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Estradiol Valerate<br />

Contains<br />

Climaval - Estradiol Valerate 1mg, 2 mgs.<br />

Estraderm MX 25 - Estradiol 25 micrograms (mcgs)/24 hours.<br />

Estraderm MX 50 - Estradiol 50 mcgs/24 hours.<br />

Estraderm MX 75 - Estradiol 75 mcgs/24 hours.<br />

Estraderm MX 100 - Estradiol 100 mcgs/24 hours.<br />

Estraderm TTS 25 - Estradiol 25 mcgs/24 hours.<br />

Estraderm TTS 50 - Estradiol 50 mcgs/24hours.<br />

Estradiol implant - Estradiol 25mgs, 50 mgs, 100 mgs.<br />

Evorel ’25’ patch - Estradiol 25 mcgs/24 hours.<br />

Evorel ’50’ patch - Estradiol 50 mcgs/24 hours.<br />

Evorel ’75’ patch - Estradiol 75 mcgs/24 hours.<br />

Evorel ’100’ patch - Estradiol 100 mcgs/24 hours.<br />

Progynova - Estradiol Valerate 1mg, 2 mgs.<br />

Progynova TS - Estradiol 50 mcgs/24 hours, Estradiol 100 mcgs/24 hours.<br />

Zumenon - Estradiol 1mg, 2mgs.<br />

Typical dosage<br />

Pre-op<br />

Progynova - 6–12 mgs/day (unknown, 2005),<br />

Progynova - 2–4 mgs/day (Asscheman and LJG Gooren, 1992),<br />

Zumenon - 4–8 mgs/day,<br />

Estraderm TTS - 0.1–0.2 mgs with the patch changed twice a week.<br />

Post-op<br />

Progynova - 2–6 mgs/day (unknown, 2005),<br />

Zumenon - 1–4 mgs/day,<br />

Estradiol implant - 25–100 mgs/4–8 months (according to oestrogen levels)<br />

(BNF, <strong>2016</strong>a),<br />

Evorel - 200mcg/twice a week.<br />

Dosage of oral Estradiol<br />

Dosage<br />

2mg Estradiol<br />

4mg Estradiol<br />

6mg Estradiol<br />

Blood levels<br />

180–250 pmol/L<br />

360–500 pmol/L<br />

540–750 pmol/L<br />

Table 6.1 – Normal range & dose of Estradiol, for oral tablets only<br />

The above table gives the approximate normal range/dose for Estradiol<br />

80<br />

Version <strong>2016</strong>.3576– – Document LATEXed – 1st May <strong>2016</strong><br />

[git] • Branch: 1.5 @ 26b5e6d • Release: 1.5 (<strong>2016</strong>-05-01)

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