 16 Nov/nov 1999
(16.11.1999)
AU
(43) 25 May/mai 2001 (25.05.2001)
(54) • AMINOALCOHOL DERIVATIVES
USEFUL FOR THE TREATMENT OF
GASTROINTESTINAL DISORDERS
• DÉRIVÉS D’AMINO ALCOOLS
UTILES POUR LE TRAITEMENT DE
TROUBLES GASTRO-INTESTINAUX
(71) FUJISAWA PHARMACEUTICAL CO.,
LTD. [JP/JP]; 4-7, Doshomachi 3-chome,
Chuo-ku, Osaka-shi, Osaka 541-8514 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) TANIGUCHI, Kiyoshi [JP/JP]; Fujisawa
Pharmaceutical Co., Ltd., 4-7,
Doshomachi 3-chome, Chuo-ku, Osaka-shi,
Osaka 541-8514 (JP). KAYAKIRI, Hiroshi
[JP/JP]; Fujisawa Pharmaceutical Co.,
Ltd., 4-7, Doshomachi 3-chome, Chuo-ku,
Osaka-shi, Osaka 541-8514 (JP). FUJII,
Naoaki [JP/JP]; Fujisawa Pharmaceutical
Co., Ltd., 4-7, Doshomachi 3-chome,
Chuo-ku, Osaka-shi, Osaka 541-8514
(JP). HAMASHIMA, Hitoshi [JP/JP];
Fujisawa Pharmaceutical Co., Ltd., 4-7,
Doshomachi 3-chome, Chuo-ku, Osaka-shi,
Osaka 541-8514 (JP). SAKURAI, Minoru
[JP/JP]; Fujisawa Pharmaceutical
Co., Ltd., 4-7, Doshomachi 3-chome,
Chuo-ku, Osaka-shi, Osaka 541-8514
(JP). WASHIZUKA, Kenichi [JP/JP];
Fujisawa Pharmaceutical Co., Ltd., 4-7,
Doshomachi 3-chome, Chuo-ku, Osaka-shi,
Osaka 541-8514 (JP). TOMISHIMA, Yasuyo
[JP/JP]; Fujisawa Pharmaceutical Co.,
Ltd., 4-7, Doshomachi 3-chome, Chuo-ku,
Osaka-shi, Osaka 541-8514 (JP). HAMADA,
Kaori [JP/JP]; Fujisawa Pharmaceutical
Co., Ltd., 4-7, Doshomachi 3-chome,
Chuo-ku, Osaka-shi, Osaka 541-8514 (JP).
YAMAMOTO, Nobuhiro [JP/JP]; Fujisawa
Pharmaceutical Co., Ltd., 4-7, Doshomachi
3-chome, Chuo-ku, Osaka-shi, Osaka
541-8514 (JP). ISHIKAWA, Hirofumi
[JP/JP]; Fujisawa Pharmaceutical Co., Ltd.,
4-7, Doshomachi 3-chome, Chuo-ku, Osaka-shi,
Osaka 541-8514 (JP). TANIMURA,
Naoko [JP/JP]; Fujisawa Pharmaceutical Co.,
Ltd., 4-7, Doshomachi 3-chome, Chuo-ku,
Osaka-shi, Osaka 541-8514 (JP).
(74) TAKASHIMA, Hajime; Yuki Bldg., 3-9,
Hiranomachi 3-chome, Chuo-ku, Osaka-shi,
Osaka 541-0046 (JP).
(81) JP US.
(84) EP (AT BE CH CY DE DK ES FI FR GB GR
IE IT LU MC NL PT SE TR).
Published / Publiée :(c)
(51) 7 C07C 233/47, 233/63, 233/81, 275/42,
311/08, 311/21, 335/22, C07D 295/18,
207/12, 211/62, 207/14, 207/16, 211/42,
211/46, 207/08, 487/08, 207/09, 265/30,
309/08, 211/22, 223/06, 207/20, 491/08,
495/08, 217/06, 471/08, 405/06, 239/38,
285/06, 239/42, A61K 31/198, 31/40,
31/495, 31/5375, 31/54, 31/445, 31/55,
31/407, 31/4025, 31/0015, 31/472, 31/4375,
31/351, 31/403, A61P 43/00, 29/00, 19/02,
1/04, 11/06, 17/06, 37/08, 3/10, 9/00, 9/10,
35/00, 35/04, 37/06
(11) WO 01/36376 (13) A1
(21) PCT/JP00/08152
(22) 20 Nov/nov 2000 (20.11.2000)
(25) ja (26) ja
(30) 11/328468 18 Nov/nov 1999 JP
(18.11.1999)
(30) 2000-197139 29 Jun/juin 2000 JP
(29.06.2000)
(43) 25 May/mai 2001 (25.05.2001)
(54) • NOVEL PHENYLALANINE DERIVA-
TIVES
• NOUVEAUX DÉRIVÉSDELAPHÉNY-
LALANINE
(71) AJINOMOTO CO., INC. [JP/JP]; 15-1, Kyobashi
1-Chome, Chuo-Ku, Tokyo 104-0031
(JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) TANAKA, Yasuhiro [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
YOSHIMURA, Toshihiko [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
IZAWA, Hiroyuki [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
EJIMA, Chieko [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
KOJIMA, Mitsuhiko [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
SATAKE, Yuko [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
NAKANISHI, Eiji [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
SUZUKI, Nobuyasu [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
MAKINO, Shingo [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
SUZUKI, Manabu [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
MURATA, Masahiro [JP/JP]; Pharmaceutical
Research Laboratories, Ajinomoto
Co., Inc., 1-1, Suzuki-Cho, Kawasaki-Ku,
Kawasaki-Shi, Kanagawa 210-0801 (JP).
(74) NAKAMURA, Minoru et al. / etc.; Room
646, Shin-Tokyo Bldg, 3-1, Marunouchi
3-Chome,
(JP).
Chiyoda-Ku, Tokyo 100-8355
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07C 249/02, 251/20
(11) WO 01/36377
(21) PCT/EP00/10970
(13) A1
(22) 7 Nov/nov 2000 (07.11.2000)
(25) en (26) en
(30) 99811055.5 16 Nov/nov 1999
(16.11.1999)
EP
(43) 25 May/mai 2001 (25.05.2001)
(54) • PROCESS FOR THE PREPARATION OF
KETIMINES
• PROCEDE DE PREPARATION DE CE-
TIMINES
(71) CIBA SPECIALTY CHEMICALS
HOLDING INC. [CH/CH]; Klybeckstrasse
141, CH-4057 Basel (CH).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) THOMMEN, Marc [CH/CH]; Steinackerweg
12, CH-3125 Toffen (CH). HAFNER,
Andreas [CH/CH]; Balkenweg 23, CH-4460
Gelterkinden (CH). KOLLY, Roman
[CH/CH]; Baselmattweg 167, CH-4123
Allschwil (CH). KIRNER, Hans-Jörg
[DE/CH]; Wartenbergstrasse 35, CH-4133
Pratteln (CH). BRUNNER, Frédéric
[CH/CH]; Les Esserts 44, CH-2054 Chézard
(CH).