section 1 - World Intellectual Property Organization

37/2000
13238 PCT Gazette - Section I - Gazette du PCT 14 Sep/sep 2000
(54) N–PROTECTED SYNTHESIS ME-
THOD FOR USE IN MAKING POR-
PHYRINS
SYNTHESE N–PROTEGEE CON-
VENANT A LA PREPARATION DE
PORPHYRINES
(71) EMORY UNIVERSITY [US/US]; 2009
Ridgewood Drive, Atlanta, GA 30322 (US).
(72) NICKEL, Eric, G.; 8356–I Roswell Road,
Atlanta, GA 30350 (US). LIEBESKIND,
Lanny, S.; 2573 Kings Lake Court, Atlanta,
GA 30345 (US).
(74) JOHNSON, William, R. et al. / etc.;
Needle & Rosenberg, P.C., 127 Peachtree
Street, N.E., Suite 1200, Atlanta, GA 30303
(US).
(81) AU CA JP; EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE).
(51) 7 C07D 207/38, 309/32, A61K 31/40,
31/365, 31/38, 31/35, C07D 307/66,
333/36, A61P 35/00
(11) WO 00/53581 (13) A2
(21) PCT/EP00/01721
(22) 1 Mar/mar 2000 (01.03.2000)
(25) en (26) en
(30) MI99A000456 5 Mar/mar 1999
(05.03.1999)
(43) 14 Sep/sep 2000 (14.09.2000)
(54) HETEROCYCLIC COMPOUNDS HA-
VING ANTITUMOR ACTIVITY
COMPOSES HETEROCYCLIQUES
AYANT UNE ACTIVITE ANTITUMO-
RALE
(71) NOVUSPHARMA S.P.A. [IT/IT]; Piazza
Durante, 11, I–20131 Milano (IT).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) MENTA, Ernesto [IT/IT]; (IT).
CONTI, Marco [IT/IT]; (IT). PESCALLI,
Nicoletta [IT/IT]; Via G.B. Stucchi, 110,
I–20052 Monza (IT).
(74) MINOJA, Fabrizio et al. / etc.; Bianchetti
Bracco Minoja S.r.l., Via Rossini, 8, I–20122
Milano (IT).
(81) AE AL AM AT AU AZ BA BB BG BR BY
CA CH CN CR CU CZ DE DK DM EE ES
FI GB GD GE GH GM HR HU ID IL IN
IS JP KE KG KP KR KZ LC LK LR LS LT
LU LV MA MD MG MK MN MW MX NO
NZ PL PT RO RU SD SE SG SI SK SL TJ
TM TR TT TZ UA UG US UZ VN YU ZA
ZW; AP (GH GM KE LS MW SD SL SZ
TZ UG ZW); EA (AM AZ BY KG KZ MD
RU TJ TM); EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE);
OA (BF BJ CF CG CI CM GA GN GW ML
MR NE SN TD TG).
(51) 7 C07D 213/73, 417/06, 401/06, 413/06,
233/88, A61K 31/44, 31/4439, 31/444,
31/506, 31/501, 31/5355, 31/427, 31/4168,
A91P 43/00, 25/28
(11) WO 00/53582 (13) A1
(21) PCT/JP00/01190
IT
(22) 1 Mar/mar 2000 (01.03.2000)
(25) ja (26) ja
(30) 11/57993 5 Mar/mar 1999
(05.03.1999)
(43) 14 Sep/sep 2000 (14.09.2000)
(54) HETEROCYCLIC COMPOUNDS HA-
VING EFFECT OF ACTIVATING
NICOTINIC ACETYLCHOLINE
RECEPTOR
4 2
COMPOSES HETEROCYCLIQUES
POSSEDANT UN EFFET
D’ACTIVATION DU RECEPTEUR
4 2 DE L’ACETYLCHOLINE
NICOTINIQUE
(71) SUNTORY LIMITED [JP/JP]; 1–40, Dojimahama
2–chome,
Osaka 530–8203 (JP).
Kita–ku, Osaka–shi,
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) IMOTO, Masahiro [JP/JP];
11–96–401, Ootani–cho, Nishinomiya–shi,
Hyogo 662–0054 (JP). IWANAMI, Tatsuya
[JP/JP]; 34–2–903, Yahata–cho 2–chome,
Ashikaga–shi, Tochigi 326–0824 (JP). AKA-
BANE, Minako [JP/JP]; 1–37–201, Sojiji
1–chome, Ibaraki–shi, Osaka 567–0801
(JP). TANI, Yoshihiro [JP/JP]; 9–38, Hoshimi–cho,
(JP).
Ibaraki–shi, Osaka 567–0843
(74) KUSAMA, Osamu; Kusama Patent Office,
7f Iwata Bldg., 5–12, Iidabashi 4–chome,
Chiyoda–ku, Tokyo 102–0072 (JP).
(81) AU CA CN JP KR US; EP (AT BE CH CY
DE DK ES FI FR GB GR IE IT LU MC NL
PT SE).
(51) 7 C07D 237/22, C07K 5/06, C07D 257/04,
405/12, 261/12, 213/81, 237/06, 207/26,
213/82, 307/68, A61K 31/165, 31/42, 31/44
(11) WO 00/53583
(21) PCT/US00/06022
(13) A1
(22) 9 Mar/mar 2000 (09.03.2000)
(25) en (26) en
(30) 09/265,410 10 Mar/mar 1999
(10.03.1999)
US
(43) 14 Sep/sep 2000 (14.09.2000)
(54) INHIBITORS OF PROTEIN TYROSINE
PHOSPHATASE
INHIBITEURS DE LA TYROSINE
PHOSPHATASE
(71) PHARMACIA & UPJOHN AB [SE/SE];
S–112 87 Stockholm (SE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) LARSEN, Scott, D. [US/US]; 56 Naples
Court, Kalamazoo, MI 49009 (US). MAY,
Paul, D. [US/US]; 7890 North 32nd Street,
Richland, MI 49083 (US). BLEASDALE,
John, E. [GB/US]; 3230 Lites End Court,
Portage, MI 49024 (US). LILJEBRIS,
Charlotta [SE/SE]; S–741 92 Knivsta (SE).
SCHOSTAREZ, Heinrich, Josef [US/US];
3236 Lost Pine Way, Portage, MI 49024
(US). BARF, Tjeerd [NL/SE]; S–753
34 Uppsala (SE). NILSSON, Marianne
[SE/SE]; S–762 94 Rimbo (SE).
JP
(74) MURPHY, Gerald, M.; Birch, Stewart,
Kolasch & Birch, L.L.P., P.O. Box 747, Falls
Church, VA 22040–0747 (US).
(81) AE AL AM AT AU AZ BA BB BG BR BY
CA CH CN CR CU CZ DE DK DM EE ES
FI GB GD GE GH GM HR HU ID IL IN
IS JP KE KG KP KR KZ LC LK LR LS LT
LU LV MA MD MG MK MN MW MX NO
NZ PL PT RO RU SD SE SG SI SK SL TJ
TM TR TT TZ UA UG US UZ VN YU ZA
ZW; AP (GH GM KE LS MW SD SL SZ
TZ UG ZW); EA (AM AZ BY KG KZ MD
RU TJ TM); EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE);
OA (BF BJ CF CG CI CM GA GN GW ML
MR NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 239/96
(11) WO 00/53584 (13) A1
(21) PCT/JP00/01360
(22) 6 Mar/mar 2000 (06.03.2000)
(25) ja (26) ja
(30) 11/61390 9 Mar/mar 1999 JP
(09.03.1999)
(43) 14 Sep/sep 2000 (14.09.2000)
(54) PROCESS FOR PRODUCING QUINA-
ZOLINE DERIVATIVE OR SALT THE-
REOF
PROCEDE DE PRODUCTION D’UN
DERIVE QUINAZOLINE OU D’UN
SEL DE CE DERIVE
(71) FUJISAWA PHARMACEUTICAL CO.,
LTD. [JP/JP]; 4–7, Doshomachi 3–chome,
Chuo–ku, Osaka–shi, Osaka 541–8514 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) FUKAGAWA, Masayasu [JP/JP]; 48,
Jinden, Kamiichimachi, Nakaniikawa–gun,
Toyama 930–0365 (JP). IEDA, Shigeru
[JP/JP]; 5–1–1, Mukogaoka, Sanda–shi,
Hyogo 669–1544 (JP). TSUBOI, Hiroyuki
[JP/JP]; 19–1, Ishizuminamimachi, Neyagawa–shi,
Osaka 572–0024 (JP). GOTO,
Shunsuke [JP/JP]; 5–5–35–701, Nankounaka,
Suminoe–ku, Osaka–shi, Osaka
559–0033 (JP). KAGARA, Kooji [JP/JP];
17–12, Onoharanishi 3–chome, Mino–shi,
Osaka 562–0032 (JP). UEMATSU, Ryoichi
[JP/JP]; 2–62–107, Takamatsu–cho,
Takarazuka–shi, Hyogo 665–0043 (JP).
NISIWAKI, Masanori [JP/JP]; 38–17,
Hashimotonishikarimata, Yawata–shi, Kyoto
614–8334 (JP).
(74) TABUSHI, Eiji; Fujisawa Pharmaceutical
Co., Ltd.Osaka Factory, 1–6, Kashima
2–chome, Yodogawa–ku, Osaka–shi, Osaka
532–8514 (JP).
(81) AE AL AM AT AU AZ BA BB BG BR BY
CA CH CN CU CZ DE DK EE ES FI GB
GD GE GH GM HR HU ID IL IN IS JP KE
KG KR KZ LC LK LR LS LT LU LV MD
MG MK MN MW MX NO NZ PL PT RO
RU SD SE SG SI SK SL TJ TM TR TT UA
UG US UZ VN YU ZA ZW; AP (GH GM
KE LS MW SD SL SZ TZ UG ZW); EA
(AM AZ BY KG KZ MD RU TJ TM); EP
(ATBECHCYDEDKESFIFRGBGR
IE IT LU MC NL PT SE); OA (BF BJ CF
CG CI CM GA GN GW ML MR NE SN TD
TG).