PCT/2001/12 : PCT Gazette, Weekly Issue No. 12, 2001 - WIPO

12/2001
4752 PCT Gazette - Section I - Gazette du PCT 22 Mar/mar 2001
(22) 13 Sep/sep 2000 (13.09.2000)
(25) en (26) en
(30) 60/153,236 13 Sep/sep 1999 US
(13.09.1999)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) AZACYCLOALKANONE SERINE
PROTEASE INHIBITORS
INHIBITEURS DE SERINE PROTEASE
AZACYCLOALCANONE
(71) 3-DIMENSIONAL PHARMACEUTI-
CALS, INC. [US/US]; Suite 104, 665
Stockton Drive, Eagleview Corporate Center,
Exton, PA 19341 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) MILLER, Scott, C. [US/US]; Apt.
D-233, 2450 Airport Road, Longmont, CO
80503 (US). MARUGÁN SÁNCHEZ,
Juan, José [ES/US]; 104 Coach Lane, Exton,
PA 19341 (US). HASLOW, Kristin,
D. [US/US]; 14 Ridgeview Road, Newtown
Square, PA 19073 (US). HALL, Jonathan,
P. [US/US]; 5795 Alpine Drive, Ontario, NY
14519 (US).
(74) COVERT, John, M. et al. / etc.; Sterne,
Kessler, Goldstein & Fox P.L.L.C., Suite 600,
1100 New York Avenue, Washington, DC
20005-3934 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 213/82, 213/81, 295/20, 333/40,
333/70, 209/08, 317/68, 215/54, 215/48,
C07C 317/28, A61K 31/5375, 31/5377,
31/455, 31/47, 31/4965, 31/381, A61P 19/02,
33/06
(11) WO 01/19796
(21) PCT/US00/25415
(13) A1
(22) 15 Sep/sep 2000 (15.09.2000)
(25) en (26) en
(30) 60/154,245 16 Sep/sep 1999
(16.09.1999)
US
(30) 60/171,831 22 Dec/déc 1999
(22.12.1999)
US
(30) 60/224,552 10 Aug/août 2000
(10.08.2000)
US
(43) 22 Mar/mar 2001 (22.03.2001)
(54) COMPOUNDS AND PHARMACEUTI-
CAL COMPOSITIONS AS CATHEPSIN
S INHIBITORS
COMPOSES ET COMPOSITIONS
PHARMACEUTIQUES UTILISES
COMME INHIBITEURS DE LA CA-
THEPSINE S
(71) AXYS PHARMACEUTICALS, INC.
[US/US]; 180 Kimball Way, South San Francisco,
CA 94080 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) GRAUPE, Michael [AT/US]; 2727 Edison
Street, Apt. 219, San Mateo, CA 94403
(US). LINK, John, O. [US/US]; 12 Prospect
Avenue, San Francisco, CA 94110 (US).
PATTERSON, John, W. [US/US]; 1619
Montalto Drive, Mountain View, CA 94040
(US). ZIPFEL, Sheila [US/US]; 380 Edlee
Avenue, Palo Alto, CA 94306 (US).
(74) MONTGOMERY, Wayne, W. et al. / etc.;
Axys Pharmaceuticals, Inc., 180 Kimball
Way, South San Francisco, CA 94080 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 223/00
(11) WO 01/19797 (13) A2
(21) PCT/US00/24967
(22) 13 Sep/sep 2000 (13.09.2000)
(25) en (26) en
(30) 60/153,511 13 Sep/sep 1999 US
(13.09.1999)
(30) 60/224,388 9 Aug/août 2000 US
(09.08.2000)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) HYDROXYALKANOYL AMINOLAC-
TAMS AND RELATED STRUCTURES
AS INHIBITORS OF Aβ PROTEIN PRO-
DUCTION
HYDROXYALKANOYL AMINOLAC-
TAMES ET STRUCTURES ASSOCIEES,
INHIBITEURS DE LA PRODUCTION
DE LA PROTEINE Aβ
(71) DU PONT PHARMACEUTICALS COM-
PANY [US/US]; Chestnut Run Plaza, 974
Centre Road, Wilmington, DE 19807 (US).
(72) OLSON, Richard, Eric; 7 Pelham Road,
Wilmington, DE 19803 (US). LIU, Hong;
6 Howe Court, Glen Mills, PA 18342 (US).
THOMPSON, Lorin, Andrew, III; 600 Silverside
Road, Wilmington, DE 19809 (US).
(74) LARSEN, Scott, K.; Du Pont Pharmaceuticals
Company, Legal Patent Records Center,
1007 Market Street, Wilmington, DE 19898
(US).
(81) AU BR CA CN CZ EE HU IL IN JP KR LT
LV MX NO NZ PL RO SG SI SK TR UA VN
ZA.
(84) EA (AM AZ BY KG KZ MD RU TJ TM); EP
(ATBECHCYDEDKESFIFRGBGRIE
IT LU MC NL PT SE).
(51) 7 C07D 231/00
(11) WO 01/19798 (13) A2
(21) PCT/US00/25195
(22) 15 Sep/sep 2000 (15.09.2000)
(25) en (26) en
(30) 60/154,332 17 Sep/sep 1999 US
(17.09.1999)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) INHIBITORS OF FACTOR Xa
INHIBITEURS DU FACTEUR Xa
(71) COR THERAPEUTICS INC. [US/US];
256 E. Grand Avenue, South San Francisco,
CA 94080 (US).
(72) ZHU, Bing-Yan; 3325 Adelaide Way, Belmont,
CA 94002 (US). JIA, Zhaozhong, Jon;
849 West Orange Avenue #2007, South San
Francisco, CA 94080 (US). HUANG, Wenrong;
7723 Huntridge Lane, Cupertino, CA
95014 (US). SONG, Yonghong; 1144 Nimitz
Lane, Foster City, CA 94404 (US). KAN-
TER, James; 132 Rosaflora Circle, South
San Francisco, CA 94080 (US). SCARBOR-
OUGH, Robert, M.; 22 Greenbrier Court,
Half Moon Bay, CA 94019 (US).
(74) LEE, Christine, S.; Morgan, Lewis & Bockius
LLP, 1800 M. Street, N.W., Washington,
DC 20036-5869 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 233/00
(11) WO 01/19799
(21) PCT/JP00/06226
(13) A2
(22) 12 Sep/sep 2000 (12.09.2000)
(25) en (26) en
(30) 11/259057 13 Sep/sep 1999
(13.09.1999)
JP
(30) 11/260315 14 Sep/sep 1999
(14.09.1999)
JP
(43) 22 Mar/mar 2001 (22.03.2001)
(54) NITROIMIDAZOLE DERIVATIVE AND
DIAGNOSTIC IMAGING AGENT CON-
TAINING THE SAME
DERIVE DE NITROIMIDAZOLE ET
AGENT D’IMAGERIE DIAGNOS-
TIQUE LE CONTENANT
(71) POLA CHEMICAL INDUSTRIES, INC.
[JP/JP]; 6-48, Yayoi-cho, Shizuoka-shi,
Shizuoka 420-0914 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(71, 72) TAKAI, Yoshihiro [JP/JP]; 2-14, Nijino-oka
3-chome, Izumi-ku, Sendai-shi,
Miyagi 981-8007 (JP). IDO, Tatsuo
[JP/JP]; 9-14, Miyagidai 3-chome, Aoba-ku,
Sendai-shi, Miyagi 989-3214 (JP).
(72, 75) TSUJITANI, Michihiko [JP/JP]; 12-1,
Futaba 2-chome, Yokosuka-shi, Kanagawa
239-0814 (JP).