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PCT/2001/45 - World Intellectual Property Organization

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<strong>45</strong>/<strong>2001</strong><br />

20008 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 8 Nov/nov <strong>2001</strong><br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 01/82913<br />

(21) <strong>PCT</strong>/JP01/03617<br />

(13) A2<br />

(22) 26 Apr/avr <strong>2001</strong> (26.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 60/201,712 3 May/mai 2000<br />

(03.05.2000)<br />

US<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) OCULAR TENSION DEPRESSOR<br />

MEDICAMENT ABAISSANT LA PRES-<br />

SION OCULAIRE<br />

(71) SUCAMPO AG [CH/CH]; Graben 5,<br />

CH-6300 Zug (CH). FUJISAWA PHAR-<br />

MACEUTICAL CO., LTD. [JP/JP]; 4-7,<br />

Doshomachi 3-chome, Chuo-ku, Osaka-shi,<br />

Osaka 541-8514 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) UENO, Ryuji [JP/US]; 11025 Stanmore<br />

Drive, Potomac, Montgomery, MD 20854<br />

(US).<br />

(74) KOTANI, Etsuji et al. / etc.; Nichimen<br />

Building 2nd Floor, 2-2, Nakanoshima<br />

2-chome, Kita-ku, Osaka-shi, Osaka<br />

530-0005 (JP).<br />

(81) AU BR CA CN HU IN JP KR MX NO NZ<br />

PL RU US.<br />

(84) EP (AT BE CH CY DE DK ES FI FR GB GR<br />

IE IT LU MC NL PT SE TR).<br />

(51) 7 A61K 31/00<br />

(11) WO 01/82914<br />

(21) <strong>PCT</strong>/US01/13546<br />

(13) A2<br />

(22) 27 Apr/avr <strong>2001</strong> (27.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 60/200,437 28 Apr/avr 2000<br />

(28.04.2000)<br />

US<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) TOPICAL ANESTHETIC/OPIOID FOR-<br />

MULATIONS AND USES THEREOF<br />

FORMULATIONS TOPIQUES A BASE<br />

D’ANESTHESIQUE ET D’OPIOIDE, ET<br />

UTILISATIONS ASSOCIEES<br />

(71) MEMORIAL SLOAN-KETTERING<br />

CANCER CENTER [US/US]; 460 East<br />

63rd Street, New York, NY 10021 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) PASTERNAK, Gavril [US/US]; Apartment<br />

21M, 500 East 83rd Street, New York,<br />

NY 10028 (US). KOLESNIKOV, Yuri<br />

[US/US]; 38 Ridge Road,<br />

07626 (US).<br />

Cresskill, NJ<br />

(74) LEHNHARDT, Susan, K.; Frommer<br />

Lawrence & Haug LLP, 7<strong>45</strong> Fifth Avenue,<br />

New York, NY 10151 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG US<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 01/82915 (13) A2<br />

(21) <strong>PCT</strong>/US01/13701<br />

(22) 27 Apr/avr <strong>2001</strong> (27.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 09/559,528 28 Apr/avr 2000 US<br />

(28.04.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) TRANS-CLITORAL ADMINISTRA-<br />

TION OF THERAPY<br />

ADMINISTRATION TRANSCLITORI-<br />

DIENNE D’UN TRAITEMENT<br />

(71, 72) NEAL, Gary, W. [US/US]; 200<br />

Fort Sanders West Boulevard, Suite 309,<br />

Knoxville, TN 37922 (US).<br />

(74) ZOLTICK, Martin, M.; Zoltick Technology<br />

Law Group, PLLC, 21515 Ridgetop Circle,<br />

Suite 200, Sterling, VA 20166 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG UZ VN YU<br />

ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 01/82916<br />

(21) <strong>PCT</strong>/US01/14393<br />

(13) A2<br />

(22) 2 May/mai <strong>2001</strong> (02.05.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 60/201,613 3 May/mai 2000<br />

(03.05.2000)<br />

US<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) COMBINATION THERAPEUTIC COM-<br />

POSITIONS AND METHODS OF USE<br />

COMPOSITIONS THERAPEUTIQUES<br />

COMBINEES ET LEURS METHODES<br />

D’UTILISATION<br />

(71) TULARIK INC. [US/US]; Two Corporate<br />

Drive, South San Francisco, CA 94080 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) JAEN, Juan, C. [US/US]; 154 Los<br />

Robles Drive, Burlingame, CA 94010 (US).<br />

CHEN, Jin-Long [CN/US]; 101 Challenge<br />

Court, Foster City, CA 94404 (US).<br />

(74) SNYDER, Joseph, R.; Townsend and<br />

Townsend and Crew LLP, Two Embarcadero<br />

Center, 8th floor, San Francisco, CA<br />

94111-3834 (US) et al. / etc.<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 01/82917 (13) A2<br />

(21) <strong>PCT</strong>/US01/1<strong>45</strong>86<br />

(22) 3 May/mai <strong>2001</strong> (03.05.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 60/201,601 3 May/mai 2000 US<br />

(03.05.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) TREATMENT OF HYPERTRIGLYC-<br />

ERIDEMIA AND OTHER CONDITIONS<br />

USING LXR MODULATORS<br />

TRAITEMENT DE L’HYPERTRIGLY-<br />

CERIDEMIE ET D’AUTRES MALA-<br />

DIES AU MOYEN DE MODULATEURS<br />

LXR<br />

(71) TULARIK INC. [US/US]; Two Corporate<br />

Drive, South San Francisco, CA 94080 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) SHAN, Bei [US/US]; 349 Quay Lane,<br />

Redwood City, CA 94065 (US). SCHULTZ,<br />

Joshua [US/US]; 302 Amesport Landing,<br />

Half Moon Bay, CA 94019 (US). TU, Hua<br />

[CN/US]; 750 Glenview Drive, Apt. 307, San<br />

Bruno, CA 94066 (US).<br />

(74) GARRETT-WACKOWSKI, Eugenia;<br />

Townsend and Townsend and Crew LLP,<br />

Two Embarcadero Center, 8th Floor, San<br />

Francisco, CA 94111-3834 (US) et al. / etc.<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

(51) 7 A61K 31/00<br />

(11) WO 01/82918<br />

(21) <strong>PCT</strong>/US01/40639<br />

(13) A2<br />

(22) 30 Apr/avr <strong>2001</strong> (30.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 09/561,663 2 May/mai 2000<br />

(02.05.2000)<br />

US<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) METHOD FOR THE PREVENTION OF<br />

APOPTOSIS

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