section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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42/1998<br />
14720 PCT Gazette - Section I - Gazette du PCT 22 Oct/oct 1998<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07B 61/00, B01J 19/00<br />
(54) • METHOD FOR THE PREPARATION OF A<br />
CHEMICAL LIBRARY<br />
• PROCEDE DE PREPARATION D’UNE<br />
BANQUE CHIMIQUE<br />
(71) ZENECA LIMITED [GB/GB]; 15 Stanhope Gate,<br />
London W1Y 6LN (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) CORLESS, Anthony, Robert [GB/GB]; CRL,<br />
Dawley Road, Hayes, Middlesex UB3 1HH (GB).<br />
WENN, David, Andrew [GB/GB]; CRL, Dawley<br />
Road, Hayes, Middlesex UB3 1HH (GB). SHUTE,<br />
Richard, Eden [GB/GB]; Zeneca Pharmaceuticals,<br />
Alderley Park, Macclesfield, Cheshire SK10 4TG<br />
(GB).<br />
(74) PHILLIPS, Neil, Godfrey, Alasdair; Zeneca<br />
Pharmaceuticals, <strong>Intellectual</strong> <strong>Property</strong> Dept.,<br />
Mereside, Alderley Park, Macclesfield, Cheshire<br />
SK10 4TG (GB).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46550 (13) A1<br />
(21) PCT/GB98/01077<br />
(22) 14 Apr/avr 1998 (14.04.1998)<br />
(25) en (26) en<br />
(31) 9707742.4 (32) 17 Apr/avr 1997 (33) GB<br />
(17.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07B 61/00, B01J 19/00<br />
(54) • METHOD FOR THE PREPARATION OF A<br />
CODED CHEMICAL LIBRARY<br />
• PROCEDE DE PREPARATION D’UNE<br />
BANQUE CHIMIQUE CODEE<br />
(71) ZENECA LIMITED [GB/GB]; 15 Stanhope Gate,<br />
London W1Y 6LN (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) CORLESS, Anthony, Robert [GB/GB]; CRL,<br />
Dawley Road, Hayes, Middlesex UB3 1HH (GB).<br />
WENN, David, Andrew [GB/GB]; CRL, Dawley<br />
Road, Hayes, Middlesex UB3 1HH (GB). GAR-<br />
MAN, Andrew, John [GB/GB]; Zeneca Pharmaceuticals,<br />
Alderley Park, Macclesfield, Cheshire<br />
SK10 4TG (GB).<br />
(74) PHILLIPS, Neil, Godfrey, Alasdair; Zeneca<br />
Pharmaceuticals, <strong>Intellectual</strong> <strong>Property</strong> Dept.,<br />
Mereside, Alderley Park, Macclesfield, Cheshire<br />
SK10 4TG (GB).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46551 (13) A1<br />
(21) PCT/US98/07870<br />
(22) 16 Apr/avr 1998 (16.04.1998)<br />
(25) en (26) en<br />
(31) 08/843,584 (32) 16 Apr/avr 1997 (33) US<br />
(16.04.1997)<br />
(31) 09/009,846 (32) 20 Jan/jan 1998 (33) US<br />
(20.01.1998)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07B 61/00 // C07D 263/42, 333/58<br />
(54) • SYNTHESIS AND USE OF BIASED ARRAYS<br />
• SYNTHESE ET UTILISATION DE SERIES<br />
BIAISEES<br />
(71) ARQULE, INC. [US/US]; Suite 1000, 200 Boston<br />
Avenue, Medford, MA 02155 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) COFFEN, David, L. [US/US]; 8 Berkeley<br />
Place, Cambridge, MA 02138 (US). HOGAN,<br />
Joseph, C., Jr. [US/US]; 50 Oak Avenue, Belmont,<br />
MA 02178 (US).<br />
(74) FASSE, J., Peter; Fish & Richardson P.C., 225<br />
Franklin Street, Boston, MA 02110–2804 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46552 (13) A1<br />
(21) PCT/US97/06291<br />
(22) 15 Apr/avr 1997 (15.04.1997)<br />
(25) en (26) en<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07C 2/68<br />
(54) • AROMATICS ALKYLATION<br />
• ALKYLATION DE COMPOSES AROMA-<br />
TIQUES<br />
(71) MOBIL OIL CORPORATION [US/US]; 3225<br />
Gallows Road, Fairfax, VA 22037 (US).<br />
(72) MAZZONE, Dominick, Nicholas; 10 North<br />
Monroe Avenue, Wenonah, NJ 08090 (US).<br />
MARLER, David, Owen; 801 Cooper Street<br />
#272B, Deptford, NJ 08096 (US). KEVILLE,<br />
Kathleen, Marie; 860 Fenway Park, Beaumont,<br />
TX 77706 (US). GREEN, Larry, Arthur; 708<br />
Union Road, Mickleton, NJ 08056 (US).<br />
(74) LOO, Blossom, E. et al. / etc.; Mobil Oil<br />
Corporation, 3225 Gallows Road, Fairfax, VA<br />
22037 (US).<br />
(81) AL AU BA BB BG BR CA CN CU CZ EE GE HU<br />
IL IS JP KR LC LK LR LT LV MG MK MN MX<br />
NO NZ PL RO RU SG SI SK TR TT UA UZ VN<br />
YU; AP (GH KE LS MW SD SZ UG); EA (AM<br />
AZ BY KG KZ MD RU TJ TM); EP (AT BE CH<br />
DE DK ES FI FR GB GR IE IT LU MC NL PT<br />
SE); OA (BF BJ CF CG CI CM GA GN ML MR<br />
NE SN TD TG).<br />
(11) WO 98/46553 (13) A1<br />
(21) PCT/US98/07341<br />
(22) 13 Apr/avr 1998 (13.04.1998)<br />
(25) en (26) en<br />
(31) 97 1 03910.0 (32) 14 Apr/avr 1997 (33) CN<br />
(14.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07C 13/00, B01D 3/34, A01N 27/00<br />
(54) • BETA–ELEMENE, METHOD TO PREPARE<br />
THE SAME AND USES THEREOF<br />
• BETA–ELEMENE, SON PROCEDE DE PRE-<br />
PARATION ET SES UTILISATIONS<br />
(63) US 97 1 03910.0 (CIP)<br />
14 Apr/avr 1997 (14.04.1997)<br />
(71) PHARMACEUTICAL R & D INSTITUTE<br />
[CN/CN]; China Academy of Science &<br />
Technology Development, 8/F, Science Hall,<br />
Shenzhen, 518031 (CN). YUAN DA INTER-<br />
NATIONAL GROUP LIMITED [CN/CN];<br />
28/F Section B, Yuan Da Building, 19 Duli<br />
Street, Zhongshan District, Dalian 116001 (CN).<br />
CHINA INNOVATION CENTER FOR LIFE<br />
SCIENCES [US/US]; State Science & Technology<br />
Commission of China, 1 <strong>World</strong> Trade Center 7803,<br />
New York, NY 10048 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) CHEN, Yuren [CN/CN]; 153–5 Shanping<br />
Street, Zhongshan District, Dalian 116015 (CN).<br />
WU, Xiu, Ying [CN/CN]; 30 West Binhai Road,<br />
Xigang District, Dalian 116013 (CN).<br />
(74) ELKINS, Mark; 1 <strong>World</strong> Trade Center 7803, New<br />
York, NY 10049–7899 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46554 (13) A1<br />
(21) PCT/IL97/00125<br />
(22) 16 Apr/avr 1997 (16.04.1997)<br />
(25) en (26) en<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07C 62/32, 51/48<br />
(54) • A NOVEL PROCESS TO PRODUCE STABI-<br />
LIZED CARNOSIC ACID IN HIGH CONCEN-<br />
TRATION<br />
• NOUVEAU PROCEDE PERMETTANT DE<br />
PRODUIRE DE L’ACIDE CARNOSIQUE<br />
STABILISE A DES CONCENTRATIONS<br />
ELEVEES<br />
(71) LYCORED NATURAL PRODUCTS INDUS-<br />
TRIES LTD. [IL/IL]; Hebron Road, Industrial<br />
Zone, 84102 Beer Sheva (IL).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) BEN–YOSEF, Gil [IL/IL]; Shomron Street<br />
36, 40500 Even Yehuda (IL). GARBAR, Arkady<br />
[IL/IL]; Alonim Street 8, 20942 Yokneam (IL).<br />
(74) COHEN, A., David; P.O. Box 60, 84100 Beer<br />
Sheva (IL).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH HU IL<br />
IS JP KE KG KP KR KZ LC LK LR LS LT LU<br />
LV MD MG MK MN MW MX NO NZ PL PT RO<br />
RU SD SE SG SI SK TJ TM TR TT UA UG US<br />
UZ VN YU; AP (GH KE LS MW SD SZ UG); EA<br />
(AM AZ BY KG KZ MD RU TJ TM); EP (AT BE<br />
CH DE DK ES FI FR GB GR IE IT LU MC NL<br />
PT SE); OA (BF BJ CF CG CI CM GA GN ML<br />
MR NE SN TD TG).