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PCT/2001/45 - World Intellectual Property Organization

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<strong>45</strong>/<strong>2001</strong><br />

20120 <strong>PCT</strong> Gazette - Section I - Gazette du <strong>PCT</strong> 8 Nov/nov <strong>2001</strong><br />

(84) EP (AT BE CH CY DE DK ES FI FR GB GR<br />

IE IT LU MC NL PT SE TR).<br />

Published / Publiée :(c)<br />

(51) 7 C07F 9/24, A61K 31/664, A61P 35/04<br />

(11) WO 01/83496 (13) A1<br />

(21) <strong>PCT</strong>/US01/14290<br />

(22) 2 May/mai <strong>2001</strong> (02.05.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 09/563,181 2 May/mai 2000 US<br />

(02.05.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) BIS-(N,N’-BIS-(2-<br />

HALOETHYL)AMINO) PHOS-<br />

PHORAMIDATES AS ANTITUMOR<br />

AGENTS<br />

PHOSPHORAMIDATES BIS-(N,N’-<br />

BIS-(2-HALOETHYL)AMINO)<br />

COMME AGENTS ANTITUMORAUX<br />

(71) TELIK, INC. [US/US]; 750 Gateway Boulevard,<br />

South San Francisco, CA 94080 (US).<br />

(72) HERR, Jason, R.; 248 New Salem South<br />

Road, Voorheesville, NY 12186 (US). LUM,<br />

Robert, T.; 781 Barron Avenue, Palo Alto,<br />

CA 94306 (US). SCHOW, Steven, R.; 127<br />

Mendocino Way, Redwood Shores, CA<br />

94065 (US). MENG, Fanying; 1444 14th<br />

Avenue, San Francisco, CA 94122 (US).<br />

KOZLOWSKI, Michael, R.; 164 Edgewood<br />

Drive, Palo Alto, CA 94303 (US).<br />

ZHICHKIN, Pavel; Apartment 1-R, 28<br />

Peyster Street, Albany, NY 12208 (US).<br />

(74) HEUSCH, Marina, I. et al. / etc.; Heller<br />

Ehrman White & McAuliffe LLP, 275 Middlefield<br />

Road, Menlo Park, CA 94025-3506<br />

(US).<br />

(81) AE AG AL AM AT AT (Utility model /<br />

modèle d’utilité) AUAZBABBBGBRBY<br />

BZ CA CH CN CO CR CU CZ CZ (Utility<br />

model / modèle d’utilité) DE DE (Utility<br />

model / modèle d’utilité) DK DK (Utility<br />

model / modèle d’utilité) DM DZ EE EE<br />

(Utility model / modèle d’utilité) ESFIFI<br />

(Utility model / modèle d’utilité)GBGDGE<br />

GH GM HR HU ID IL IN IS JP KE KG KP<br />

KR KZ LC LK LR LS LT LU LV MA MD<br />

MG MK MN MW MX MZ NO NZ PL PT<br />

RO RU SD SE SG SI SK SK (Utility model<br />

/ modèle d’utilité) SLTJTMTRTTTZUA<br />

UG UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07F 9/6574, A61K 31/665, A61P 3/10,<br />

C12P 9/00, C12N 1/20<br />

(11) WO 01/83497<br />

(21) <strong>PCT</strong>/EP01/04652<br />

(13) A1<br />

(22) 25 Apr/avr <strong>2001</strong> (25.04.<strong>2001</strong>)<br />

(25) de (26) de<br />

(30) 100 21 731.1 4 May/mai 2000<br />

(04.05.2000)<br />

DE<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) CYCLIPOSTINS, A METHOD FOR<br />

THEIR PRODUCTION AND THE USE<br />

OF THE SAME<br />

CYCLIPOSTINES, LEUR PROCEDE DE<br />

PRODUCTION ET LEUR UTILISATION<br />

(71) AVENTIS PHARMA DEUTSCHLAND<br />

GMBH [DE/DE]; Brüningstrasse 50, 65929<br />

Frankfurt (DE).<br />

(72) VERTESY, Laszlo; Eppenhainer Weg<br />

6, 65817 Eppstein-Vockenhausen (DE).<br />

EHRLICH, Klaus; Düsseldorfer Strasse 11,<br />

65428 Rüsselsheim (DE). KURZ, Michael;<br />

Erlenweg 7, 65719 Hofheim (DE). WINK,<br />

Joachim; Magdeburger Strasse 14, 63322<br />

Rödermark (DE).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG UZ<br />

VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07F 07/18<br />

(11) WO 01/83498 (13) A1<br />

(21) <strong>PCT</strong>/US01/13830<br />

(22) 27 Apr/avr <strong>2001</strong> (27.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 09/561,306 28 Apr/avr 2000 US<br />

(28.04.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) POLYMERIZATION CATALYST COM-<br />

POSITIONS AND PROCESSES TO PRO-<br />

DUCE POLYMERS AND BIMODAL<br />

POLYMERS<br />

COMPOSITIONS CATALYTIQUES DE<br />

POLYMERISATION ET PROCEDES DE<br />

PRODUCTION DE POLYMERES ET DE<br />

POLYMERES BIMODAUX<br />

(63) US 09/561,306 (CON)<br />

28 Apr/avr 2000 (28.04.2000)<br />

(71) PHILLIPS PETROLEUM COMPANY<br />

[US/US]; 4th and Keeler, Bartlesville, OK<br />

74004 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) JENSEN, Michael, D. [US/US]; 2008<br />

Skyline Pl., Bartlesville, OK 74006 (US).<br />

McDANIEL, Max, P. [US/US]; 1601 Melmart<br />

Drive, Bartlesville, OK 74006 (US).<br />

BENHAM, Elizabeth, A. [US/US]; 9310<br />

Katie Grace Circle, Spring, TX 77379 (US).<br />

EATON, Anthony, P. [US/US]; <strong>45</strong>0 Williams<br />

Landing Dr., Sugar Land, TX 77479 (US).<br />

MARTIN, Joel, L. [US/US]; 636 Kenwood<br />

Drive, Bartlesville, OK 74006 (US). HAW-<br />

LEY, Gil, R. [US/US]; 1022 N. Wyandotte,<br />

Dewey, OK 74029 (US). CRAIN, Tony, R.<br />

[US/US]; Rt. 1 Box 11, Niotaze, KS 67355<br />

(US). TANNER, Martha, J. [US/US]; 3976<br />

East 600 South, Cutler, IN 46920 (US).<br />

(74) RICHARDS, John; Ladas & Parry, 26West<br />

61st Street, New York, NY 10023 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CO CR CU CZ DE DK<br />

DM DZ EE ES FI GB GD GE GH GM HR<br />

HU ID IL IN IS JP KE KG KP KR KZ LC<br />

LK LR LS LT LU LV MA MD MG MK MN<br />

MW MX MZ NO NZ PL PT RO RU SD SE<br />

SG SI SK SL TJ TM TR TT TZ UA UG US<br />

UZ VN YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 C07H<br />

(11) WO 01/83499 (13) A2<br />

(21) <strong>PCT</strong>/US01/13957<br />

(22) 30 Apr/avr <strong>2001</strong> (30.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 60/200,416 28 Apr/avr 2000 US<br />

(28.04.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

(54) HAPLOTYPES OF THE IL8 GENE<br />

HAPLOTYPES DU GENE DE L’IL8<br />

(71) GENAISSANCE PHARMACEUTICALS,<br />

INC. [US/US]; Five Science Park, New<br />

Haven, CT 06511 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) BENTIVEGNA, Steven, C. [US/US];<br />

49 Greenview Terrace, Middletown, CT<br />

06<strong>45</strong>7 (US). CHEW, Anne [US/US]; 1477<br />

Beacon Street, #64, Brookline, MA 02446<br />

(US). CHOI, Julie, Y. [US/US]; 38 Elizabeth<br />

Street, West Haven, CT 06516 (US). DEN-<br />

TON, R., Rex [US/US]; 129 Hunter’s Trail,<br />

Madison, CT 06443 (US). NANDABALAN,<br />

Krishnan [IN/US]; 228 Village Pond Road,<br />

Guilford, CT 06437 (US).<br />

(74) SHANER, Sandra, L. et al. / etc.; Genaissance<br />

Pharmaceuticals, Inc., Five Science<br />

Park, New Haven, CT 06511 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY BZ CA CH CN CR CU CZ DE DK DM<br />

DZ EE ES FI GB GD GE GH GM HR HU<br />

ID IL IN IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MA MD MG MK MN MW<br />

MX MZ NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG US UZ VN<br />

YU ZA ZW.<br />

(84) AP (GH GM KE LS MW MZ SD SL SZ TZ<br />

UG ZW); EA (AM AZ BY KG KZ MD RU<br />

TJ TM); EP (AT BE CH CY DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE TR); OA<br />

(BF BJ CF CG CI CM GA GN GW ML MR<br />

NE SN TD TG).<br />

Published / Publiée :(q2)<br />

(51) 7 C07H 19/01, A01N 43/90<br />

(11) WO 01/83500 (13) A1<br />

(21) <strong>PCT</strong>/JP01/03656<br />

(22) 26 Apr/avr <strong>2001</strong> (26.04.<strong>2001</strong>)<br />

(25) en (26) en<br />

(30) 2000-127209 27 Apr/avr 2000<br />

(27.04.2000)<br />

(43) 8 Nov/nov <strong>2001</strong> (08.11.<strong>2001</strong>)<br />

JP

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