section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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37/2000<br />
13242 PCT Gazette - Section I - Gazette du PCT 14 Sep/sep 2000<br />
(54) PYRAN DERIVATIVES<br />
DERIVES PYRANNE<br />
(71) KABUSHIKI KAISHA HAYASHI-<br />
BARA SEIBUTSU KAGAKU KEN-<br />
KYUJO [JP/JP]; 2–3, Shimoishii 1–chome,<br />
Okayama–shi, Okayama 700–0907 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) SATSUKI, Makoto [JP/JP]; 996–28,<br />
Ooaza Hayashima, Hayashima–cho, Tsukubo–gun,<br />
Okayama 701–0300 (JP).<br />
SHINPO, Akira [JP/JP]; 2473–3, Nagahama,<br />
Ushimado–cho, Oku–gun, Okayama<br />
701–4301 (JP). OOGA, Yasuyo [JP/JP];<br />
10–2, Shimotsui 1–chome, Kurashiki–shi,<br />
Okayama 711–0927 (JP). SUGA, Sadaharu<br />
[JP/JP]; 1–7, Uno 8–chome, Tamano–shi,<br />
Okayama 706–0011 (JP). ODA, Atsushi<br />
[JP/JP]; Nippon Denki Kabushiki<br />
Gaisha–nai, 1–1, Miyazaki 4–chome,<br />
Miyamae–ku, Kawasaki–shi, Kanagawa<br />
216–8555 (JP). TADA, Hiroshi [JP/JP];<br />
Nippon Denki Kabushiki Gaisha–nai, 1–1,<br />
Miyazaki 4–chome, Miyamae–ku, Kawasaki–shi,<br />
Kanagawa 216–8555 (JP).<br />
SAKAGUCHI, Yoshikazu [JP/JP]; Nippon<br />
Denki Kabushiki Gaisha–nai, 1–1, Miyazaki<br />
4–chome, Miyamae–ku, Kawasaki–shi,<br />
Kanagawa 216–8555 (JP).<br />
(81) KR US; EP (AT BE CH CY DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE).<br />
(51) 7 C07D 413/04, 417/04, A01N 43/88<br />
(11) WO 00/53599 (13) A1<br />
(21) PCT/US00/03251<br />
(22) 8 Feb/fév 2000 (08.02.2000)<br />
(25) en (26) en<br />
(30) 09/264,310 8 Mar/mar 1999 US<br />
(08.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) PESTICIDAL HETERO–<br />
SUBSTITUTED OXADIAZINE<br />
COMPOUNDS<br />
COMPOSES D’OXADIAZINES<br />
HETERO–SUBSTITUEES<br />
(71) UNIROYAL CHEMICAL COMPANY,<br />
INC. [US/US]; <strong>World</strong> Headquarters, Middlebury,<br />
CT 06749 (US). UNIROYAL<br />
CHEMICAL CO./UNIROYAL CHEMI-<br />
CAL CIE. [CA/CA]; 25 Erb Street, Elmira,<br />
Ontario N3B 3A3 (CA).<br />
(72) DEKEYSER, Mark, Achiel; 333 Boxbury<br />
Drive, Waterloo, Ontario N2K 1W3 (CA).<br />
MCDONALD, Paul, Thomas; 43 Mirey<br />
Dam Road, Middlebury, CT 06762 (US).<br />
(74) REITENBACH, Daniel; Uniroyal Chemical<br />
Company, Inc., <strong>World</strong> Headquarters,<br />
Middlebury, CT 06749 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK EE ES FI<br />
GB GD GE GH GM HR HU ID IL IN IS JP<br />
KE KG KP KR KZ LC LK LR LS LT LU<br />
LV MD MG MK MN MW MX NO NZ PL<br />
PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG UZ VN YU ZA ZW; AP (GH<br />
GM KE LS MW SD SL SZ TZ UG ZW);<br />
EA (AM AZ BY KG KZ MD RU TJ TM);<br />
EP (AT BE CH CY DE DK ES FI FR GB<br />
GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
(51) 7 C07D 413/12, 417/12, 417/14, A61K<br />
31/454, A61P 43/00, 31/00, 29/00, 37/08,<br />
11/00, 19/02, 37/00, 35/00, 9/00<br />
(11) WO 00/53600 (13) A1<br />
(21) PCT/JP00/01479<br />
(22) 10 Mar/mar 2000 (10.03.2000)<br />
(25) ja (26) ja<br />
(30) 11/64194 11 Mar/mar 1999<br />
(11.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) NOVEL PIPERIDINE DERIVATIVES<br />
DERIVES PIPERIDINIQUES<br />
(71) BANYU PHARMACEUTICAL CO.,<br />
LTD. [JP/JP]; 2–3, Nihombashi Honcho<br />
2–chome, Chuo–ku, Tokyo 103–8416 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) NAYA, Akira [JP/JP]; Banyu Pharmaceutical<br />
Co., Ltd. Tsukuba Research<br />
Institute, 3, Okubo, Tsukuba–shi, Ibaraki<br />
300–2611 (JP). KOBAYASHI, Kensuke<br />
[JP/JP]; Banyu Pharmaceutical Co., Ltd.<br />
Tsukuba Research Institute, 3, Okubo,<br />
Tsukuba–shi, Ibaraki 300–2611 (JP). ISHI-<br />
KAWA, Makoto [JP/JP]; Banyu Pharmaceutical<br />
Co., Ltd. Tsukuba Research<br />
Institute, 3, Okubo, Tsukuba–shi, Ibaraki<br />
300–2611 (JP). SAEKI, Toshihiko [JP/JP];<br />
Banyu Pharmaceutical Co., Ltd. Tsukuba<br />
Research Institute, 3, Okubo, Tsukuba–shi,<br />
Ibaraki 300–2611 (JP). OHWAKI, Kenji<br />
[JP/JP]; Banyu Pharmaceutical Co., Ltd.<br />
Tsukuba Research Institute, 3, Okubo, Tsukuba–shi,<br />
Ibaraki 300–2611 (JP). OTAKE,<br />
Norikazu [JP/JP]; Banyu Pharmaceutical<br />
Co., Ltd. Tsukuba Research Institute, 3,<br />
Okubo, Tsukuba–shi, Ibaraki 300–2611<br />
(JP). NOGUCHI, Kazuhito [JP/JP]; Banyu<br />
Pharmaceutical Co., Ltd. Tsukuba Research<br />
Institute, 3, Okubo, Tsukuba–shi, Ibaraki<br />
300–2611 (JP).<br />
(74) BANYU PHARMACEUTICAL CO.,<br />
LTD.; 2–3, Nihombashi Honcho 2–chome,<br />
Chuo–ku, Tokyo 103–8416 (JP).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM DZ EE<br />
ES FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
(51) 7 C07D 417/12, 339/04, C07C 327/18,<br />
327/36, A61K 31/216, 31/192, 31/427,<br />
31/385<br />
(11) WO 00/53601 (13) A1<br />
(21) PCT/US00/05895<br />
(22) 7 Mar/mar 2000 (07.03.2000)<br />
(25) en (26) en<br />
(30) 09/264,370 8 Mar/mar 1999<br />
(08.03.1999)<br />
JP<br />
US<br />
(30) 09/497,324 3 Feb/fév 2000<br />
(03.02.2000)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) 1,2–DITHIOLANE DERIVATIVES<br />
DERIVES DE 1,2–DITHIOLANE<br />
US<br />
(71) THE UNIVERSITY OF MISSISSIPPI<br />
[US/US]; 1006 Natural Products Center,<br />
University, MS 38677 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) PERSHADSINGH, Harrihar, A.<br />
[US/US]; 404 Windsor Park Drive, Bakersfield,<br />
CA 93311 (US). AVERY, Mitchell,<br />
A. [US/US]; 303 Woodland Hills Drive,<br />
Oxford, MS 38655 (US).<br />
(74) SNYDER, Joseph, R. et al. / etc.; Townsend<br />
and Townsend and Crew LLP, Two Embarcadero<br />
Center, 8th floor, San Francisco,<br />
CA 94111 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 471/04, 471/08, 401/06, 401/12,<br />
A61K 31/44<br />
(11) WO 00/53602 (13) A1<br />
(21) PCT/US00/05799<br />
(22) 6 Mar/mar 2000 (06.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,620 10 Mar/mar 1999<br />
(10.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />
TAGONISTS OF GONADOTROPIN RE-<br />
LEASING HORMONE<br />
COMPOSES 6–AZAINDOLE UTILISES<br />
COMME ANTAGONISTES D’UNE<br />
HORMONE LIBERANT LA GONADO-<br />
TROPINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065–0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WALSH, Thomas, F. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065–0907 (US). UJJAINWALLA,<br />
Feroze [GB/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065–0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065–0907 (US).