section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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37/2000<br />
13244 PCT Gazette - Section I - Gazette du PCT 14 Sep/sep 2000<br />
(71) SIGMA–TAU INDUSTRIE FARMACEU-<br />
TICHE S.P.A. [IT/IT]; Viale Shakespeare,<br />
47, I–00144 Rome (IT). ISTITUTO NA-<br />
ZIONALE PER LO STUDIO E LA<br />
CURA DEI TUMORI [IT/IT]; Via Venezian,<br />
1, I–20133 Milan (IT).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) PENCO, Sergio [IT/IT]; Via Milly<br />
Carla Mignone, 5, I–20133 Milan (IT).<br />
MERLINI, Lucio [IT/IT]; Via Carlo Crivelli,<br />
14, I–20122 Milan (IT). ZUNINO,<br />
Franco [IT/IT]; Istituto Nazionale per lo<br />
Studio e la Cura dei Tum, ori, Via Venezian,<br />
1, I–20133 Milan (IT). CARMINATI, Paolo<br />
[IT/IT]; Sigma–Tau Industrie Farmaceutiche<br />
Riunite S.p.A., Via Pontina, Km. 30,400,<br />
I–00040 Pomezia (IT).<br />
(74) SPADARO, Marco; Sigma–Tau Industrie<br />
Farmaceutiche Riunite S.p.A., Viale Shakespeare,<br />
47, I–00144 Rome (IT).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM DZ EE<br />
ES FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 491/22, A61K 31/44, A61P 25/00 //<br />
(C07D 491/22, 311:00, 221:00, 221:00,<br />
209:00)<br />
(11) WO 00/53608 (13) A1<br />
(21) PCT/FR00/00502<br />
(22) 1 Mar/mar 2000 (01.03.2000)<br />
(25) fr (26) fr<br />
(30) 99/02784 5 Mar/mar 1999<br />
(05.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
FR<br />
(54) PYRIDOPYRANOAZEPINE DERIVA-<br />
TIVES, PREPARATION AND THERA-<br />
PEUTIC USE<br />
DERIVES DE PYRIDOPYRANOA-<br />
ZEPINES, LEUR PREPARATION ET<br />
LEUR APPLICATION EN THERAPEU-<br />
TIQUE<br />
(71) SANOFI–SYNTHELABO [FR/FR]; 174,<br />
avenue de France, F–75013 Paris (FR).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) GALLI, Frédéric [FR/FR]; 6, avenue<br />
de Rueil, F–92420 Vaucresson (FR). JE-<br />
GHAM, Samir [TN/FR]; 201, chemin de la<br />
Draille, F–34980 Montferrier–sur–Lez (FR).<br />
LOCHEAD, Alistair [GB/FR]; 95, rue de<br />
Paris, F–94220 Charenton (FR). SAMSON,<br />
Axelle [FR/FR]; 15, rue Louis Braille,<br />
F–75012 Paris (FR).<br />
(74) LUDWIG, Jacques; Sanofi–Synthelabo,<br />
174, avenue de France, F–75013 Paris (FR).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
(51) 7 C07D 501/04, 501/12, 501/24, 501/00<br />
(11) WO 00/53609 (13) A1<br />
(21) PCT/IB00/00240<br />
(22) 8 Mar/mar 2000 (08.03.2000)<br />
(25) en (26) en<br />
(30) 09/264,977 9 Mar/mar 1999<br />
(09.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) PROCESS FOR THE PREPARATION<br />
OF CEFUROXIME<br />
PROCEDE DE PREPARATION DE CE-<br />
FUROXIME<br />
(71) RANBAXY LABORATORIES LIMITED<br />
[IN/IN]; 19, Nehru Place, New Delhi 110<br />
019 (IN).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) HANDA, Vijay, Kumar [IN/IN];<br />
K–1/7, Chittaranjan Enclave, New Dehli 110<br />
019 (IN). DANDALA, Ramesh [IN/IN];<br />
110, Doctors Hostel II, Kidwai Nagar<br />
(West), New Delhi 110 023 (IN). KHANNA,<br />
JagMohan [IN/IN]; J1/23, DLF Qutab Enclave,<br />
Phase II, Gurgaon, Haryana 122 001<br />
(IN).<br />
(74) RANBAXY LABORATORIES LIMI-<br />
TED; Deshmukh, Jayadeep, R., Ranbaxy<br />
Pharmaceuticals Inc., Suite 2100, 600 College<br />
Road East, Princeton, NJ 08540 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM DZ EE<br />
ES FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 513/04, 333/38, A61K 31/435,<br />
A61P 31/22, 31/20 // (C07D 513/04,<br />
333:00, 221:00)<br />
(11) WO 00/53610 (13) A2<br />
(21) PCT/US00/05937<br />
(22) 7 Mar/mar 2000 (07.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,660 9 Mar/mar 1999<br />
(09.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) 4–OXO–4,7–DIHYDRO–THIENO[2,3–<br />
b]PYRIDINE–5–CARBOXAMIDES AS<br />
ANTIVIRAL AGENTS<br />
AGENTS ANTIVIRAUX DE 4–<br />
OXO–4,7–DIHYDRO–THIENO[2,3–<br />
b]PYRIDINE–5–CARBOXAMIDES<br />
(71) PHARMACIA & UPJOHN COMPANY<br />
[US/US]; 301 Henrietta Street, Kalamazoo,<br />
MI 49001 (US).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) SCHNUTE, Mark, E. [US/US]; 4459<br />
Wimbleton Way, Kalamazoo, MI 49009<br />
(US). CUDAHY, Michele, M. [US/US];<br />
6047–D San Gabriel Drive, Kalamazoo, MI<br />
49009 (US). SCOTT, Allen [US/US]; 5287<br />
Saddle Club Drive, Kalamazoo, MI 49009<br />
(US).<br />
(74) VIKSNINS, Ann, S.; Schwegman, Lundberg,<br />
Woessner & Kluth, P.O. Box 2938,<br />
Minneapolis, MN 55402 (US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
(51) 7 C07F 3/00, 5/00, 5/02, 5/06, 7/02, 7/22,<br />
7/28, 7/30, 9/02, 9/66, 9/94<br />
(11) WO 00/53611 (13) A1<br />
(21) PCT/US00/06293<br />
(22) 10 Mar/mar 2000 (10.03.2000)<br />
(25) en (26) en<br />
(30) 60/123,599 10 Mar/mar 1999<br />
(10.03.1999)<br />
(43) 14 Sep/sep 2000 (14.09.2000)<br />
US<br />
(54) WEAKLY COORDINATING<br />
ANIONS CONTAINING POLY-<br />
FLUOROALKOXIDE LIGANDS<br />
ANIONS A COORDINATION FAIBLE<br />
CONTENANT DES LIGANDS POLY-<br />
FLUOROALCOXYDE<br />
(71) COLORADO STATE UNIVERSITY RE-<br />
SEARCH FOUNDATION [US/US]; P.O.<br />
Box 483, Fort Collins, CO 80522 (US).<br />
(72) STRAUSS, Steven, H.; 5849 Plateau Court,<br />
Fort Collins, CO 80526 (US). NOLAN,<br />
Benjamin, G.; 1225 W. Prospect Road<br />
#J202, Fort Collins, CO 80526 (US). FAU-<br />
BER, Benjamin, P.; 260 W. Prospect Road<br />
#102, Fort Collins, CO 80526 (US).<br />
(74) CHA, Don, D. et al. / etc.; Sheridan Ross<br />
P.C., Suite 1200, 1560 Broadway, Denver,<br />
CO 80202–5141 (US).