section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
section 1 - World Intellectual Property Organization
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42/1998<br />
22 Oct/oct 1998 PCT Gazette - Section I - Gazette du PCT 14729<br />
(74) PALMBERG, Arleen et al. / etc.; Eli Lilly and<br />
Company, Lilly Corporate Center, Indianapolis, IN<br />
46285 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46602 (13) A1<br />
(21) PCT/CA98/00360<br />
(22) 15 Apr/avr 1998 (15.04.1998)<br />
(25) en (26) en<br />
(31) 08/840,559 (32) 15 Apr/avr 1997<br />
(15.04.1997)<br />
(31) 60/076,426 (32) 24 Feb/fév 1998<br />
(24.02.1998)<br />
(33) US<br />
(33) US<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 471/04, A61K 31/435<br />
(54) • ALKALOID HALIDE SALTS OF SWAINSO-<br />
NINE AND METHODS OF USE<br />
• SELS HALOGENES D’ALCALOIDE<br />
DE SWAINSONINE ET PROCEDES<br />
D’UTILISATION<br />
(71) GLYCODESIGN INC. [CA/CA]; Suite 900, 480<br />
University Avenue, Toronto, Ontario M5G 1V2<br />
(CA).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(72, 75) DENNIS, James, W. [CA/CA]; 17 Maple<br />
Dawn Road, Etobicoke, Ontario M9C 2V7 (CA).<br />
SHAH, Rajan, N. [CA/CA]; 57 Charles Street<br />
West #1109, Toronto, Ontario M5S 2X1 (CA).<br />
ZISER, Lothar [DE/CA]; 20 Carlton Street #1434,<br />
Toronto, Ontario M5B 2H5 (CA).<br />
(74) BERESKIN & PARR; 40th floor, 40 King Street<br />
West, Toronto, Ontario M5H 3Y2 (CA).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46603 (13) A1<br />
(21) PCT/US98/04127<br />
(22) 16 Apr/avr 1998 (16.04.1998)<br />
(25) en (26) en<br />
(31) 08/834,393 (32) 16 Apr/avr 1997<br />
(16.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 471/04, A61K 31/505<br />
(33) US<br />
(54) • 6,7–DISUBSTITUTED–4–<br />
AMINOPYRIDO[2,3–D]PYRIMIDINE<br />
COMPOUNDS<br />
• COMPOSES DE 4–AMINOPYRIDO[2,3–<br />
D]PYRIMIDINE DISUBSTITUEE EN POSI-<br />
TION 6, 7<br />
(71) ABBOTT LABORATORIES [US/US]; CHAD<br />
0377/AP6D, 100 Abbott Park Road, Abbott Park,<br />
IL 60064–3500 (US).<br />
(72) BHAGWAT, Shripad, S.; 30055 N. Waukegan<br />
Road, Lake Bluff, IL 60044 (US). LEE, Chih–<br />
Hung; 966 Dunhill Road, Grayslake, IL 60030<br />
(US). PERNER, Richard, J.; 1655 Pinetree<br />
Drive, Gurnee, IL 60031 (US). GU, Yu–Gui; 312<br />
Cambridge Drive, Grayslake, IL 60030 (US).<br />
(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />
D377/AP6D, 100 Abbott Park Road, Abbott Park,<br />
IL 60064–3500 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46604<br />
(21) PCT/US98/07201<br />
(13) A1<br />
(22) 13 Apr/avr 1998 (13.04.1998)<br />
(25) en (26) en<br />
(31) 08/843,484 (32) 16 Apr/avr 1997<br />
(16.04.1997)<br />
(33) US<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 471/04, A61K 31/505<br />
(54) • 5,6,7–TRISUBSTITUTED–4–<br />
AMINOPYRIDOL[2,3–D]PYRIMIDINE<br />
COMPOUNDS<br />
• COMPOSES DE 4–AMINOPYRIDOL[2,3–<br />
D]PYRIMIDINE A TRISUBSTITUTION 5,6,7<br />
(71) ABBOTT LABORATORIES [US/US];<br />
CHAD–0377/AP6D–2, 100 Abbott Park Road,<br />
Abbott Park, IL 60064–3500 (US).<br />
(72) BHAGWAT, Shripad, S.; 1310 Kristin Drive,<br />
Libertyville, IL 60048 (US). PERNER, Richard,<br />
J.; 704 Penny Lake, Gurnee, IL 60031 (US). GU,<br />
Yu, Gui; 312 Cambridge Drive, Grayslake, IL<br />
60030 (US).<br />
(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />
CHAD 0377/AP6D–2, 100 Abbott Park Road,<br />
Abbott Park, IL 60064–3500 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
Published / Publiée : (c)<br />
(11) WO 98/46605 (13) A1<br />
(21) PCT/US98/07207<br />
(22) 14 Apr/avr 1998 (14.04.1998)<br />
(25) en (26) en<br />
(31) 08/838,216 (32) 16 Apr/avr 1997<br />
(16.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 471/04, A61K 31/495<br />
(33) US<br />
(54) • 5,7–DISUBSTITUTED 4–<br />
AMINOPYRIDO[2,3–D]PYRIMIDINE<br />
COMPOUNDS AND THEIR USE AS<br />
ADENOSINE KINASE INHIBITORS<br />
• COMPOSES DE 4–AMINOPYRIDO[2,3–<br />
D]PYRIMIDINE 5,7–DISUBSTITUES ET<br />
LEUR UTILISATION COMME INHIBITEURS<br />
DE L’ADENOSINE KINASE<br />
(71) ABBOTT LABORATORIES [US/US]; CHAD<br />
0377/AP6D–2, 100 Abbott Park Road, Abbott<br />
Park, IL 60064–3500 (US).<br />
(72) BHAGWAT, Shripad, S.; 30055 N. Waukegan<br />
Road, Lake Bluff, IL 60044 (US). LEE, Chih–<br />
Hung; 966 Dunhill Road, Grayslake, IL 60030<br />
(US). COWART, Marlon, D.; 43 E. Dahlia Lane,<br />
Round Lake Beach, IL 60073 (US). MCKIE,<br />
Jeffrey; Apartment 211, 716 Water’s Edge Drive,<br />
Lake Villa, IL 60046 (US). GRILLOT, Anne,<br />
Laure; Apartment 2, 99 Hammond Street, Cambridge,<br />
MA 02138 (US).<br />
(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />
CHAD 0377/AP6D–2, 100 Abbott Park Road,<br />
Abbott Park, IL 60064–3500 (US).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM<br />
GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />
LR LS LT LU LV MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />
TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).<br />
(11) WO 98/46606 (13) A1<br />
(21) PCT/SE98/00640<br />
(22) 7 Apr/avr 1998 (07.04.1998)<br />
(25) en (26) en<br />
(31) 9701398–1 (32) 15 Apr/avr 1997 (33) SE<br />
(15.04.1997)<br />
(43) 22 Oct/oct 1998 (22.10.1998)<br />
(51) 6 C07D 487/04, A61K 31/505, 31/415 // (C07D<br />
487/04, 239:00, 231:00)<br />
(54) • NOVEL COMPOUNDS<br />
• NOUVEAUX COMPOSES<br />
(71) ASTRA PHARMACEUTICALS LTD. [GB/GB];<br />
Home Park, Kings Langley, Herts WD4 8DH (GB).<br />
(for all designated States except / pour tous les États<br />
désignés sauf US)<br />
(71) ASTRA AKTIEBOLAG [SE/SE]; S–151 85<br />
Södertälje (SE).<br />
(only for / seulement pour MG)<br />
(72, 75) CHESHIRE, David [GB/GB]; Astra Charnwood,<br />
Bakewell Road, Loughborough, Leics.<br />
LE11 5RH (GB). COOPER, Martin [GB/GB];<br />
Astra Charnwood, Bakewell Road, Loughborough,<br />
Leics. LE11 5RH (GB). DONALD, David<br />
[GB/GB]; Astra Charnwood, Bakewell<br />
Road, Loughborough, Leics. LE11 5RH (GB).<br />
THORNE, Philip [GB/GB]; Astra Charnwood,<br />
Bakewell Road, Loughborough, Leics. LE11 5RH<br />
(GB).<br />
(74) ASTRA AKTIEBOLAG; Patent Dept., S–151 85<br />
Södertälje (SE).<br />
(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />
CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />
HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MD MG MK MN MW MX NO NZ<br />
PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />
TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />
LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />
ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />
(BF BJ CF CG CI CM GA GN ML MR NE SN<br />
TD TG).