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37/2000<br />

13160 PCT Gazette - Section I - Gazette du PCT 14 Sep/sep 2000<br />

(43) 14 Sep/sep 2000 (14.09.2000)<br />

(54) 3–CYCLOPROPYLMETHOXY–<br />

4–DIFLUOROMETHOXY–N–<br />

(3,5–DICHLOROPYRID–4–<br />

YL)BENZAMIDE IN THE TREAT-<br />

MENT OF MULTIPLE SCLEROSIS<br />

3–CYCLOPROPYLMETHOXY–<br />

4–DIFLUOROMETHOXY–N–<br />

(3,5–DICHLOROPYRID–4–<br />

YL)BENZAMIDE POUR LE TRAI-<br />

TEMENT<br />

PLAQUES<br />

DE LA SCLEROSE EN<br />

(71) BYK GULDEN LOMBERG CHE-<br />

MISCHE FABRIK GMBH [DE/DE];<br />

Byk–Gulden–Strasse 2, D–78467 Konstanz<br />

(DE).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72) AMSCHLER, Hermann (deceased /<br />

décédé).<br />

(72) HATZELMANN, Armin; Alter Wall 3,<br />

D–78467 Konstanz (DE). SCHUDT, Christian;<br />

Schützenstrasse 20, D–78462 Konstanz<br />

(DE).<br />

(for all designated States except / pour tous<br />

les États désignés sauf CA US)<br />

(72, 75) KLEY, Hans–Peter [DE/DE]; Im Weinberg<br />

3b, D–78476 Allensbach (DE). SAN-<br />

DERS, Karl [DE/DE]; Mainaustrasse 207d,<br />

D–78464 Konstanz (DE).<br />

(74) BYK GULDEN LOMBERG<br />

CHEMISCHE FABRIK GMBH;<br />

Byk–Gulden–Strasse 2, D–78467 Konstanz<br />

(DE).<br />

(81) AE AL AU BA BG BR CA CN CZ EE GE<br />

HR HU ID IL IN JP KR LT LV MK MX<br />

NO NZ PL RO SG SI SK TR UA US VN<br />

YU ZA ZW; EA (AM AZ BY KG KZ MD<br />

RU TJ TM); EP (AT BE CH CY DE DK ES<br />

FI FR GB GR IE IT LU MC NL PT SE).<br />

(51) 7 A61K 31/445, 31/16<br />

(11) WO 00/53183 (13) A1<br />

(21) PCT/US00/03782<br />

(22) 12 Feb/fév 2000 (12.02.2000)<br />

(25) en (26) en<br />

(30) 09/265,502 10 Mar/mar 1999<br />

(10.03.1999)<br />

(43) 14 Sep/sep 2000 (14.09.2000)<br />

US<br />

(54) MEDICAMENT AGAINST DYS-<br />

MENORRHOEA AND PREMENS-<br />

TRUAL SYNDROME<br />

MEDICAMENT CONTRE LA DYS-<br />

MENORRHEE ET LE SYNDROME<br />

PREMENSTRUEL<br />

(63) US 08/800,737 (CIP)<br />

15 Feb/fév 1997 (15.02.1997)<br />

(71) EDELSTAM INC. [US/US]; Fasth Law<br />

Offices, 509 Queensferry Road, Cary, NC<br />

27511–6319 (US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(71, 72) EDELSTAM, Greta [SE/SE]; Saltangsvagen<br />

2, S–131 50 Saltsjo–Duvnas (SE).<br />

(74) FASTH, Rolf; Fasth Law Offices, 509<br />

Queensferry Road, Cary, NC 27511–6319<br />

(US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CU CZ DE DK EE ES FI GB<br />

GD GE GH GM HR HU ID IL IN IS JP KE<br />

KG KP KR KZ LC LK LR LS LT LU LV<br />

MD MG MK MN MW MX NO NZ PL PT<br />

RO RU SD SE SG SI SK SL TJ TM TR TT<br />

UA UG US UZ VN YU ZA ZW; AP (GH<br />

GM KE LS MW SD SL SZ TZ UG ZW);<br />

EA (AM AZ BY KG KZ MD RU TJ TM);<br />

EP (AT BE CH CY DE DK ES FI FR GB<br />

GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN GW ML MR NE SN<br />

TD TG).<br />

Published / Publiée :(a)<br />

(51) 7 A61K 31/517, 9/70, A61P 13/02, 9/12<br />

(11) WO 00/53184 (13) A1<br />

(21) PCT/JP00/01429<br />

(22) 9 Mar/mar 2000 (09.03.2000)<br />

(25) ja (26) ja<br />

(30) 11/64274 11 Mar/mar 1999 JP<br />

(11.03.1999)<br />

(43) 14 Sep/sep 2000 (14.09.2000)<br />

(54) DRUG COMPOSITION FOR PERCU-<br />

TANEOUS ABSORPTION<br />

COMPOSITION MEDICAMENTEUSE<br />

A ABSORPTION PERCUTANEE<br />

(71) SAITAMA DAIICHI PHARMACEU-<br />

TICAL CO., LTD. [JP/JP]; 8–1, Minamisakae–cho,<br />

Kasukabe–shi, Saitama<br />

344–0057 (JP). MITSUBISHI CHEMI-<br />

CAL CORPORATION [JP/JP]; 5–2,<br />

Marunouchi 2–chome, Chiyoda–ku, Tokyo<br />

100–0005 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) YAMAUCHI, Hitoshi [JP/JP]; Daiichi<br />

Pharmaceutical Co., Ltd., Tokyo R<br />

& DCenter, 16–13, Kita–kasai 1–chome,<br />

Edogawa–ku, Tokyo 134–8630 (JP). NA-<br />

KAJIMA, Noriko [JP/JP]; Saitama Daiichi<br />

Pharmaceutical Co., Ltd., 8–1, Minamisakae–cho,<br />

Kasukabe–shi, Saitama 344–0057<br />

(JP). NISHI, Hiroyoshi [JP/JP]; Mitsubishi<br />

Tokyo Pharmaceuticals, Inc., 2–6, Nihonbashi–honcho<br />

2–chome, Chuo–ku, Tokyo<br />

103–8405 (JP). MATSUOKA, Yoshinori<br />

[JP/JP]; Mitsubishi Tokyo Pharmaceuticals,<br />

Inc., 2–6, Nihonbashi–honcho 2–chome,<br />

Chuo–ku, Tokyo 103–8405 (JP). YANO,<br />

Shinji [JP/JP]; Mitsubishi Tokyo Pharmaceuticals,<br />

Inc., 2–6, Nihonbashi–honcho<br />

2–chome, Chuo–ku, Tokyo 103–8405 (JP).<br />

(74) IMAMURA, Masazumi et al. / etc.;<br />

5th Floor, KRF Building, 5–5, Kyobashi<br />

1–chome, Chuo–ku, Tokyo 104–0031 (JP).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM DZ EE<br />

ES FI GB GD GE GH GM HR HU ID IL IN<br />

IS JP KE KG KR KZ LC LK LR LS LT LU<br />

LV MA MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM<br />

TR TT TZ UA UG US UZ VN YU ZA ZW;<br />

AP (GH GM KE LS MW SD SL SZ TZ UG<br />

ZW); EA (AM AZ BY KG KZ MD RU TJ<br />

TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF<br />

BJ CF CG CI CM GA GN GW ML MR NE<br />

SN TD TG).<br />

(51) 7 A61K 31/519, 31/4985, 31/5025, 31/437,<br />

A61P 5/04, 5/10, 15/02, 15/18, 17/14,<br />

35/00, 37/02, C07D 519/00<br />

(11) WO 00/53185 (13) A1<br />

(21) PCT/US00/05836<br />

(22) 6 Mar/mar 2000 (06.03.2000)<br />

(25) en (26) en<br />

(30) 60/123,616 10 Mar/mar 1999 US<br />

(10.03.1999)<br />

(43) 14 Sep/sep 2000 (14.09.2000)<br />

(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />

TAGONISTS OF GONADOTROPIN RE-<br />

LEASING HORMONE<br />

COMPOSES 6–AZAINDOLE UTILISES<br />

COMME ANTAGONISTES D’UNE<br />

HORMONE LIBERANT LA GONADO-<br />

TROPINE<br />

(71) MERCK & CO., INC. [US/US]; 126 East<br />

Lincoln Avenue, Rahway, NJ 07065–0907<br />

(US).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) WALSH, Thomas, F. [US/US];<br />

126 East Lincoln Avenue, Rahway, NJ<br />

07065–0907 (US). UJJAINWALLA,<br />

Feroze [GB/US]; 126 East Lincoln Avenue,<br />

Rahway, NJ 07065–0907 (US).<br />

(74) MERCK & CO., INC.; 126 East Lincoln<br />

Avenue, Rahway, NJ 07065–0907 (US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES<br />

FI GB GD GE GH GM HR HU ID IL IN<br />

IS JP KE KG KR KZ LC LK LR LS LT LU<br />

LV MA MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM<br />

TR TT TZ UA UG US UZ VN YU ZA ZW;<br />

AP (GH GM KE LS MW SD SL SZ TZ UG<br />

ZW); EA (AM AZ BY KG KZ MD RU TJ<br />

TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF<br />

BJ CF CG CI CM GA GN GW ML MR NE<br />

SN TD TG).<br />

(51) 7 A61K 31/57, 31/135<br />

(11) WO 00/53186<br />

(21) PCT/US99/05188<br />

(13) A1<br />

(22) 10 Mar/mar 1999 (10.03.1999)<br />

(25) en (26) en<br />

(43) 14 Sep/sep 2000 (14.09.2000)<br />

(54) TOPICAL COMPOSITIONS CONTAI-<br />

NING A COMBINATION OF AN ANTI-<br />

FUNGAL AGENT AND A STEROIDAL<br />

ANTIINFLAMMATORY AGENT<br />

COMPOSITIONS TOPIQUES CONTE-<br />

NANT UNE COMBINAISON D’UN<br />

AGENT ANTIFONGIQUE ET D’UN<br />

AGENT ANTI–INFLAMMATOIRE<br />

STEROIDIQUE<br />

(71) PENEDERM, INC. [US/US]; Suite A, 320<br />

Lakeside Drive, Foster City, CA 94404 (US).<br />

(72) QUIGLEY, John, W., Jr.; 603 San Nicholas<br />

Lane, Foster City, CA 94404 (US). HOU,<br />

Sui, Yuen, Eddie; 380 Shad Court, Foster<br />

City, CA 94404 (US). CHAUDHURI,<br />

Bhaskar; 10281 Parlett Place, Cupertino,<br />

CA 95014 (US).

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