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42/1998<br />

14670 PCT Gazette - Section I - Gazette du PCT 22 Oct/oct 1998<br />

(74) PALMBERG, Arleen et al. / etc.; Eli Lilly and<br />

Company, Lilly Corporate Center, Indianapolis, IN<br />

46285 (US).<br />

(81) AL AM AU AZ BA BB BG BR BY CA CN CU<br />

CZ EE GE GH GM GW HU ID IL IS JP KE KG<br />

KP KR KZ LC LK LR LS LT LV MD MG MK<br />

MN MW MX NO NZ PL RO RU SD SG SI SK<br />

SL TJ TM TR TT UA UG US UZ VN YU ZW;<br />

AP (GH GM KE LS MW SD SZ UG ZW); EA<br />

(AM AZ BY KG KZ MD RU TJ TM); OA (BF BJ<br />

CF CG CI CM GA GN ML MR NE SN TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/46231 (13) A1<br />

(21) PCT/US97/06187<br />

(22) 15 Apr/avr 1997 (15.04.1997)<br />

(25) en (26) en<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 A61K 31/505, C07D 239/06, 239/14<br />

(54) • MUSCARINIC AGONIST COMPOUNDS<br />

• COMPOSES AGONISTES MUSCARINIQUES<br />

(71) THE UNIVERSITY OF TOLEDO [US/US];<br />

2801 W. Bancroft Street, Toledo, OH 43606–3390<br />

(US).<br />

(71, 72) OJO, Babatunde [NG/US]; Apartment H,<br />

4119 Townhouse Road, Richmond, VA 23228<br />

(US). DUNBAR, Philip, G. [US/US]; South<br />

13224 Clear Lake Road, Medical Lake, WA 99022<br />

(US).<br />

(74) MEENAN, Larry, R. et al. / etc.; Brinks Hofer<br />

Gilson & Lione, 1130 Edison Plaza, Toledo, OH<br />

43604–1537 (US).<br />

(81) AL AM AT AU AZ BB BG BR BY CA CH CN<br />

CZ DE DK EE ES FI GB GE HU IL IS JP KE KG<br />

KP KR KZ LK LR LS LT LU LV MD MG MK<br />

MN MW MX NO NZ PL PT RO RU SD SE SG<br />

SI SK TJ TM TR TT UA UG UZ VN; AP (GH<br />

KE LS MW SD SZ UG); EA (AM AZ BY KG KZ<br />

MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN ML MR NE SN TD TG).<br />

(11) WO 98/46232 (13) A1<br />

(21) PCT/US97/06218<br />

(22) 15 Apr/avr 1997 (15.04.1997)<br />

(25) en (26) en<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 A61K 31/505, C07D 239/06<br />

(54) • MUSCARINIC AGONISTS<br />

• AGONISTES MUSCARINIQUES<br />

(71) THE UNIVERSITY OF TOLEDO [US/US];<br />

2801 W. Bancroft, Toledo, OH 43606–3390 (US).<br />

(72) MESSER, William, S., Jr.; 2619 Algonquin Parkway,<br />

Toledo, OH 43606 (US). OJO, Babatunde;<br />

Apartment H, 4119 Townhouse Road, Richmond,<br />

VA 23228 (US).<br />

(74) MEENAN, Larry, R. et al. / etc.; Brinks Hofer<br />

Gilson & Lione, 1130 Edison Plaza, Toledo, OH<br />

43604–1537 (US).<br />

(81) AL AM AT AU AZ BB BG BR BY CA CH CN<br />

CZ DE DK EE ES FI GB GE HU IL IS JP KE KG<br />

KP KR KZ LK LR LS LT LU LV MD MG MK<br />

MN MW MX NO NZ PL PT RO RU SD SE SG<br />

SI SK TJ TM TR TT UA UG UZ VN; AP (GH<br />

KE LS MW SD SZ UG); EA (AM AZ BY KG KZ<br />

MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN ML MR NE SN TD TG).<br />

(11) WO 98/46233 (13) A1<br />

(21) PCT/IT98/00076<br />

(22) 3 Apr/avr 1998 (03.04.1998)<br />

(25) en (26) en<br />

(31) RM97A000217 (32) 16 Apr/avr 1997 (33) IT<br />

(16.04.1997)<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 A61K 31/565<br />

(54) • OSTEOBLAST–PROMOTING PHARMACEU-<br />

TICAL COMPOSITION COMPRISING A<br />

CARNITINE COMPOUND AND DHEA OR<br />

DHEA–S<br />

• COMPOSITION PHARMACEUTIQUE STI-<br />

MULANT LES OSTEOBLASTES, CONTE-<br />

NANT UN COMPOSE DE CARNITINE ET<br />

DE LA DHEA OU DHEA–S<br />

(71) SIGMA–TAU INDUSTRIE FARMACEUTICHE<br />

RIUNITE S.P.A. [IT/IT]; Viale Shakespeare, 47,<br />

I–00144 Rome (IT).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) CAVAZZA, Claudio [IT/IT]; Piazza Campitelli,<br />

2, I–00186 Rome (IT).<br />

(74) SIGMA–TAU INDUSTRIE FARMACEUTICHE<br />

RIUNITE S.P.A.; Viale Shakespeare, 47, I–00144<br />

Rome (IT).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/46234 (13) A1<br />

(21) PCT/AU98/00260<br />

(22) 14 Apr/avr 1998 (14.04.1998)<br />

(25) en (26) en<br />

(31) PO 6123 (32) 11 Apr/avr 1997 (33) AU<br />

(11.04.1997)<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 A61K 31/60, 31/605, C07C 67/08, 67/14, 69/353<br />

(54) • NOVEL DIFLUNISAL ESTERS AND RELA-<br />

TED COMPOUNDS<br />

• NOUVEAUX ESTERS DE DIFLUNISAL ET<br />

COMPOSES ASSOCIES<br />

(71) THE UNIVERSITY OF QUEENSLAND<br />

[AU/AU]; St. Lucia, QLD 4072 (AU).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) YUNG–YU HUNG, Daniel [CN/AU]; 116<br />

Arenga Street, Wakerley, QLD 4154 (AU). RO-<br />

BERTS, Michael, Stephen [AU/AU]; 34 Tolaga<br />

Street, Westlake, QLD 4074 (AU).<br />

(74) KELLY, Robin, Thomas; Fisher Adams Kelly,<br />

Level 13, 10 Eagle Street, G.P.O. Box 1413,<br />

Brisbane, QLD 4000 (AU).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/46235 (13) A1<br />

(21) PCT/EP98/01926<br />

(22) 2 Apr/avr 1998 (02.04.1998)<br />

(25) de (26) de<br />

(31) 197 15 594.4 (32) 15 Apr/avr 1997 (33) DE<br />

(15.04.1997)<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 A61K 31/60, 31/19<br />

(54) • ANALGESIC COMBINATION<br />

• ASSOCIATION D’ANALGESIQUES<br />

(71) BAYER AKTIENGESELLSCHAFT [DE/DE];<br />

D–51368 Leverkusen (DE).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) NEUSER, Dieter [DE/DE]; Kirschbaum 39,<br />

D–40764 Langenfeld (DE). FIERUS, Monika<br />

[DE/DE]; Am Gierlichshof 10, D–51381 Leverkusen<br />

(DE). WIEHL, Wolfgang [DE/DE];<br />

Rembrandtstrasse 11, D–50999 Köln (DE).<br />

(74) BAYER AKTIENGESELLSCHAFT; D–51368<br />

Leverkusen (DE).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/46236<br />

(21) PCT/US98/06285<br />

(13) A1<br />

(22) 31 Mar/mar 1998 (31.03.1998)<br />

(25) en (26) en<br />

(31) 08/843,042 (32) 11 Apr/avr 1997<br />

(11.04.1997)<br />

(33) US<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 A61K 31/675<br />

(54) • METHOD OF INHIBITING BONE RESORP-<br />

TION<br />

• PROCEDE EMPECHANT LA RESORBPTION<br />

OSSEUSE<br />

(71) COLGATE–PALMOLIVE<br />

[US/US]; 300 Park Avenue,<br />

10022 (US).<br />

COMPANY<br />

New York, NY<br />

(72) GAFFAR, Abdul; 89 Carter Road, Princeton, NJ<br />

08902 (US).<br />

(74) GOLDFINE, Henry, S.; Colgate–Palmolive Company,<br />

909 River Road, Piscataway, NJ 08855–1343<br />

(US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG UZ VN YU ZW; AP (GH GM KE LS<br />

MW SD SZ UG ZW); EA (AM AZ BY KG KZ<br />

MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />

FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />

CF CG CI CM GA GN ML MR NE SN TD TG).<br />

(11) WO 98/46237 (13) A1<br />

(21) PCT/US98/07517

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