PCT/2001/12 : PCT Gazette, Weekly Issue No. 12, 2001 - WIPO

12/2001
4754 PCT Gazette - Section I - Gazette du PCT 22 Mar/mar 2001
(51) 7 C07D 251/68, C11D 3/42, D06L 3/12,
D21H 21/30
(11) WO 01/19804 (13) A1
(21) PCT/EP00/08621
(22) 4 Sep/sep 2000 (04.09.2000)
(25) en (26) en
(30) 99810813.8 10 Sep/sep 1999 EP
(10.09.1999)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) TRIAZINYLAMINOSTILBENE
DERIVATIVE AS FLUORESCENT
WHITENING AGENTS
DERIVES DE TRIAZINYLAMINOS-
TILBENE TENANT LIEU D’AGENTS
ECLAIRCISSANTS FLUORESCENTS
(71) CIBA SPECIALTY CHEMICALS
HOLDING INC. [CH/CH]; Klybeckstrasse
141, CH-4057 Basel (CH).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) METZGER, Georges [FR/FR];
Herrenweg 228, F-68480 Moernach
(FR). HAUGER, Serge [FR/FR]; 10,
rue de Michelbach-le-Bas, F-68730
Ranspach-le-Bas (FR). CUESTA, Fabienne
[FR/FR]; 80 D, rue Principale, F-68480 Roppentzwiller
(FR). BULLIARD, Christophe
[CH/CH]; Turnerstrasse 25, CH-4058 Basel
(CH). ROHRINGER, Peter [CH/CH]; Sechs
Juchartenstrasse 1, CH-4124 Schönenbuch
(CH). GRIENENBERGER, Marc, Roger
[FR/FR]; 13, rue de la Forêt, F-68870 Bartenheim
(FR).
(74) CIBA SPECIALTY CHEMICALS
HOLDING INC.; Patentabteilung, Klybeckstrasse
141, CH-4057 Basel (CH).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU
ID IL IN IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MA MD MG MK MN MW
MX MZ NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ VN
YU ZA ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 263/32, 277/22, 277/24, 417/12,
263/44
(11) WO 01/19805
(21) PCT/JP00/06140
(13) A1
(22) 8 Sep/sep 2000 (08.09.2000)
(25) ja (26) ja
(30) 11/257540 10 Sep/sep 1999
(10.09.1999)
JP
(43) 22 Mar/mar 2001 (22.03.2001)
(54) HETEROCYCLIC COMPOUNDS AND
PROCESS FOR THE PREPARATION
THEREOF
COMPOSES HETEROCYCLIQUES ET
PROCEDE DE PREPARATION DE CES
DERNIERS
(71) TAKEDA CHEMICAL INDUSTRIES,
LTD. [JP/JP]; 1-1, Doshomachi 4-chome,
Chuo-ku, Osaka-shi, Osaka 541-0045 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) YAMANE, Taihei [JP/JP]; 1-3, Satsukigaoka
5-chome, Ikeda-shi, Osaka 563-0029
(JP).
(74) TAKAHASHI, Shuichi et al. / etc.; Osaka
Plant of Takeda Chemical Industries,
Ltd., 17-85, Jusohonmachi 2-chome, Yodogawa-ku,
Osaka-shi, Osaka 532-0024 (JP).
(81) AE AG AL AM AU AZ BA BB BG BR BY
BZ CA CN CR CU CZ DM DZ EE GD GE
HR HU ID IL IN IS JP KG KR KZ LC LK
LR LT LV MA MD MG MK MN MX MZ
NO NZ PL RO RU SG SI SK TJ TM TR TT
UA US UZ VN YU ZA.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 263/38, 263/48, 413/04
(11) WO 01/19806
(21) PCT/JP00/06302
(13) A1
(22) 14 Sep/sep 2000 (14.09.2000)
(25) ja (26) ja
(30) 11/262470 16 Sep/sep 1999
(16.09.1999)
JP
(30) 2000/81823 17 Mar/mar 2000
(17.03.2000)
JP
(43) 22 Mar/mar 2001 (22.03.2001)
(54) PROCESS FOR THE PREPARATION OF
OXAZOLE DERIVATIVES
PROCEDE DE PREPARATION DE DE-
RIVES DE L’OXAZOLE
(71) TAKEDA CHEMICAL INDUSTRIES,
LTD. [JP/JP]; 1-1, Doshomachi 4-chome,
Chuo-ku, Osaka-shi, Osaka 541-0045 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) TAWADA, Hiroyuki [JP/JP]; 11-1,
Miyanokawahara 1-chome, Takatsuki-shi,
Osaka 569-1032 (JP). OHASHI, Norihiko
[JP/JP]; 10-3-804, Kamihamuro
1-chome, Takatsuki-shi, Osaka 569-1044
(JP). IKEUCHI, Motoki [JP/JP]; 6-13-303,
Wakayamacho,
663-8016 (JP).
Nishinomiya-shi, Hyogo
(74) TAKAHASHI, Shuichi et al. / etc.; Osaka
Plant of Takeda Chemical Industries,
Ltd., 17-85, Jusohonmachi 2-chome, Yodogawa-ku,
Osaka-shi, Osaka 532-0024 (JP).
(81) AE AG AL AM AU AZ BA BB BG BR BY
BZ CA CN CR CU CZ DM DZ EE GD GE
HR HU ID IL IN IS JP KG KR KZ LC LK
LR LT LV MA MD MG MK MN MX MZ
NO NZ PL RO RU SG SI SK TJ TM TR TT
UA US UZ VN YU ZA.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 277/18, 279/06, 279/08, 417/12,
A61K 31/426, 31/541, 31/5415, 31/547,
A61P 13/12, 29/00, 37/06, 43/00 // (C07D
417/12, 213:36, 279:06) (C07D 417/12,
215:12, 279:06) (C07D 417/12, 279:06,
333:34)
(11) WO 01/19807 (13) A1
(21) PCT/JP00/06185
(22) 11 Sep/sep 2000 (11.09.2000)
(25) ja (26) ja
(30) 11/260780 14 Sep/sep 1999 JP
(14.09.1999)
(43) 22 Mar/mar 2001 (22.03.2001)
(54) 2-IMINO-1,3-THIAZINE DERIVATIVES
DERIVES DE 2-IMINO-1,3-THIAZINE
(71) SHIONOGI & CO., LTD. [JP/JP]; 1-8,
Doshomachi 3-chome, Chuo-ku, Osaka-shi,
Osaka 541-0045 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) HANASAKI, Koji [JP/JP]; Shionogi
& Co., Ltd., 12-4, Sagisu 5-chome,
Fukushima-ku, Osaka-shi, Osaka 553-0002
(JP). MURASHI, Takami [JP/JP]; Shionogi
& Co., Ltd., 1405, Oaza Gotanda, Kokacho,
Koka-gun, Shiga 520-3423 (JP). KAI, Hiroyuki
[JP/JP]; Shionogi & Co., Ltd., 1405,
Oaza Gotanda, Kokacho, Koka-gun, Shiga
520-3423 (JP).
(74) YAMAUCHI, Hideaki et al. / etc.; Shionogi
& Co., Ltd. Intellectual Property Department,
12-4, Sagisu 5-chome, Fukushima-ku, Osakashi,
Osaka 553-0002 (JP).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY BZ CA CH CN CR CU CZ DE DK DM
DZ EE ES FI GB GD GE GH GM HR HU ID
IL IN IS JP KE KG KR KZ LC LK LR LS LT
LU LV MA MD MG MK MN MW MX MZ
NO NZ PL PT RO RU SD SE SG SI SK SL
TJ TM TR TT TZ UA UG US UZ VN YU ZA
ZW.
(84) AP (GH GM KE LS MW MZ SD SL SZ TZ
UG ZW); EA (AM AZ BY KG KZ MD RU
TJ TM); EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN GW ML MR NE SN
TD TG).
(51) 7 C07D 295/20, 211/66, 213/89, 213/82,
213/81, 241/24, 309/08, 333/38, 333/40,
209/08, 317/68, 333/70, 215/54, 215/48,
C07C 317/28, A61K 31/5375, 31/5377,
31/455, 31/47, 31/4965, 31/381, A61P 19/02,
33/06
(11) WO 01/19808
(21) PCT/US00/25341
(13) A1
(22) 15 Sep/sep 2000 (15.09.2000)
(25) en (26) en
(30) 60/154,245 16 Sep/sep 1999
(16.09.1999)
US
(30) 60/171,831 22 Dec/déc 1999
(22.12.1999)
US
(30) 60/224,552 10 Aug/août 2000
(10.08.2000)
US
(43) 22 Mar/mar 2001 (22.03.2001)
(54) CHEMICAL COMPOUNDS AND COM-
POSITIONS AND THEIR USE AS
CATHEPSIN S INHIBITORS
COMPOSES ET COMPOSITIONS CHI-
MIQUES ET LEUR UTILISATION EN
TANT QU’INHIBITEURS DE LA CA-
THEPSINE S