PCT/2001/21 : PCT Gazette, Weekly Issue No. 21, 2001 - WIPO

21/2001
8700 PCT Gazette - Section I - Gazette du PCT 25 May/mai 2001
(22) 20 Oct/oct 2000 (20.10.2000)
(25) de (26) de
(30) A 1914/99 15 Nov/nov 1999 AT
(15.11.1999)
(30) A 46/2000 14 Jan/jan 2000 AT
(14.01.2000)
(43) 25 May/mai 2001 (25.05.2001)
(54) • METHOD FOR PRODUCING
2-CHLORO-5-CHLOROMETHYL-1,3-
THIAZOL
• PROCEDE DE PRODUCTION
DE 2-CHLORO-5-CHLOROME-
THYL-1,3-THIAZOL
(71) DSM FINE CHEMICALS AUSTRIA
GMBH [AT/AT]; St. Peterstrasse 25, A-4021
Linz (AT).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) HENDEL, Wolfram [AT/AT]; Gaumbergstrasse
82, A-4060 Leonding (AT).
KRICH, Silvia [AT/AT]; Raiffeisenweg
24/5, A-4203 Altenberg/Linz (AT).
(74) KLOSTERMANN, Ingrid; DSM Fine
Chemicals Austria GmbH, St. Peterstrasse
25, A-4021 Linz (AT).
(81) AE AG AL AM AU AZ BA BB BG BR BY
BZ CA CN CR CU CZ DM DZ EE GD GE
HR HU ID IL IN IS JP KG KP KR KZ LC LK
LR LT LV MA MD MG MK MN MX NO NZ
PL RO RU SG SI SK SL TJ TM TR TT UA
UG US UZ VN YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE); OA (BF
BJ CF CG CI CM GA GN GW ML MR NE
SN TD TG).
(51) 7 C07D 277/34, A61K 31/425
(11) WO 01/36401 (13) A1
(21) PCT/US00/31705
(22) 17 Nov/nov 2000 (17.11.2000)
(25) en (26) en
(30) 60/166,515 19 Nov/nov 1999 US
(19.11.1999)
(43) 25 May/mai 2001 (25.05.2001)
(54) • SOLID STATE FORMS OF 5-[[6-[(2-
FLUOROPHENYL)METHOXY]-2-
NAPHTHALENYL]METHYL]-2,4-THI-
AZOLIDINEDIONE
• FORMES A L’ETAT SOLIDE DE
5-[[6-[(2-FLUOROPHENYL)ME-
THOXY]-2-NAPHTALENYL]ME-
THYL]-2,4-THIAZOLIDINEDIONE
(71) ORTHO-MCNEIL PHARMACEUTI-
CAL, INC. [US/US]; U.S. Route #202, P.O.
Box 300, Raritan, NJ 08869-0602 (US).
(72) ANDRES, Mark, C.; 1315 El Prado Road,
Lafayette, IN 47905 (US). BRYN, Stephen,
R.; 824 Barrow Street, Lafayette, IN 47906
(US). NEWMAN, Ann, W.; 615 South 7th
Street, Lafayette, IN 47905 (US). RUS-
SELL, Catherine; 2018 Winflower Place,
West Lafayette, IN 47906 (US).
(74) JOHNSON, Philip, S. et al. / etc.; Johnson &
Johnson, One Johnson & Johnson Plaza, New
Brunswick, NJ 08933 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI
FR GB GR IE IT LU MC NL PT SE TR); OA
(BF BJ CF CG CI CM GA GN GW ML MR
NE SN TD TG).
(51) 7 C07D 277/38, 277/64, 277/66, 277/68,
277/70, 277/82, 417/10, 417/12, A61K
31/425, 31/427, 31/428, 31/4439, A61P 3/06,
43/00
(11) WO 01/36402 (13) A1
(21) PCT/JP99/06352
(22) 12 Nov/nov 1999 (12.11.1999)
(25) ja (26) ja
(43) 25 May/mai 2001 (25.05.2001)
(54) • NOVEL 2-(N-CYANOIMINO)THIAZO-
LIDIN-4-ONE DERIVATIVES
• NOUVEAUX DERIVES DE 2-(N-
CYANO-IMINO)THIAZOLIDIN-4-ONE
(71) FUJIMOTO BROTHERS CO., LTD.
[JP/JP]; 3-40, Nishiotsuka 1-chome, Matsubara-shi,
Osaka 580-0011 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) YONEDA, Fumio [JP/JP]; c/o Soyaku
Kenkyusyo, Fujimoto Pharmaceutical
Co., Ltd., 3-40, Nishiotsuka 1-chome, Matsubara-shi,
Osaka 580-0011 (JP). OHDE,
Hironori [JP/JP]; c/o Soyaku Kenkyusyo,
Fujimoto Pharmaceutical Co., Ltd., 3-40,
Nishiotsuka 1-chome, Matsubara-shi, Osaka
580-0011 (JP). WATANABE, Mayumi
[JP/JP]; c/o Soyaku Kenkyusyo, Fujimoto
Pharmaceutical Co., Ltd., 3-40, Nishiotsuka
1-chome, Matsubara-shi, Osaka 580-0011
(JP). ANDO, Takashi [JP/JP]; c/o Soyaku
Kenkyusyo, Fujimoto Pharmaceutical Co.,
Ltd., 3-40, Nishiotsuka 1-chome, Matsubara-shi,
Osaka 580-0011 (JP). YASUSA,
Takuya [JP/JP]; c/o Soyaku Kenkyusyo,
Fujimoto Pharmaceutical Co., Ltd., 3-40,
Nishiotsuka 1-chome, Matsubara-shi, Osaka
580-0011 (JP). UEGAKI, Yuko [JP/JP]; c/o
Soyaku Kenkyusyo, Fujimoto Pharmaceutical
Co., Ltd., 3-40, Nishiotsuka 1-chome,
Matsubara-shi, Osaka 580-0011 (JP).
(74) FUJIMOTO BROTHERS CO., LTD.;
3-40, Nishiotsuka 1-chome, Matsubara-shi,
Osaka 580-0011 (JP).
(81) AL AM AT AU AZ BA BB BG BR BY CA
CH CN CU CZ DE DK EE ES FI GB GD GE
GH GM HR HU ID IL IN IS JP KE KG KP
KR KZ LC LK LR LS LT LU LV MD MG
MK MN MW MX NO NZ PL PT RO RU SD
SE SG SI SK SL TJ TM TR TT UA UG US
UZ VN YU ZW.
(84) AP (GH GM KE LS MW SD SL SZ TZ UG
ZW); EA (AM AZ BY KG KZ MD RU TJ
TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF
BJ CF CG CI CM GA GN GW ML MR NE
SN TD TG).
(51) 7 C07D 295/08, A61P 29/00, C07D 213/73,
295/12, 213/63
(11) WO 01/36403 (13) A1
(21) PCT/US00/31582
(22) 16 Nov/nov 2000 (16.11.2000)
(25) en (26) en
(30) 60/165,903 16 Nov/nov 1999 US
(16.11.1999)
(43) 25 May/mai 2001 (25.05.2001)
(54) • UREA DERIVATIVES AS ANTI-IN-
FLAMMATORY AGENTS
• DERIVES D’UREE UTILISES COMME
AGENTS ANTI-INFLAMMATOIRES
(71) BOEHRINGER INGELHEIM PHAR-
MACEUTICALS, INC. [US/US]; 900
Ridgebury Road, Ridgefield, CT 06877 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BREITFELDER, Steffen [DE/US];
93 Park Avenue, #1305, Danbury, CT 06810
(US). CIRILLO, Pier, F. [IT/US]; 180 Washington
Road, Woodbury, CT 06798 (US).
HAO, Ming-Hong [US/US]; 11 Scodon
Drive, Ridgefield, CT 06877 (US). HICKEY,
Eugene, R. [US/US]; 5 Woodbury Drive,
Danbury, CT 06811 (US). SHARMA, Rajiv
[IN/US]; 37 Midrocks Road, Ridgefield, CT
06877 (US). SUN, Sanxing [CN/US]; 38
Padanaram Avenue, 21B, Danbury, CT 06811
(US). TAKAHASHI, Hidenori [JP/US];
68 Ehmer Drive, LaGrangeville, NY 12540
(US).
(74) RAYMOND, Robert et al. / etc.; Boehringer
Ingelheim Pharmaceuticals, Inc., 900 Ridgebury
Road, P.O. Box 368, Ridgefield, CT
06877 (US).
(81) AE AU BG BR BY CA CN CZ EE HR HU
ID IL IN JP KR KZ LT LV MX NO NZ PL RO
RU SG SI SK TR UA US UZ VN YU ZA.
(84) EP (AT BE CH CY DE DK ES FI FR GB GR
IE IT LU MC NL PT SE TR).
Published / Publiée :(c)
(51) 7 C07D 295/215, A61K 31/165
(11) WO 01/36404
(21) PCT/US00/31580
(13) A1
(22) 17 Nov/nov 2000 (17.11.2000)
(25) en (26) en
(30) 60/166,555 19 Nov/nov 1999
(19.11.1999)
US
(43) 25 May/mai 2001 (25.05.2001)
(54) • COMPOUNDS AND METHODS
• COMPOSES ET PROCEDES
(71) SMITHKLINE BEECHAM CORPO-
RATION [US/US]; One Franklin
Philadelphia, PA 19103 (US).
Plaza,
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) MARINO, Joseph, P., Jr. [US/US]; 214
Rock Glen Road, Wynnewood, PA 19606
(US). RYAN, M., Dominic [CA/US]; 2146
Foxtail Drive, Pottstown, PA 19464 (US).
THOMPSON, Scott, Kevin [US/US]; 75
Guilford Circle, Phoenixville, PA 19460
(US). VEBER, Daniel, Frank [US/US]; 290
Batleson Road, Ambler, PA 19002 (US).
(74) STEIN-FERNANDEZ, Nora et al. / etc.;
SmithKline Beecham Corporation, Corporate
Intellectual Property, UW2220, 709 Swedeland
Road, P.O. Box 1539, King of Prussia,
PA 19406-0939 (US).