PCT/2001/12 : PCT Gazette, Weekly Issue No. 12, 2001 - WIPO

12/2001
4760 PCT Gazette - Section I - Gazette du PCT 22 Mar/mar 2001
(71) NOVO NORDISK A/S [DK/DK]; Novo
Allé, DK-2880 Bagsvaerd (DK). ONTO-
GEN CORPORATION [US/US]; 6451 El
Camino Real, Carlsbad, CA 92009 (US).
(72) ANDERSEN, Henrik, Sune; Gustav
Adolphsvej 2, DK-2800 Lyngby (DK).
HANSEN, Thomas, Kruse; Tibbevangen
78, DK-2730 Herlev (DK). LAU, Jesper;
Dybedalsvej 27, DK-3520 Farum (DK).
MØLLER, Niels, Peter, Hundahl; Midtermolen
4, 3., DK-2100 Copenhagen Ø (DK).
OLSEN, Ole, Hvilsted; Bækkeskovvej 38,
DK-2700 Brønshøj (DK). AXE, Frank,
Urban; 1250 Birch Avenue, Escondido, CA
92027 (US). GE, Yu; 12455 Brickella Street,
San Diego, CA 92129 (US). HOLSWORTH,
Daniel, Dale; 9462 Chabola Road, San
Diego, CA 92129 (US). JONES, Todd,
Kevin; 546 Marview Drive, Solana Beach,
CA 92075 (US). JUDGE, Luke, Milburn;
644 ? Bonair Way, La Jolla, CA 92037
(US). RIPKA, Wiliam, Charles; 10819
Red Rock Drive, San Diego, CA 92131
(US). SHAPIRA, Barry, Zvi; 5925 La Jolla
Corona Drive, La Jolla, CA 92037 (US).
UYEDA, Roy, Teruyuki; 5385 Toscana
Way, Apt. 342, San Diego, CA 92122 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(c)
(51) 7 C07D 495/04, 513/04, 493/04, A61K
31/381, 31/395, A61P 3/00, 5/00, 7/00,
17/00, 19/00, 25/00, 31/00, 35/00, 37/00
(11) WO 01/19831
(21) PCT/DK00/00503
(13) A1
(22) 11 Sep/sep 2000 (11.09.2000)
(25) en (26) en
(30) PA 1999 01278 10 Sep/sep 1999
(10.09.1999)
DK
(43) 22 Mar/mar 2001 (22.03.2001)
(54) MODULATORS OF PROTEIN TYRO-
SINE PHOSPHATASES (PTPases)
MODULATEURS DE PROTEINES TY-
ROSINE PHOSPHATAGES (PTPases)
(71) NOVO NORDISK A/S [DK/DK]; Novo
Allé, DK-2880 Bagsvaerd (DK). ONTO-
GEN CORPORATION [US/US]; 6451 El
Camino Real, Carlsbad, CA 92009 (US).
(72) ANDERSEN, Henrik, Sune; Gustav
Adolphsvej 2, DK-2800 Lyngby (DK).
HANSEN, Thomas, Kruse; Tibbevangen
78, DK-2730 Herlev (DK). LAU, Jesper;
Dybedalsvej 27, DK-3520 Farum (DK).
MØLLER, Niels, Peter, Hundahl; Midtermolen
4, 3., DK-2100 Copenhagen Ø (DK).
OLSEN, Ole, Hvilsted; Bækkeskovvej 38,
DK-2700 Brønshøj (DK). AXE, Frank,
Urban; 1250 Birch Avenue, Escondido, CA
92027 (US). GE, Yu; 12455 Brickella Street,
San Diego, CA 92129 (US). HOLSWORTH,
Daniel, Dale; 9462 Chabola Road, San
Diego, CA 92129 (US). JONES, Todd,
Kevin; 546 Marview Drive, Solana Beach,
CA 92075 (US). JUDGE, Luke, Milburn;
644 ? Bonair Way, La Jolla, CA 92037
(US). RIPKA, Wiliam, Charles; 10819
Red Rock Drive, San Diego, CA 92131
(US). SHAPIRA, Barry, Zvi; 5925 La Jolla
Corona Drive, La Jolla, CA 92037 (US).
UYEDA, Roy, Teruyuki; 5385 Toscana
Way, Apt. 342, San Diego, CA 92122 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG UZ VN YU
ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(c)
(51) 7 C07D 498/04, A61K 31/40, 31/55, 31/501,
31/42, 31/44, 31/506, A61P 25/18 // (C07D
498/04, 333:00, 261:00)
(11) WO 01/19832 (13) A2
(21) PCT/US00/24949
(22) 13 Sep/sep 2000 (13.09.2000)
(25) en (26) en
(30) 09/396,156 14 Sep/sep 1999 US
(14.09.1999)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) THIENOISOXAZOLE PHENOXY UN-
SUBSTITUTED ETHYL AND PROPYL
DERIVATIVES USEFUL AS D4 ANTAG-
ONISTS
DERIVES DE PROPYLE ET D’ETHYLE
NON SUBSTITUES DE PHENOXY
THIENOISOXAZOLE UTILES COMME
ANTAGONISTES D4
(63) US 09/396,156 (CON)
14 Sep/sep 1999 (14.09.1999)
(71) AVENTIS PHARMACEUTICALS, INC.
[US/US]; Route 202-206, P.O. Box 6800,
Bridgewater, NJ 08876-0800 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) LEE, George, E. [US/US]; 2 Seville
Drive, Somerville, NJ 08876 (US). AYERS,
Timothy, A. [US/US]; 179 Glen Lake Road,
Loveland, OH 45140 (US). JURCAK, John,
G. [US/US]; 2431 13th Street, Bethlehem,
PA 18017 (US).
(74) KURYS, Barbara et al. / etc.; Aventis Pharmaceuticals
Inc, Route 202-206, P.O. Box
6800, Mail Code: EMC-G1, Bridgewater, NJ
08807-0800 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 498/04, 519/00, A61K 31/40, 31/55,
31/501, 31/42, 31/44, 31/506, A61P 25/18
// (C07D 498/04, 333:00, 261:00) (C07D
519/00, 498:00, 451:00) (C07D 519/00,
498:00, 495:00)
(11) WO 01/19833 (13) A1
(21) PCT/US00/24962
(22) 13 Sep/sep 2000 (13.09.2000)
(25) en (26) en
(30) 09/396,081 14 Sep/sep 1999 US
(14.09.1999)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) THIENOISOXAZOLYL- AND
THIENYLPYRRAZOLYL-PHENOXY
SUBSTITUTED PROPYL DERIVA-
TIVES USEFUL AS D4 ANTAGONISTS
DERIVES THIENOISOXAZOLYLE ET
THIENYLPYRRAZOLYLE DU PRO-
PYLE A SUBSTITUTION PHENOXY,
ANTAGONISTES DU D4
(63) US 09/396,081 (CON)
14 Sep/sep 1999 (14.09.1999)
(71) AVENTIS PHARMACEUTICALS, INC.
[US/US]; Route 202-206, P.O. Box 6800,
Bridgewater, NJ 08876-0800 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) FINK, David, M. [US/US]; One Kensington
Court, Lebanon, NJ 08833 (US).
FREED, Brian, S. [US/US]; 47 Puddingstone
Way, Phillipsburg, NJ 08865
(US). HRIB, Nicholas, J. [US/US]; 2402
Jamestown Common, Somerville, NJ
08876 (US). KOSLEY, Raymond, W.,
Jr. [US/US]; 659 Cedarbrook Road, Bridgewater,
NJ 08807 (US). LEE, George, E.
[US/US]; 2 Seville Drive, Somerville, NJ
08876 (US). MERRIMAN, Gregory, H.
[US/US]; 248 Stonehenge Drive, Phillipsburg,
NJ 08865 (US). RAUCKMAN, Barbara,
S. [US/US]; 21 Barley Sheaf Road,
Flemington, NJ 08822 (US).
(74) KURYS, Barbara, E. et al. / etc.; Aventis
Pharmaceuticals Inc., Route 202-206, P.O.
Box 6800, Mail Code: EMC-G1, Bridgewater,
NJ 08807-0800 (US).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
Published / Publiée :(c)
(51) 7 C07F 5/02, C08G 61/10, H01B 1/12,
H05B 33/14
(11) WO 01/19834 (13) A1
(21) PCT/GB00/03554