section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
You also want an ePaper? Increase the reach of your titles
YUMPU automatically turns print PDFs into web optimized ePapers that Google loves.
42/1998<br />
14730 PCT Gazette - Section I - Gazette du PCT 22 Oct/oct 1998<br />
(11) WO 98/46607 (13) A1<br />
(21) PCT/US98/05614<br />
(22) 23 Mar/mar 1998 (23.03.1998)<br />
(25) en (26) en<br />
(31) 08/843,322 (32) 14 Apr/avr 1997<br />
(14.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(33) US<br />
(51) 6 C07D 487/04, A01N 43/90 // (C07D 487/04,<br />
249:00, 239:00)<br />
(54) • FUNGICIDAL TRIFLUOROPHENYL–<br />
TRIAZOLOPYRIMIDINES<br />
• TRIFLUOROPHENYL–<br />
TRIAZOLOPYRIMIDINES FONGICIDES<br />
(71) AMERICAN CYANAMID COMPANY [US/US];<br />
Five Giralda Farms, Madison, NJ 07940 (US).<br />
(72) PEES, Klaus–Jürgen; Soonwaldstrasse 9,<br />
D–55129 Mainz (DE). ALBERT, Guido; Volxheimer<br />
Strasse 4, D–55546 Hackenheim (DE).<br />
(74) MAZZARESE, Joseph, M.; American Home Products<br />
Corporation, Patent Law Dept. – 2B2, One<br />
Campus Drive, Parsippany, NJ 07054 (US) et al. /<br />
etc.<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG UZ VN YU ZW; AP (GH GM KE LS<br />
MW SD SZ UG ZW); EA (AM AZ BY KG KZ<br />
MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN ML MR NE SN TD TG).<br />
(11) WO 98/46608 (13) A1<br />
(21) PCT/US98/05615<br />
(22) 23 Mar/mar 1998 (23.03.1998)<br />
(25) en (26) en<br />
(31) 08/843,323 (32) 14 Apr/avr 1997<br />
(14.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(33) US<br />
(51) 6 C07D 487/04, A01N 43/90, C07F 7/08 // (C07D<br />
487/04, 249:00, 239:00)<br />
(54) • FUNGICIDAL<br />
TRIFLUOROMETHYLALKYLAMINO–<br />
TRIAZOLOPYRIMIDINES<br />
• TRIFLUOROMETHYLALKYLAMINO–<br />
TRIAZOLOPYRIMIDINES FONGICIDES<br />
(71) AMERICAN CYANAMID COMPANY [US/US];<br />
Five Giralda Farms, Madison, NJ 07940 (US).<br />
(72) PEES, Klaus–Juergen; Soonwaldstrasse 9,<br />
D–55129 Mainz (DE). KRUMMEL, Guenter;<br />
Raiffeisenstrasse 13, D–55578 Vendersheim (DE).<br />
COTTER, Henry, Van, Tuyl; Eisenacherstrasse<br />
49, D–55218 Ingelheim (DE). REHNIG, Annerose;<br />
Rathenaustrasse 11, D–55218 Ingelheim<br />
(DE). MAY, Leslie; Peter–Bischof–Strasse 2A,<br />
D–55435 Gau–Algesheim (DE). PFRENGLE,<br />
Waldemar; Junkermuehle 1, D–55444 Seibersbach<br />
(DE). ALBERT, Guido; Volxheimer Strasse<br />
4, D–55546 Hackenheim (DE).<br />
(74) MAZZARESE, Joseph, M.; American Home Products<br />
Corporation, Patent Law Dept. – 2B2, One<br />
Campus Drive, Parsippany, NJ 07054 (US) et al. /<br />
etc.<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG UZ VN YU ZW; AP (GH GM KE LS<br />
MW SD SZ UG ZW); EA (AM AZ BY KG KZ<br />
MD RU TJ TM); EP (AT BE CH DE DK ES FI<br />
FR GB GR IE IT LU MC NL PT SE); OA (BF BJ<br />
CF CG CI CM GA GN ML MR NE SN TD TG).<br />
(11) WO 98/46609 (13) A1<br />
(21) PCT/US98/07128<br />
(22) 10 Apr/avr 1998 (10.04.1998)<br />
(25) en (26) en<br />
(31) 08/834,053 (32) 11 Apr/avr 1997<br />
(11.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(33) US<br />
(51) 6 C07D 491/048, A61K 31/435, C07D 495/04,<br />
519/00 // (C07D 491/048, 307:00, 221:00) (C07D<br />
519/00, 495:00, 487:00)<br />
(54) •<br />
•<br />
FUROPYRIDINE, THIENOPYRIDINE,<br />
PYRROLOPYRIDINE AND RELATED PY-<br />
RIMIDINE, PYRIDAZINE AND TRIAZINE<br />
COMPOUNDS USEFUL IN CONTROLLING<br />
CHEMICAL SYNAPTIC TRANSMISSION<br />
FUROPYRIDINE, THIENOPYRIDINE,<br />
PYRROLOPYRIDINE, ET COMPOSES<br />
CORRESPONDANTS DE PYRIMIDINE,<br />
PYRIDAZINE ET TRIAZINE CONVENANT<br />
PARTICULIEREMENT AU CONTROLE DE<br />
LA CHIMIO–TRANSMISSION SYNAPTIQUE<br />
(71) ABBOTT LABORATORIES [US/US]; CHAD<br />
0377/AP6D–2, 100 Abbott Park Road, Abbott<br />
Park, IL 60064–3500 (US).<br />
(72) ELLIOTT, Richard, L.; 17419 Woodland Drive,<br />
Grayslake, IL 60030 (US). RYTHER, Keith, B.;<br />
862 Waterview Drive, Round Lake Park, IL 60073<br />
(US). HOLLADAY, Mark, W.; 1003 Dawes<br />
Street, Libertyville, IL 60048 (US). WASCIAK,<br />
James, T.; 28440 Dorie Lane, Waterford, WI<br />
53185 (US). DAANEN, Jerome, F.; 4137 Nantucket<br />
Place, Racine, WI 53405 (US). LIN, Nan–<br />
Horng; 220 Knightsbridge, Mundelein, IL 60060<br />
(US). DART, Michael, J.; 1026 Priceton Avenue,<br />
Highland Park, IL 60035 (US). HE, Yun;<br />
Apartment 2B, 4208 Birch Drive, Zion, IL 60099<br />
(US). LI, Yihong; 1020 Talbot Lane, Grayslake,<br />
IL 60060 (US).<br />
(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />
CHAD 0377/APGD–2, 100 Abbott Park Road,<br />
Abbott Park, IL 60064–3500 (US).<br />
(81) CA JP MX; EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE).<br />
(11) WO 98/46610 (13) A1<br />
(21) PCT/GB98/01029<br />
(22) 8 Apr/avr 1998 (08.04.1998)<br />
(25) en (26) en<br />
(31) 9707413.2 (32) 11 Apr/avr 1997<br />
(11.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 491/10 // A61K 31/55, (C07D 491/10,<br />
307:00, 223:00)<br />
(54) •<br />
•<br />
(33) GB<br />
PROCESS FOR PREPARING SINGLE ENAN-<br />
TIOMER NARWEDINE<br />
PROCEDE DE PREPARATION DE NARWE-<br />
DINE POSSEDANT UN SEUL ENANTIO-<br />
MERE<br />
(71) CHIROTECH TECHNOLOGY LIMITED<br />
[GB/GB]; Cambridge Science Park, Milton Road,<br />
Cambridge CB4 4WE (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) POTTER, Gerard, Andrew [GB/GB]; De<br />
Montfort University, Dept. of Pharmacy, The Gateway,<br />
Leicester LE7 3BH (GB). TIFFEN, Peter,<br />
David [GB/GB]; Chirotech Technology Limited,<br />
Cambridge Science Park, Milton Road, Cambridge<br />
CB4 4WE (GB).<br />
(74) GILL JENNINGS & EVERY; Broadgate House,<br />
7 Eldon Street, London EC2M 7LH (GB).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46611<br />
(21) PCT/SE98/00642<br />
(13) A1<br />
(22) 7 Apr/avr 1998 (07.04.1998)<br />
(25) en (26) en<br />
(31) 9701396–5 (32) 15 Apr/avr 1997<br />
(15.04.1997)<br />
(33) SE<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 498/10, 495/20, A61K 31/445, 31/535<br />
(54) • COMPOUNDS<br />
• COMPOSES<br />
(71) ASTRA PHARMACEUTICALS LTD. [GB/GB];<br />
Home Park, Kings Langley, Herts WD4 8DH (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(71) ASTRA AKTIEBOLAG [SE/SE]; S–151 85<br />
Södertälje (SE).<br />
(only for / seulement pour MG)<br />
(72, 75) HAMLEY, Peter [GB/GB]; 25 Fowke Street,<br />
Rothley, Leics. LE7 7PJ (GB). McINALLY, Thomas<br />
[GB/GB]; 271 Beacon Road, Loughborough,<br />
Leics. LE11 2RA (GB). TINKER, Alan [GB/GB];<br />
97 Knighttorpe Road, Loughborough, Leics. LE11<br />
5JR (GB).<br />
(74) ASTRA AKTIEBOLAG; Patent Dept., S–151 85<br />
Södertälje (SE).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46612 (13) A1<br />
(21) PCT/US98/01473<br />
(22) 27 Jan/jan 1998 (27.01.1998)<br />
(25) en (26) en<br />
(31) 08/833,745 (32) 11 Apr/avr 1997<br />
(11.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07F 9/09, 9/117<br />
(33) US