PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO
PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO
PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO
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<strong>21</strong>/<strong>2001</strong><br />
25 May/mai <strong>2001</strong> <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 8703<br />
(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />
(54) • ANTITHROMBOTIC AGENTS<br />
• AGENTS ANTITHROMBOTIQUES<br />
(71) ELI LILLY AND COMPANY [US/US];<br />
Lilly Corporate Center, Indianapolis, IN<br />
46285 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) MCCOWAN, Jefferson, Ray [US/US];<br />
2653 Crescent Hill Lane, Indianapolis, IN<br />
46208 (US). SALL, Daniel, Jon [US/US];<br />
376 Leisure Lane, Greenwood, IN 46142<br />
(US). TOTH, John, Eldon [US/US]; 6759<br />
Perrier Court, Indianapolis, IN 46278 (US).<br />
(74) ANDERSON, Arvie, J. et al. / etc.; Eli Lilly<br />
and Company, Lilly Corporate Center, Indianapolis,<br />
IN 46285 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ VN<br />
YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 417/12, A01N 43/82<br />
(11) WO 01/36415 (13) A1<br />
(<strong>21</strong>) <strong>PCT</strong>/EP00/11387<br />
(22) 16 <strong>No</strong>v/nov 2000 (16.11.2000)<br />
(25) en (26) en<br />
(30) <strong>21</strong>07/99 18 <strong>No</strong>v/nov 1999 CH<br />
(18.11.1999)<br />
(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />
(54) • PESTICIDAL AMINOHETEROCY-<br />
CLAMIDE COMPOUNDS<br />
• COMPOSES PESTICIDES AMINOHE-<br />
TEROCYCLAMIDE<br />
(71) NOVARTIS AG [CH/CH]; Schwarzwaldallee<br />
<strong>21</strong>5, CH-4058 Basel (CH).<br />
(for all designated States except / pour tous<br />
les États désignés sauf AT US)<br />
(71) NOVARTIS-ERFINDUNGEN VER-<br />
WALTUNGSGESELLSCHAFT M.B.H.<br />
[AT/AT]; Brunner Strasse 59, A-1230 Vienna<br />
(AT).<br />
(only for / seulement pour AT)<br />
(72, 75) DUCRAY, Pierre [FR/FR]; 15A, rue de<br />
Huningue, F-68300 Saint-Louis (FR). BOU-<br />
VIER, Jacques [CH/CH]; Rue des Parcs<br />
2, CH-2000 Neuchatel (CH). MÜLLER,<br />
Urs [CH/CH]; Drosselstrasse 6, CH-4142<br />
Münchenstein (CH).<br />
(74) BECKER, Konrad; <strong>No</strong>vartis AG, Corporate<br />
Intellectual Property, Patent & Trademark Department,<br />
CH-4002 Basel (CH).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ VN<br />
YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 417/12, A61K 31/427, 31/505, A61P<br />
31/10 // (C07D 417/12, <strong>21</strong>7:34, 239:00)<br />
(11) WO 01/36416 (13) A1<br />
(<strong>21</strong>) <strong>PCT</strong>/ES00/00432<br />
(22) 15 <strong>No</strong>v/nov 2000 (15.11.2000)<br />
(25) es (26) es<br />
(30) P 9902533 18 <strong>No</strong>v/nov 1999 ES<br />
(18.11.1999)<br />
(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />
(54) • NOVEL THIAZOLIDINEDIONE<br />
DERIVATIVES AS ANTIDIABETIC<br />
AGENTS<br />
• NOUVEAUX DERIVES DE THIA-<br />
ZOLIDINDIONE UTILISES COMME<br />
AGENTS ANTIDIABETIQUES<br />
(71) VITA-INVEST, S. A. [ES/ES]; C. Fontsanta,<br />
12-14, E-08970 Sant Joan Despi (ES).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) MOURELLE MANCINI, Marisabel<br />
[ES/ES]; Avenida Xile, 28, E-08028<br />
Barcelona (ES). DEL CASTILLO NIETO,<br />
Juan Carlos [ES/ES]; C. Castillejos, 389,<br />
E-08025 Barcelona (ES). DE RAMON<br />
AMAT, Elisabet [ES/ES]; C. Poesía, 11,<br />
E-08035 Barcelona (ES).<br />
(74) PONTI SALES, Adelaida et al. / etc.; C.<br />
Consell de Cent, 322, E-08007 Barcelona<br />
(ES).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ VN<br />
YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 451/04, 453/02, 453/06, 487/08,<br />
A61K 31/439, 31/46, 31/40, A61P 25/00<br />
(11) WO 01/36417<br />
(<strong>21</strong>) <strong>PCT</strong>/SE00/02262<br />
(13) A1<br />
(22) 16 <strong>No</strong>v/nov 2000 (16.11.2000)<br />
(25) en (26) en<br />
(30) 9904176-6 18 <strong>No</strong>v/nov 1999<br />
(18.11.1999)<br />
SE<br />
(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />
(54) • NEW USE AND NOVEL N-AZABICY-<br />
CLO-AMIDE DERIVATIVES<br />
• NOUVELLE UTILISATION ET NOU-<br />
VEAUX DERIVES DE N-AZABICY-<br />
CLO-AMIDE<br />
(71) ASTRAZENECA AB [SE/SE]; S-151 85<br />
Södertälje (SE).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) BALESTRA, Michael [US/US]; AstraZeneca<br />
US, 1800 Concord Pike, P.O.<br />
Box 15437, Wilmington, DE 19850-5437<br />
(US). MULLEN, George [US/US]; AstraZeneca<br />
R & D Boston, 35 Gatehouse Drive,<br />
Waltham, MA 02451 (US). PHILLIPS,<br />
Eifion [GB/US]; AstraZeneca US, 1800<br />
Concord Pike, P.O. Box 15437, Wilmington,<br />
DE 19850-5437 (US). SCHMIESING,<br />
Richard [US/US]; AstraZeneca US, 1800<br />
Concord Pike, P.O. Box 15437, Wilmington,<br />
DE 19850-5437 (US).<br />
(74) ASTRAZENECA AB; Global Intellectual<br />
Property, S-151 85 Södertälje (SE).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ VN<br />
YU ZA ZW.<br />
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />
UG ZW); EA (AM AZ BY KG KZ MD RU<br />
TJ TM); EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE TR); OA<br />
(BF BJ CF CG CI CM GA GN GW ML MR<br />
NE SN TD TG).<br />
(51) 7 C07D 471/10, A61K 31/445<br />
(11) WO 01/36418 (13) A1<br />
(<strong>21</strong>) <strong>PCT</strong>/DK00/00641<br />
(22) 17 <strong>No</strong>v/nov 2000 (17.11.2000)<br />
(25) en (26) en<br />
(30) PA 1999 01653 17 <strong>No</strong>v/nov 1999 DK<br />
(17.11.1999)<br />
(30) 60/167,819 29 <strong>No</strong>v/nov 1999 US<br />
(29.11.1999)<br />
(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />
(54) • NOVEL TRIAZASPIRODECANONES<br />
WITH HIGH AFFINITY FOR OPIOID<br />
RECEPTOR SUBTYPES<br />
• NOUVELLES TRIAZASPIRODECA-<br />
NONES A AFFINITE ELEVEE POUR<br />
DES SOUSTYPES DE RECEPTEURS<br />
OPIOIDES<br />
(71) NOVO NORDISK A/S [DK/DK]; <strong>No</strong>vo<br />
Allé, DK-2880 Bagsværd (DK).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) HOHLWEG, Rolf [DE/DK]; Nybovej<br />
6, DK-3490 Kvistgaard (DK). WATSON,<br />
Brett [US/DK]; Vildrosevej 17, Hareskovby,<br />
DK-3500 Værløse (DK). PETTERSSON,<br />
Ingrid [SE/DK]; Grundtvigsvej 18, 2th,<br />
DK-1864 Frederiksberg (DK).<br />
(74) NOVO NORDISK A/S; Corporate Patents,<br />
<strong>No</strong>vo Allé, DK-2880 Bagsværd (DK).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY BZ CA CH CN CR CU CZ DE DK DM<br />
DZ EE ES FI GB GD GE GH GM HR HU<br />
ID IL IN IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MA MD MG MK MN MW<br />
MX MZ NO NZ PL PT RO RU SD SE SG SI