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PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO

PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO

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<strong>21</strong>/<strong>2001</strong><br />

25 May/mai <strong>2001</strong> <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 8703<br />

(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />

(54) • ANTITHROMBOTIC AGENTS<br />

• AGENTS ANTITHROMBOTIQUES<br />

(71) ELI LILLY AND COMPANY [US/US];<br />

Lilly Corporate Center, Indianapolis, IN<br />

46285 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) MCCOWAN, Jefferson, Ray [US/US];<br />

2653 Crescent Hill Lane, Indianapolis, IN<br />

46208 (US). SALL, Daniel, Jon [US/US];<br />

376 Leisure Lane, Greenwood, IN 46142<br />

(US). TOTH, John, Eldon [US/US]; 6759<br />

Perrier Court, Indianapolis, IN 46278 (US).<br />

(74) ANDERSON, Arvie, J. et al. / etc.; Eli Lilly<br />

and Company, Lilly Corporate Center, Indianapolis,<br />

IN 46285 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07D 417/12, A01N 43/82<br />

(11) WO 01/36415 (13) A1<br />

(<strong>21</strong>) <strong>PCT</strong>/EP00/11387<br />

(22) 16 <strong>No</strong>v/nov 2000 (16.11.2000)<br />

(25) en (26) en<br />

(30) <strong>21</strong>07/99 18 <strong>No</strong>v/nov 1999 CH<br />

(18.11.1999)<br />

(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />

(54) • PESTICIDAL AMINOHETEROCY-<br />

CLAMIDE COMPOUNDS<br />

• COMPOSES PESTICIDES AMINOHE-<br />

TEROCYCLAMIDE<br />

(71) NOVARTIS AG [CH/CH]; Schwarzwaldallee<br />

<strong>21</strong>5, CH-4058 Basel (CH).<br />

(for all designated States except / pour tous<br />

les États désignés sauf AT US)<br />

(71) NOVARTIS-ERFINDUNGEN VER-<br />

WALTUNGSGESELLSCHAFT M.B.H.<br />

[AT/AT]; Brunner Strasse 59, A-1230 Vienna<br />

(AT).<br />

(only for / seulement pour AT)<br />

(72, 75) DUCRAY, Pierre [FR/FR]; 15A, rue de<br />

Huningue, F-68300 Saint-Louis (FR). BOU-<br />

VIER, Jacques [CH/CH]; Rue des Parcs<br />

2, CH-2000 Neuchatel (CH). MÜLLER,<br />

Urs [CH/CH]; Drosselstrasse 6, CH-4142<br />

Münchenstein (CH).<br />

(74) BECKER, Konrad; <strong>No</strong>vartis AG, Corporate<br />

Intellectual Property, Patent & Trademark Department,<br />

CH-4002 Basel (CH).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07D 417/12, A61K 31/427, 31/505, A61P<br />

31/10 // (C07D 417/12, <strong>21</strong>7:34, 239:00)<br />

(11) WO 01/36416 (13) A1<br />

(<strong>21</strong>) <strong>PCT</strong>/ES00/00432<br />

(22) 15 <strong>No</strong>v/nov 2000 (15.11.2000)<br />

(25) es (26) es<br />

(30) P 9902533 18 <strong>No</strong>v/nov 1999 ES<br />

(18.11.1999)<br />

(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />

(54) • NOVEL THIAZOLIDINEDIONE<br />

DERIVATIVES AS ANTIDIABETIC<br />

AGENTS<br />

• NOUVEAUX DERIVES DE THIA-<br />

ZOLIDINDIONE UTILISES COMME<br />

AGENTS ANTIDIABETIQUES<br />

(71) VITA-INVEST, S. A. [ES/ES]; C. Fontsanta,<br />

12-14, E-08970 Sant Joan Despi (ES).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) MOURELLE MANCINI, Marisabel<br />

[ES/ES]; Avenida Xile, 28, E-08028<br />

Barcelona (ES). DEL CASTILLO NIETO,<br />

Juan Carlos [ES/ES]; C. Castillejos, 389,<br />

E-08025 Barcelona (ES). DE RAMON<br />

AMAT, Elisabet [ES/ES]; C. Poesía, 11,<br />

E-08035 Barcelona (ES).<br />

(74) PONTI SALES, Adelaida et al. / etc.; C.<br />

Consell de Cent, 322, E-08007 Barcelona<br />

(ES).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07D 451/04, 453/02, 453/06, 487/08,<br />

A61K 31/439, 31/46, 31/40, A61P 25/00<br />

(11) WO 01/36417<br />

(<strong>21</strong>) <strong>PCT</strong>/SE00/02262<br />

(13) A1<br />

(22) 16 <strong>No</strong>v/nov 2000 (16.11.2000)<br />

(25) en (26) en<br />

(30) 9904176-6 18 <strong>No</strong>v/nov 1999<br />

(18.11.1999)<br />

SE<br />

(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />

(54) • NEW USE AND NOVEL N-AZABICY-<br />

CLO-AMIDE DERIVATIVES<br />

• NOUVELLE UTILISATION ET NOU-<br />

VEAUX DERIVES DE N-AZABICY-<br />

CLO-AMIDE<br />

(71) ASTRAZENECA AB [SE/SE]; S-151 85<br />

Södertälje (SE).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) BALESTRA, Michael [US/US]; AstraZeneca<br />

US, 1800 Concord Pike, P.O.<br />

Box 15437, Wilmington, DE 19850-5437<br />

(US). MULLEN, George [US/US]; AstraZeneca<br />

R & D Boston, 35 Gatehouse Drive,<br />

Waltham, MA 02451 (US). PHILLIPS,<br />

Eifion [GB/US]; AstraZeneca US, 1800<br />

Concord Pike, P.O. Box 15437, Wilmington,<br />

DE 19850-5437 (US). SCHMIESING,<br />

Richard [US/US]; AstraZeneca US, 1800<br />

Concord Pike, P.O. Box 15437, Wilmington,<br />

DE 19850-5437 (US).<br />

(74) ASTRAZENECA AB; Global Intellectual<br />

Property, S-151 85 Södertälje (SE).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 C07D 471/10, A61K 31/445<br />

(11) WO 01/36418 (13) A1<br />

(<strong>21</strong>) <strong>PCT</strong>/DK00/00641<br />

(22) 17 <strong>No</strong>v/nov 2000 (17.11.2000)<br />

(25) en (26) en<br />

(30) PA 1999 01653 17 <strong>No</strong>v/nov 1999 DK<br />

(17.11.1999)<br />

(30) 60/167,819 29 <strong>No</strong>v/nov 1999 US<br />

(29.11.1999)<br />

(43) 25 May/mai <strong>2001</strong> (25.05.<strong>2001</strong>)<br />

(54) • NOVEL TRIAZASPIRODECANONES<br />

WITH HIGH AFFINITY FOR OPIOID<br />

RECEPTOR SUBTYPES<br />

• NOUVELLES TRIAZASPIRODECA-<br />

NONES A AFFINITE ELEVEE POUR<br />

DES SOUSTYPES DE RECEPTEURS<br />

OPIOIDES<br />

(71) NOVO NORDISK A/S [DK/DK]; <strong>No</strong>vo<br />

Allé, DK-2880 Bagsværd (DK).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) HOHLWEG, Rolf [DE/DK]; Nybovej<br />

6, DK-3490 Kvistgaard (DK). WATSON,<br />

Brett [US/DK]; Vildrosevej 17, Hareskovby,<br />

DK-3500 Værløse (DK). PETTERSSON,<br />

Ingrid [SE/DK]; Grundtvigsvej 18, 2th,<br />

DK-1864 Frederiksberg (DK).<br />

(74) NOVO NORDISK A/S; Corporate Patents,<br />

<strong>No</strong>vo Allé, DK-2880 Bagsværd (DK).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI

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