section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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42/1998<br />
14734 PCT Gazette - Section I - Gazette du PCT 22 Oct/oct 1998<br />
(71) PEPTIDE THERAPEUTICS LIMITED<br />
[GB/GB]; 321 Cambridge Science Park, Milton<br />
Road, Cambridge CB4 4WG (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) HART, Terance [GB/GB]; 12 Perry Court,<br />
Clerk Maxwell Road, Cambridge CB3 0RS (GB).<br />
QUIBELL, Martin [GB/GB]; 23 Fennec Close,<br />
Cherry Hinton, Cambridge CB1 4GG (GB).<br />
(74) DAVIES, Jonathan, Mark; Reddie & Grose, 16<br />
Theobalds Road, London WC1X 8PL (GB).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46631 (13) A1<br />
(21) PCT/US98/07135<br />
(22) 8 Apr/avr 1998 (08.04.1998)<br />
(25) en (26) en<br />
(31) 60/043,532 (32) 11 Apr/avr 1997 (33) US<br />
(11.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07K 5/12, 7/50, G01N 33/53, 33/566, C12Q<br />
1/00<br />
(54) • COMBINATORIAL LIBRARIES OF PEP-<br />
TIDOMIMETIC MACROCYCLES AND<br />
PROCESSES THEREFOR<br />
• ECHANTILLOTHEQUES COMBINATOIRES<br />
DE MACROCYCLES PEPTIDOMIMETIQUES<br />
ET PROCEDES CORRESPONDANTS<br />
(71) ELI LILLY AND COMPANY [US/US]; Lilly<br />
Corporate Center, Indianapolis, IN 46285 (US).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) MENDEL, David [US/US]; 11348 Woods Bay<br />
Lane, Indianapolis, IN 46236 (US).<br />
(74) COLLINS, Daniel, W. et al. / etc.; Eli Lilly and<br />
company, Lilly Corporate Center, Indianapolis, IN<br />
46285 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46632<br />
(21) PCT/EP98/02179<br />
(13) A2<br />
(22) 14 Apr/avr 1998 (14.04.1998)<br />
(25) de (26) de<br />
(31) 97 106 024.9<br />
(34) DE et al. / etc.<br />
(32) 11 Apr/avr 1997<br />
(11.04.1997)<br />
(33) EP<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07K 7/00<br />
(54) • INHIBITORS FOR UROKINASE RECEPTOR<br />
•<br />
INHIBITEURS POUR LE RECEPTEUR DE<br />
L’UROKINASE<br />
(71) WILEX BIOTECHNOLOGY GMBH [DE/DE];<br />
Grillparzer Strasse 10 B, D–81675 München (DE).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) KESSLER, Horst [DE/DE]; Friedrich–Stolze–Strasse<br />
53, D–65824 Schwalbach–Limes<br />
(DE). GRAEFF, Heinrich [DE/DE];<br />
Josef–Schwarz–Weg 11, D–81479 München (DE).<br />
SCHMITT, Manfred [DE/DE]; Hohenaschauer<br />
Strasse 10, D–81669 München (DE). MAGDO-<br />
LEN, Viktor [US/DE]; Moosachweg 3, D–85551<br />
Kirchheim (DE). WILHELM, Olaf, G. [DE/DE];<br />
Säbener Strasse 188, D–81545 München (DE).<br />
RIEMER, Christoph [DE/DE]; Prinzregentenstrasse<br />
139, D–81677 München (DE). BÜRGLE,<br />
Markus [DE/DE]; Ötschmannweg 10, D–81369<br />
München (DE).<br />
(74) WEICKMANN, H. et al. / etc.; Kopernikusstrasse<br />
9, D–81679 München (DE).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46633<br />
(21) PCT/US98/07231<br />
(13) A1<br />
(22) 10 Apr/avr 1998 (10.04.1998)<br />
(25) en (26) en<br />
(31) 08/838,916 (32) 11 Apr/avr 1997<br />
(11.04.1997)<br />
(33) US<br />
(31) 09/028,083 (32) 23 Feb/fév 1998<br />
(23.02.1998)<br />
(33) US<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07K 7/06, 7/08, A61K 38/08<br />
(54) • CYTOMODULATING LIPOPHILIC PEP-<br />
TIDES FOR MODULATING IMMUNE<br />
SYSTEM ACTIVITY AND INHIBITING IN-<br />
FLAMMATION<br />
• CYTOMODULATION DE PEPTIDES LIPO-<br />
PHILES AUX FINS D’UNE MODULATION<br />
DE L’ACTIVITE DU SYSTEME IMMU-<br />
NITAIRE ET DE LA SUPPRESSION DE<br />
L’INFLAMMATION<br />
(71) SANGSTAT MEDICAL CORPORATION<br />
[US/US]; 1505–B Adams Drive, Menlo Park, CA<br />
94025 (US).<br />
(72) BUELOW, Roland; 2747 Ross Road, Palo Alto,<br />
CA 94303 (US). GRASSY, Gerard; 32, rue du<br />
Pradas, F–34470 Perols (FR). CALAS, Bernard;<br />
360, avenue du Père Prévost, F–34090 Montpellier<br />
(FR).<br />
(74) TRECARTIN, Richard, F. et al. / etc.; Flehr,<br />
Hohbach, Test, Albritton & Herbert LLP, Suite<br />
3400, 4 Embarcadero Center, San Francisco, CA<br />
94111–4187 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46634 (13) A1<br />
(21) PCT/US98/07438<br />
(22) 13 Apr/avr 1998 (13.04.1998)<br />
(25) en (26) en<br />
(31) 08/837,042 (32) 11 Apr/avr 1997 (33) US<br />
(11.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07K 7/23, A61K 38/09<br />
(54) • GnRH ANTAGONISTS BEING MODIFIED IN<br />
POSITIONS 5 AND 6<br />
• ANTAGONISTES DE GnRH MODIFIES AUX<br />
POSITIONS 5 ET 6<br />
(71) FERRING B.V. [NL/NL]; Marsstraat 9, P.O. Box<br />
3129, NL–2130 KC Hoofddorp (NL).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) SEMPLE, Graeme [GB/GB]; 2 Station Road,<br />
Romsey, Hampshire SO51 8DP (GB). JIANG,<br />
Guangcheng [CN/US]; Apartment #39, 8020 Avenida<br />
Navidad, San Diego, CA 92122 (US).<br />
(74) SAMPLES, Kenneth, H. et al. / etc.; Fitch, Even,<br />
Tabin & Flannery, Room 900, 135 S. LaSalle,<br />
Chicago, IL 60603 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG US UZ VN YU ZW; AP (GH GM<br />
KE LS MW SD SZ UG ZW); EP (AT BE CH CY<br />
DE DK ES FI FR GB GR IE IT LU MC NL PT<br />
SE); OA (BF BJ CF CG CI CM GA GN ML MR<br />
NE SN TD TG).<br />
(11) WO 98/46635 (13) A1<br />
(21) PCT/US98/07519<br />
(22) 13 Apr/avr 1998 (13.04.1998)<br />
(25) en (26) en<br />
(31) 08/837,041 (32) 11 Apr/avr 1997 (33) US<br />
(11.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07K 7/23, A61K 38/09, G01N 33/74<br />
(54) • GnRH ANTAGONISTS<br />
• ANTAGONISTES DE GnRH<br />
(71) FERRING BV [NL/NL]; Marsstraat 9, P.O. Box<br />
3129, NL–2130 KC Hoofddorp (NL).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) JIANG, Guangcheng [CN/US]; Apartment<br />
#39, 8020 Avenida Navidad, San Diego, CA 92122<br />
(US). SEMPLE, Graeme [GB/GB]; 2 Station<br />
Road, Romsey, Hampshire SO51 8DP (GB).<br />
(74) SAMPLES, Kenneth, H. et al. / etc.; Fitch, Even,<br />
Tabin & Flannery, Room 900, 135 S. LaSalle,<br />
Chicago, IL 60603 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG US UZ VN YU ZW; AP (GH GM<br />
KE LS MW SD SZ UG ZW); EP (AT BE CH CY<br />
DE DK ES FI FR GB GR IE IT LU MC NL PT<br />
SE); OA (BF BJ CF CG CI CM GA GN ML MR<br />
NE SN TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46636 (13) A2<br />
(21) PCT/US98/07462