section 1 - World Intellectual Property Organization

42/1998
22 Oct/oct 1998 PCT Gazette - Section I - Gazette du PCT 14727
(31) 9/100675 (32) 17 Apr/avr 1997 (33) JP
(17.04.1997)
(31) 10/41495 (32) 24 Feb/fév 1998 (33) JP
(24.02.1998)
(43) 22 Oct/oct 1998 (22.10.1998)
(51) 6 C07D 401/06, A61K 31/55, C07D 413/06,
413/14, 401/14, A61K 31/44, 31/40, C07D
417/14, 405/14, 409/14
(54) • THERMOGENIC COMPOSITION AND BEN-
ZAZEPINE THERMOGENICS
• COMPOSITION THERMOGENIQUE ET
COMPOSES THERMOGENIQUES A BASE
DE BENZAZEPINE
(71) TAKEDA CHEMICAL INDUSTRIES, LTD.
[JP/JP]; 1–1, Doshomachi 4–chome, Chuo–ku,
Osaka–shi, Osaka 541–0045 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) ISHIHARA, Yuji [JP/JP]; 3–8, Yamada
3–chome, Itami–shi, Hyogo 664–0874 (JP).
FUJISAWA, Yukio [JP/JP]; 1–31–104, Mikagenakamachi
4–chome, Higashinada–ku, Kobe–shi,
Hyogo 658–0054 (JP). FURUYAMA, Naoki
[JP/JP]; 6–2, Shinoharadai, Nada–ku, Kobe–shi,
Hyogo 657–0016 (JP).
(74) ASAHINA, Tadao et al. / etc.; Osaka Plant of
Takeda Chemical Industries, Ltd., 17–85, Jusohonmachi
2–chome, Yodogawa–ku, Osaka–shi, Osaka
532–0024 (JP).
(81) AL AM AU AZ BA BB BG BR BY CA CN CU
CZ EE GE GW HU ID IL IS KG KR KZ LC LK
LR LT LV MD MG MK MN MX NO NZ PL RO
RU SG SI SK SL TJ TM TR TT UA US UZ VN
YU; AP (GH GM KE LS MW SD SZ UG ZW);
EA (AM AZ BY KG KZ MD RU TJ TM); EP (AT
BE CH CY DE DK ES FI FR GB GR IE IT LU
MC NL PT SE); OA (BF BJ CF CG CI CM GA
GN ML MR NE SN TD TG).
Published / Publiée : (c)
(11) WO 98/46591 (13) A1
(21) PCT/US98/07158
(22) 13 Apr/avr 1998 (13.04.1998)
(25) en (26) en
(31) 60/069,884 (32) 14 Apr/avr 1997 (33) US
(14.04.1997)
(43) 22 Oct/oct 1998 (22.10.1998)
(51) 6 C07D 401/06, 241/08, 295/20, 417/12, A61K
31/495
(54) • SELECTIVE FACTOR Xa INHIBITORS
• INHIBITEURS SELECTIFS DU FACTEUR Xa
(71) COR THERAPEUTICS, INC. [US/US]; 256 E.
Grand Avenue, South San Francisco, CA 94080
(US).
(72) MARLOWE, Charles, K.; 3691 Brandy
Rock Way, Redwood City, CA 94061 (US).
SCARBOROUGH, Robert, M.; 2544 Belmont
Canyon Road, Belmont, CA 94002 (US). ZHU,
Bing–Yan; Apartment K302, 1125 Balclutha
Drive, Foster City, CA 94404 (US).
(74) ADLER, Reid, G. et al. / etc.; Morgan, Lewis &
Bockius LLP, 1800 M Street, N.W., Washington,
DC 20036 (US).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM
GW HU ID IL IS JP KE KG KP KR KZ LC LK
LR LS LT LU LV MD MG MK MN MW MX NO
NZ PL PT RO RU SD SE SG SI SK SL TJ TM
TR TT UA UG UZ VN YU ZW; AP (GH GM KE
LS MW SD SZ UG ZW); EA (AM AZ BY KG
KZ MD RU TJ TM); EP (AT BE CH CY DE DK
ES FI FR GB GR IE IT LU MC NL PT SE); OA
(BF BJ CF CG CI CM GA GN ML MR NE SN
TD TG).
(11) WO 98/46592 (13) A1
(21) PCT/EP98/01847
(22) 30 Mar/mar 1998 (30.03.1998)
(25) de (26) de
(31) 197 15 017.9 (32) 11 Apr/avr 1997
(11.04.1997)
(33) DE
(43) 22 Oct/oct 1998 (22.10.1998)
(51) 6 C07D 401/12, 403/12, 405/12, 413/12, 417/12,
A01N 43/54
(54) • SUBSTITUTED ARYLURACILS
• ARYLURACILES SUBSTITUES
(71) BAYER AKTIENGESELLSCHAFT [DE/DE];
D–51368 Leverkusen (DE).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) ANDREE, Roland [DE/DE]; Dechant–Miebach–Weg
37, D–40764 Langenfeld
(DE). DOLLINGER, Markus [DE/DE]; Burscheider
Strasse 154b, D–51381 Leverkusen
(DE). ERDELEN, Christoph [DE/DE]; Unterbüscherhof
15, D–42799 Leichlingen (DE).
(74) BAYER AKTIENGESELLSCHAFT; D–51368
Leverkusen (DE).
(81) AL AM AT AU AZ BA BB BG BR BY CA CH
CN CU CZ DE DK EE ES FI GB GE GH GM GW
HU ID IL IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MD MG MK MN MW MX NO NZ
PL PT RO RU SD SE SG SI SK SL TJ TM TR TT
UA UG US UZ VN YU ZW; AP (GH GM KE LS
MW SD SZ UG ZW); EA (AM AZ BY KG KZ
MD RU TJ TM); EP (AT BE CH DE DK ES FI
FR GB GR IE IT LU MC NL PT SE); OA (BF BJ
CF CG CI CM GA GN ML MR NE SN TD TG).
(11) WO 98/46593 (13) A1
(21) PCT/JP98/01726
(22) 15 Apr/avr 1998 (15.04.1998)
(25) en (26) en
(31) 9/98694 (32) 16 Apr/avr 1997
(16.04.1997)
(33) JP
(43) 22 Oct/oct 1998 (22.10.1998)
(51) 6 C07D 401/12, C07H 15/18, A61K 31/47, 31/70
(54) • NOVEL CARBOSTYRIL DERIVATIVE
• NOUVEAU PROCEDE DE CARBOSTYRILE
(71) OTSUKA PHARMACEUTICAL CO., LTD.
[JP/JP]; 2–9, Kanda–Tsukasacho, Chiyoda–ku,
Tokyo 101–0048 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) OHTANI, Tadaaki [JP/JP]; Shandofururu
C–211, 80–2, Aza Inamoto, Nakakirai, Matsushigecho,
Itano–gun, Tokushima 771–0212 (JP).
OTSUBO, Kenji [JP/JP]; Birudo.Nosaido 201, 45,
Kitayasocho 4–chome, Tokushima–shi, Tokushima
770–0006 (JP). MATSUBARA, Jun [JP/JP];
Zeneraru Nezu, 1–1–21, Nezu, Bunkyo–ku, Tokyo
113–0031 (JP). KITANO, Kazuyoshi [JP/JP];
1–53, Aza Nishiyamada, Hinoki, Oasacho, Naruto–shi,
Tokushima 779–0225 (JP). MORITA,
Seiji [JP/JP]; 1076–44, Kagasuno, Kawauchicho,
Tokushima–shi, Tokushima 771–0130 (JP).
KAWANO, Yoshikazu [JP/JP]; 463–30, Kagasuno,
Kawauchicho, Tokushima–shi, Tokushima
771–0130 (JP). UCHIDA, Minoru [JP/JP]; 11,
Aza Honson, Ohayashicho, Komatsushima–shi,
Tokushima 773–0022 (JP). YAMASHITA, Shuji
[JP/JP]; 5–39, Aza Ekokawa, Shinkirai, Kitajimacho,
Itano–gun, Tokushima 771–0207 (JP).
(74) ASAMURA, Kiyoshi et al. / etc.; New Ohtemachi
Building, Room 331, 2–1, Ohtemachi 2–chome,
Chiyoda–ku, Tokyo 100–0004 (JP).
(81) AU BR CA CN ID KR MX SG US; EP (AT BE
CH CY DE DK ES FI FR GB GR IE IT LU MC
NL PT SE).
(11) WO 98/46594 (13) A1
(21) PCT/JP98/01664
(22) 10 Apr/avr 1998 (10.04.1998)
(25) ja (26) ja
(31) 9/108299 (32) 11 Apr/avr 1997 (33) JP
(11.04.1997)
(43) 22 Oct/oct 1998 (22.10.1998)
(51) 6 C07D 403/04, 413/04, 417/04, A61K 31/415,
31/42, 31/425
(54) • PYRAZOLE DERIVATIVES AND COX INHI-
BITORS CONTAINING THEM
• DERIVES DE PYRAZOLE ET INHIBITEURS
DE COX LES RENFERMANT
(71) GRELAN PHARMACEUTICAL CO., LTD.
[JP/JP]; 3–9, Nozawa 3–chome, Setagaya–ku,
Tokyo 154–0003 (JP).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) AOTSUKA, Tomoji [JP/JP]; Grelan Research
Center, 4–3, Sakaecho 3–chome, Hamura–shi,
Tokyo 205–0002 (JP). WAGATSUMA, Nagatoshi
[JP/JP]; Grelan Research Center, 4–3, Sakaecho
3–chome, Hamura–shi, Tokyo 205–0002 (JP).
KATO, Hideo [JP/JP]; 26–1–302, Higashiyama
143, Kusamacho, Toyohashi–shi, Aichi 441–8141
(JP). ASHIZAWA, Naoki [JP/JP]; Grelan Research
Center, 4–3, Sakaecho 3–chome, Hamura–shi, Tokyo
205–0002 (JP).
(74) MIZUNO, Akinobu; Gloria Miyamasuzaka III
305, 10–7, Shibuya 1–chome, Shibuya–ku, Tokyo
150–0002 (JP).
(81) JP US; EP (AT BE CH CY DE DK ES FI FR GB
GR IE IT LU MC NL PT SE).
(11) WO 98/46595
(21) PCT/IB98/00540
(13) A1
(22) 9 Apr/avr 1998 (09.04.1998)
(25) en (26) en
(31) 60/042,316 (32) 15 Apr/avr 1997
(15.04.1997)
(33) US
(43) 22 Oct/oct 1998 (22.10.1998)
(51) 6 C07D 403/12, A61K 31/415
(54) • 5–(2–
IMIDAZOLINYLAMINO)BENZIMIDAZOLE
COMPOUNDS USEFUL AS ALPHA–2
ADRENOCEPTOR AGONISTS
• COMPOSES DE 5–(2–
IMIDAZOLINYLAMINO)BENZIMIDAZOLE
UTILES EN TANT QU’AGONISTES DE
L’ADRENORECEPTEUR ALPHA–2
(71) THE PROCTER & GAMBLE COMPANY
[US/US]; One Procter & Gamble Plaza, Cincinnati,
OH 45202 (US).
(for all designated States except / pour tous les États
désignés sauf US)
(72, 75) CUPPS, Thomas, Lee [US/US]; 193 North
Broad Street, Norwich, NY 13815 (US). BOG-
DAN, Sophie, Eva [US/US]; 714 East Foster–Maineville
Road, Maineville, OH 45039
(US). MIELING, Glen, Edward [US/US]; 7395
Desert Spring Court, West Chester, OH 45069
(US). NIKOLAIDES, Nick [US/US]; 5357
Prescott Court, Mason, OH 45040 (US). HENRY,
Raymond, Todd [US/US]; 877 Hechterman Road,
Pleasant Plain, OH 45162 (US). SHELDON,
Russell, James [US/US]; 5023 Winton Road,
Fairfield, OH 45014 (US).