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PCT/2001/45 - World Intellectual Property Organization

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<strong>45</strong>/<strong>2001</strong><br />

20104 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 8 Nov/nov <strong>2001</strong><br />

PROCEDE D’INHIBITION DE L’AGRE-<br />

GATION DE PROTEINES AMYLOIDES<br />

ET D’IMAGERIE DE DEPOTS AMY-<br />

LOIDES FAISANT APPEL A DES DE-<br />

RIVES AMINO-INDANES<br />

(71) WARNER-LAMBERT COMPANY<br />

[US/US]; 201 Tabor Road, Morris Plains,<br />

NJ 07950 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) BARTA, Nancy, Sue [US/US]; Pfizer<br />

Inc., PGRD, Ann Arbor Laboratories, 2800<br />

Plymouth Road, Ann Arbor, MI 48105 (US).<br />

BIGGE, Christopher, Franklin [US/US];<br />

Pfizer Inc., PGRD, Ann Labor Laboratories,<br />

2800 Plymouth Road, Ann Arbor, MI 48105<br />

(US).<br />

(74) FEDERMAN, Evan, J.; Warner-Lambert<br />

Company, 201 Tabor Road, Morris Plains, NJ<br />

07950 (US) et al. / etc.<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG US<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07C 233/13, 233/15, 233/18, 233/25,<br />

233/54, 327/42, C07D 333/36, 333/40,<br />

277/46, 277/82, 261/14, 231/40, 213/75,<br />

215/38, 239/42, 239/52, 253/06, C07F 9/40,<br />

A01N 37/18, 37/20, 37/24, 43/10, 43/40,<br />

43/56, 43/54, 43/64, 43/78, 43/80<br />

(11) WO 01/83426<br />

(21) <strong>PCT</strong>/JP01/03703<br />

(13) A1<br />

(22) 27 Apr/avr <strong>2001</strong> (27.04.<strong>2001</strong>)<br />

(25) ja (26) ja<br />

(30) 2000-126931 27 Apr/avr 2000<br />

(27.04.2000)<br />

JP<br />

(30) 2000-135840 9 May/mai 2000<br />

(09.05.2000)<br />

JP<br />

(30) 2000-176535 13 Jun/juin 2000<br />

(13.06.2000)<br />

JP<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) 2-FLUOROALKANAMIDE COM-<br />

POUND AND PEST CONTROL AGENT<br />

FOR AGRICULTURAL OR HORTICUL-<br />

TURAL USE<br />

COMPOSE 2-FLUOROALCANAMIDE<br />

ET PESTICIDE POUR L’AGRICUL-<br />

TURE OU L’HORTICULTURE<br />

(71) UBE INDUSTRIES, LTD. [JP/JP];<br />

1978-96, Oaza Kogushi, Ube-shi, Yamaguchi<br />

755-8633 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) TSUTSUMIUCHI, Kiyoshi [JP/JP];<br />

Ube Research Laboratory, Ube Industries,<br />

Ltd., 1978-5, Oaza Kogushi, Ube-shi,<br />

Yamaguchi 755-8633 (JP). SHIKITA,<br />

Shoji [JP/JP]; Ube Research Laboratory,<br />

Ube Industries, Ltd., 1978-5, Oaza Kogushi,<br />

Ube-shi, Yamaguchi 755-8633 (JP).<br />

KUWATA, Takaaki [JP/JP]; Ube Industries,<br />

Ltd., Ube Research Laboratory, 1978-5, Oaza<br />

Kogushi, Ube-shi, Yamaguchi 755-8633<br />

(JP). ASAHARA, Takehiko [JP/JP]; Ube<br />

Research Laboratory, Ube Industries, Ltd.,<br />

1978-5, Oaza Kogushi, Ube-shi, Yamaguchi<br />

755-8633 (JP). NORITAKE, Tomoya<br />

[JP/JP]; Ube Research Laboratory,<br />

Ube Industries, Ltd., 1978-5, Oaza Kogushi,<br />

Ube-shi, Yamaguchi 755-8633 (JP).<br />

(74) TSUKUNI, Hajime; SVAX TS Building,<br />

22-12, Toranomon 1-chome, Minato-ku,<br />

Tokyo 105-0001 (JP).<br />

(81) AE AG AL AU BA BB BG BR BZ CA CN<br />

CO CR CU CZ DM DZ EE GD GE HR HU<br />

ID IL IN IS KR LC LK LR LT LV MA MG<br />

MK MN MX NO NZ PL RO SG SI SK TT<br />

UA US UZ VN YU ZA.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07C 233/65, 233/66, 233/75, 233/80,<br />

233/81, 271/28, 311/08, 311/21, 311/58,<br />

311/64, C07D 207/325, 213/40, 213/75,<br />

213/76, 213/81, 213/82, 215/38, 215/40,<br />

217/22, 231/40, 231/42, 231/56, 233/61,<br />

235/32, 237/04, 237/20, 239/20, 239/22,<br />

239/26, 239/42, 239/69, 241/20, 261/16,<br />

263/48, 263/58, 277/42, 277/44, 277/46,<br />

277/50, 277/52, 277/66, 277/82, 285/10,<br />

285/12, 295/12, 295/18, 295/20, 295/22,<br />

311/22, 333/38, 333/66, 417/04, 471/04,<br />

A61K 31/167, 31/352, 31/381, 31/40, 31/415,<br />

31/4164, 31/4184, 31/423, 31/426, 31/427,<br />

31/428, 31/433, 31/437, 31/44, 31/4402,<br />

31/4406, 31/4409, 31/4439, 31/4<strong>45</strong>3, 31/<strong>45</strong>5,<br />

31/47, 31/472, 31/495, 31/4965, 31/50,<br />

31/505, 31/5375, 31/55, 31/635, A61P 1/16,<br />

1/18, 13/12, 19/02, 19/06, 19/08, 19/10,<br />

25/28, 29/00, 3/04, 3/06, 3/10, 35/00, 35/02,<br />

37/06, 5/14, 7/06, 9/00, 9/10, 9/12<br />

(11) WO 01/83427 (13) A1<br />

(21) <strong>PCT</strong>/JP01/03655<br />

(22) 26 Apr/avr <strong>2001</strong> (26.04.<strong>2001</strong>)<br />

(25) ja (26) ja<br />

(30) 2000-129565 28 Apr/avr 2000 JP<br />

(28.04.2000)<br />

(30) <strong>2001</strong>-060366 5 Mar/mar <strong>2001</strong> JP<br />

(05.03.<strong>2001</strong>)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) PPARγ MODULATORS<br />

MODULATEURS DE PPARγ<br />

(71) SANKYO COMPANY, LIMITED [JP/JP];<br />

5-1, Nihonbashi Honcho 3-chome, Chuo-ku,<br />

Tokyo 103-8426 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) AMEMIYA, Yoshiya [JP/JP]; c/o<br />

SANKYO COMPANY, LIMITED, 2-58,<br />

Hiromachi 1-chome, Shinagawa-ku, Tokyo<br />

140-8710 (JP). WAKABAYASHI, Kenji<br />

[JP/JP]; c/o SANKYO COMPANY, LIM-<br />

ITED, 2-58, Hiromachi 1-chome, Shinagawa-ku,<br />

Tokyo 140-8710 (JP). TAKAISHI,<br />

Sachiko [JP/JP]; c/o SANKYO COMPANY,<br />

LIMITED, 2-58, Hiromachi 1-chome, Shinagawa-ku,<br />

Tokyo 140-8710 (JP). FUKUDA,<br />

Chie [JP/JP]; c/o SANKYO COMPANY,<br />

LIMITED, 2-58, Hiromachi 1-chome, Shinagawa-ku,<br />

Tokyo 140-8710 (JP).<br />

(74) OHNO, Akio et al. / etc.; c/o SANKYO<br />

COMPANY, LIMITED, 2-58, Hiromachi<br />

1-chome, Shinagawa-ku, Tokyo 140-8710<br />

(JP).<br />

(81) AU BR CA CN CZ HU ID IL IN KR MX NO<br />

NZ PL RU US ZA.<br />

(84) EP (AT BE CH CY DE DK ES FI FR GB GR<br />

IE IT LU MC NL PT SE TR).<br />

Published / Publiée :(c)<br />

(51) 7 C07C 255/37, A01N 37/34, C07C 253/00<br />

(11) WO 01/83428 (13) A1<br />

(21) <strong>PCT</strong>/EP01/04958<br />

(22) 3 May/mai <strong>2001</strong> (03.05.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 60/201,826 4 May/mai 2000 US<br />

(04.05.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) 1,4-DIARYL-2-FLUORO-4-CYANO-2-<br />

BUTENES, PROCESS FOR THEIR<br />

PREPARATION AND INTERMEDI-<br />

ATES USEFUL THEREFOR<br />

1,4-DIARYL-2-FLUORO-4-CYANO-2-<br />

BUTENES, LEUR PROCEDE DE PRE-<br />

PARATION ET LEURS PRODUITS<br />

INTERMEDIAIRES UTILES<br />

(71) BASF AKTIENGESELLSCHAFT<br />

[DE/DE]; 67056 Ludwigshafen (DE).<br />

(72) HU, Yulin; 54 Hampshire Drive, Plainsboro,<br />

NJ (US). HUNT, David, Allen; 703 Daventry<br />

Drive, Greenville, NC 27858 (US).<br />

(74) BASF AKTIENGESELLSCHAFT; 67056<br />

Ludwigshafen (DE).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG UZ<br />

VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07C 275/40, 279/18, 335/20, 335/32,<br />

A61K 31/155, A61P 43/00, 9/10, 25/00,<br />

7/02, 25/04, 25/06, 25/16, 25/28, 25/08,<br />

25/36<br />

(11) WO 01/83429 (13) A1<br />

(21) <strong>PCT</strong>/JP01/03721<br />

(22) 27 Apr/avr <strong>2001</strong> (27.04.<strong>2001</strong>)<br />

(25) ja (26) ja<br />

(30) 2000-129725 28 Apr/avr 2000<br />

(28.04.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) ANILINE DERIVATIVES<br />

DERIVES D’ANILINE<br />

JP

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