section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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37/2000<br />
14 Sep/sep 2000 PCT Gazette - Section I - Gazette du PCT 13159<br />
OHTOMO, Kazumi [JP/JP]; 11–3, Funakicho,<br />
Ibaraki–shi, Osaka 567–0828 (JP).<br />
(74) KOTANI, Etsuji et al. / etc.; Sumisei<br />
Naniwasuji Honmachi Building, 3–2,<br />
Utsubohonmachi 2–chome, Nishi–ku,<br />
Osaka–shi, Osaka 550–0004 (JP).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
(51) 7 A61K 31/435, C07D 471/04<br />
(11) WO 00/53178 (13) A1<br />
(21) PCT/US00/05814<br />
(22) 6 Mar/mar 2000 (06.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,649 10 Mar/mar 1999<br />
(10.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />
TAGONISTS OF GONADOTROPIN RE-<br />
LEASING HORMONE<br />
COMPOSES 6–AZAINDOLE UTILISES<br />
COMME ANTAGONISTES D’UNE<br />
HORMONE LIBERANT LA GONADO-<br />
TROPINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065–0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WALSH, Thomas, F. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065–0907 (US). UJJAINWALLA,<br />
Feroze [GB/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065–0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065–0907 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KR KZ LC LK LR LS LT LU<br />
LV MA MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 A61K 31/435, C07D 471/04<br />
(11) WO 00/53179 (13) A1<br />
(21) PCT/US00/05815<br />
(22) 6 Mar/mar 2000 (06.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,648 10 Mar/mar 1999<br />
(10.03.1999)<br />
US<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />
TAGONISTS OF GONADOTROPIN RE-<br />
LEASING HORMONE<br />
COMPOSES 6–AZAINDOLE UTILISES<br />
COMME ANTAGONISTES D’UNE<br />
HORMONE LIBERANT LA GONADO-<br />
TROPINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065–0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WALSH, Thomas, F. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065–0907 (US). UJJAINWALLA,<br />
Feroze [GB/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065–0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065–0907 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KR KZ LC LK LR LS LT LU<br />
LV MA MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(51) 7 A61K 31/437, 31/435, A61P 5/04, C07D<br />
471/04, 221/02<br />
(11) WO 00/53180<br />
(21) PCT/US00/05727<br />
(13) A1<br />
(22) 6 Mar/mar 2000 (06.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,639 10 Mar/mar 1999<br />
(10.03.1999)<br />
US<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />
TAGONISTS OF GONADOTROPIN RE-<br />
LEASING HORMONE<br />
COMPOSES DE 6–AZAINDOLE AN-<br />
TAGONISTES DE LA GONADOLIBE-<br />
RINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065–0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WALSH, Thomas, F. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065–0907 (US). UJJAINWALLA,<br />
Feroze [GB/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065–0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065–0907 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KR KZ LC LK LR LS LT LU<br />
LV MA MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(51) 7 A61K 31/437, 31/435, 31/495, 31/497,<br />
31/498, 31/506, 31/517, 31/541, 31/5355,<br />
A61P 5/04, C07D 221/22, 239/74, 241/42,<br />
401/12, 401/14, 403/12, 403/14, 413/12,<br />
413/14, 417/12, 417/14, 471/04, 473/00,<br />
475/00, 487/04<br />
(11) WO 00/53181 (13) A1<br />
(21) PCT/US00/05933<br />
(22) 6 Mar/mar 2000 (06.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,640 10 Mar/mar 1999<br />
(10.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) 6–AZAINDOLE COMPOUNDS AS AN-<br />
TAGONISTS OF GONADOTROPIN RE-<br />
LEASING HORMONE<br />
COMPOSES DE 6–AZAINDOLE<br />
COMME ANTAGONISTES DE LA<br />
GONADOLIBERINE<br />
(71) MERCK & CO., INC. [US/US]; 126 East<br />
Lincoln Avenue, Rahway, NJ 07065–0907<br />
(US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) WALSH, Thomas, F. [US/US];<br />
126 East Lincoln Avenue, Rahway, NJ<br />
07065–0907 (US). UJJAINWALLA,<br />
Feroze [GB/US]; 126 East Lincoln Avenue,<br />
Rahway, NJ 07065–0907 (US).<br />
(74) MERCK & CO., INC.; 126 East Lincoln<br />
Avenue, Rahway, NJ 07065–0907 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KR KZ LC LK LR LS LT LU<br />
LV MA MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT TZ UA UG US UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(51) 7 A61K 31/44<br />
(11) WO 00/53182 (13) A2<br />
(21) PCT/EP00/01703<br />
(22) 1 Mar/mar 2000 (01.03.2000)<br />
(25) en (26) en<br />
(30) 99104793.7 10 Mar/mar 1999<br />
(10.03.1999)<br />
EP