section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
Create successful ePaper yourself
Turn your PDF publications into a flip-book with our unique Google optimized e-Paper software.
37/2000<br />
13160 PCT Gazette - Section I - Gazette du PCT 14 Sep/sep 2000<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) 3–CYCLOPROPYLMETHOXY–<br />
4–DIFLUOROMETHOXY–N–<br />
(3,5–DICHLOROPYRID–4–<br />
YL)BENZAMIDE IN THE TREAT-<br />
MENT OF MULTIPLE SCLEROSIS<br />
3–CYCLOPROPYLMETHOXY–<br />
4–DIFLUOROMETHOXY–N–<br />
(3,5–DICHLOROPYRID–4–<br />
YL)BENZAMIDE POUR LE TRAI-<br />
TEMENT<br />
PLAQUES<br />
DE LA SCLEROSE EN<br />
(71) BYK GULDEN LOMBERG CHE-<br />
MISCHE FABRIK GMBH [DE/DE];<br />
Byk–Gulden–Strasse 2, D–78467 Konstanz<br />
(DE).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72) AMSCHLER, Hermann (deceased /<br />
décédé).<br />
(72) HATZELMANN, Armin; Alter Wall 3,<br />
D–78467 Konstanz (DE). SCHUDT, Christian;<br />
Schützenstrasse 20, D–78462 Konstanz<br />
(DE).<br />
(for all designated States except / pour tous<br />
les États désignés sauf CA US)<br />
(72, 75) KLEY, Hans–Peter [DE/DE]; Im Weinberg<br />
3b, D–78476 Allensbach (DE). SAN-<br />
DERS, Karl [DE/DE]; Mainaustrasse 207d,<br />
D–78464 Konstanz (DE).<br />
(74) BYK GULDEN LOMBERG<br />
CHEMISCHE FABRIK GMBH;<br />
Byk–Gulden–Strasse 2, D–78467 Konstanz<br />
(DE).<br />
(81) AE AL AU BA BG BR CA CN CZ EE GE<br />
HR HU ID IL IN JP KR LT LV MK MX<br />
NO NZ PL RO SG SI SK TR UA US VN<br />
YU ZA ZW; EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE).<br />
(51) 7 A61K 31/445, 31/16<br />
(11) WO 00/53183 (13) A1<br />
(21) PCT/US00/03782<br />
(22) 12 Feb/fév 2000 (12.02.2000)<br />
(25) en (26) en<br />
(30) 09/265,502 10 Mar/mar 1999<br />
(10.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) MEDICAMENT AGAINST DYS-<br />
MENORRHOEA AND PREMENS-<br />
TRUAL SYNDROME<br />
MEDICAMENT CONTRE LA DYS-<br />
MENORRHEE ET LE SYNDROME<br />
PREMENSTRUEL<br />
(63) US 08/800,737 (CIP)<br />
15 Feb/fév 1997 (15.02.1997)<br />
(71) EDELSTAM INC. [US/US]; Fasth Law<br />
Offices, 509 Queensferry Road, Cary, NC<br />
27511–6319 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(71, 72) EDELSTAM, Greta [SE/SE]; Saltangsvagen<br />
2, S–131 50 Saltsjo–Duvnas (SE).<br />
(74) FASTH, Rolf; Fasth Law Offices, 509<br />
Queensferry Road, Cary, NC 27511–6319<br />
(US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CU CZ DE DK EE ES FI GB<br />
GD GE GH GM HR HU ID IL IN IS JP KE<br />
KG KP KR KZ LC LK LR LS LT LU LV<br />
MD MG MK MN MW MX NO NZ PL PT<br />
RO RU SD SE SG SI SK SL TJ TM TR TT<br />
UA UG US UZ VN YU ZA ZW; AP (GH<br />
GM KE LS MW SD SL SZ TZ UG ZW);<br />
EA (AM AZ BY KG KZ MD RU TJ TM);<br />
EP (AT BE CH CY DE DK ES FI FR GB<br />
GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN GW ML MR NE SN<br />
TD TG).<br />
Published / Publiée :(a)<br />
(51) 7 A61K 31/517, 9/70, A61P 13/02, 9/12<br />
(11) WO 00/53184 (13) A1<br />
(21) PCT/JP00/01429<br />
(22) 9 Mar/mar 2000 (09.03.2000)<br />
(25) ja (26) ja<br />
(30) 11/64274 11 Mar/mar 1999 JP<br />
(11.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) DRUG COMPOSITION FOR PERCU-<br />
TANEOUS ABSORPTION<br />
COMPOSITION MEDICAMENTEUSE<br />
A ABSORPTION PERCUTANEE<br />
(71) SAITAMA DAIICHI PHARMACEU-<br />
TICAL CO., LTD. [JP/JP]; 8–1, Minamisakae–cho,<br />
Kasukabe–shi, Saitama<br />
344–0057 (JP). MITSUBISHI CHEMI-<br />
CAL CORPORATION [JP/JP]; 5–2,<br />
Marunouchi 2–chome, Chiyoda–ku, Tokyo<br />
100–0005 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) YAMAUCHI, Hitoshi [JP/JP]; Daiichi<br />
Pharmaceutical Co., Ltd., Tokyo R<br />
& DCenter, 16–13, Kita–kasai 1–chome,<br />
Edogawa–ku, Tokyo 134–8630 (JP). NA-<br />
KAJIMA, Noriko [JP/JP]; Saitama Daiichi<br />
Pharmaceutical Co., Ltd., 8–1, Minamisakae–cho,<br />
Kasukabe–shi, Saitama 344–0057<br />
(JP). NISHI, Hiroyoshi [JP/JP]; Mitsubishi<br />
Tokyo Pharmaceuticals, Inc., 2–6, Nihonbashi–honcho<br />
2–chome, Chuo–ku, Tokyo<br />
103–8405 (JP). MATSUOKA, Yoshinori<br />
[JP/JP]; Mitsubishi Tokyo Pharmaceuticals,<br />
Inc., 2–6, Nihonbashi–honcho 2–chome,<br />
Chuo–ku, Tokyo 103–8405 (JP). YANO,<br />
Shinji [JP/JP]; Mitsubishi Tokyo Pharmaceuticals,<br />
Inc., 2–6, Nihonbashi–honcho<br />
2–chome, Chuo–ku, Tokyo 103–8405 (JP).<br />
(74) IMAMURA, Masazumi et al. / etc.;<br />
5th Floor, KRF Building, 5–5, Kyobashi<br />
1–chome, Chuo–ku, Tokyo 104–0031 (JP).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM DZ EE<br />
ES FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KR KZ LC LK LR LS LT LU<br />
LV MA MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(51) 7 A61K 31/519, 31/4985, 31/5025, 31/437,<br />
A61P 5/04, 5/10, 15/02, 15/18, 17/14,<br />
35/00, 37/02, C07D 519/00<br />
(11) WO 00/53185 (13) A1<br />
(21) PCT/US00/05836<br />
(22) 6 Mar/mar 2000 (06.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,616 10 Mar/mar 1999 US<br />
(10.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />
TAGONISTS OF GONADOTROPIN RE-<br />
LEASING HORMONE<br />
COMPOSES 6–AZAINDOLE UTILISES<br />
COMME ANTAGONISTES D’UNE<br />
HORMONE LIBERANT LA GONADO-<br />
TROPINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065–0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WALSH, Thomas, F. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065–0907 (US). UJJAINWALLA,<br />
Feroze [GB/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065–0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065–0907 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KR KZ LC LK LR LS LT LU<br />
LV MA MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(51) 7 A61K 31/57, 31/135<br />
(11) WO 00/53186<br />
(21) PCT/US99/05188<br />
(13) A1<br />
(22) 10 Mar/mar 1999 (10.03.1999)<br />
(25) en (26) en<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) TOPICAL COMPOSITIONS CONTAI-<br />
NING A COMBINATION OF AN ANTI-<br />
FUNGAL AGENT AND A STEROIDAL<br />
ANTIINFLAMMATORY AGENT<br />
COMPOSITIONS TOPIQUES CONTE-<br />
NANT UNE COMBINAISON D’UN<br />
AGENT ANTIFONGIQUE ET D’UN<br />
AGENT ANTI–INFLAMMATOIRE<br />
STEROIDIQUE<br />
(71) PENEDERM, INC. [US/US]; Suite A, 320<br />
Lakeside Drive, Foster City, CA 94404 (US).<br />
(72) QUIGLEY, John, W., Jr.; 603 San Nicholas<br />
Lane, Foster City, CA 94404 (US). HOU,<br />
Sui, Yuen, Eddie; 380 Shad Court, Foster<br />
City, CA 94404 (US). CHAUDHURI,<br />
Bhaskar; 10281 Parlett Place, Cupertino,<br />
CA 95014 (US).