24.12.2012 Views

section 1 - World Intellectual Property Organization

section 1 - World Intellectual Property Organization

section 1 - World Intellectual Property Organization

SHOW MORE
SHOW LESS

You also want an ePaper? Increase the reach of your titles

YUMPU automatically turns print PDFs into web optimized ePapers that Google loves.

42/1998<br />

22 Oct/oct 1998 PCT Gazette - Section I - Gazette du PCT 14729<br />

(74) PALMBERG, Arleen et al. / etc.; Eli Lilly and<br />

Company, Lilly Corporate Center, Indianapolis, IN<br />

46285 (US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/46602 (13) A1<br />

(21) PCT/CA98/00360<br />

(22) 15 Apr/avr 1998 (15.04.1998)<br />

(25) en (26) en<br />

(31) 08/840,559 (32) 15 Apr/avr 1997<br />

(15.04.1997)<br />

(31) 60/076,426 (32) 24 Feb/fév 1998<br />

(24.02.1998)<br />

(33) US<br />

(33) US<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 C07D 471/04, A61K 31/435<br />

(54) • ALKALOID HALIDE SALTS OF SWAINSO-<br />

NINE AND METHODS OF USE<br />

• SELS HALOGENES D’ALCALOIDE<br />

DE SWAINSONINE ET PROCEDES<br />

D’UTILISATION<br />

(71) GLYCODESIGN INC. [CA/CA]; Suite 900, 480<br />

University Avenue, Toronto, Ontario M5G 1V2<br />

(CA).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(72, 75) DENNIS, James, W. [CA/CA]; 17 Maple<br />

Dawn Road, Etobicoke, Ontario M9C 2V7 (CA).<br />

SHAH, Rajan, N. [CA/CA]; 57 Charles Street<br />

West #1109, Toronto, Ontario M5S 2X1 (CA).<br />

ZISER, Lothar [DE/CA]; 20 Carlton Street #1434,<br />

Toronto, Ontario M5B 2H5 (CA).<br />

(74) BERESKIN & PARR; 40th floor, 40 King Street<br />

West, Toronto, Ontario M5H 3Y2 (CA).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/46603 (13) A1<br />

(21) PCT/US98/04127<br />

(22) 16 Apr/avr 1998 (16.04.1998)<br />

(25) en (26) en<br />

(31) 08/834,393 (32) 16 Apr/avr 1997<br />

(16.04.1997)<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 C07D 471/04, A61K 31/505<br />

(33) US<br />

(54) • 6,7–DISUBSTITUTED–4–<br />

AMINOPYRIDO[2,3–D]PYRIMIDINE<br />

COMPOUNDS<br />

• COMPOSES DE 4–AMINOPYRIDO[2,3–<br />

D]PYRIMIDINE DISUBSTITUEE EN POSI-<br />

TION 6, 7<br />

(71) ABBOTT LABORATORIES [US/US]; CHAD<br />

0377/AP6D, 100 Abbott Park Road, Abbott Park,<br />

IL 60064–3500 (US).<br />

(72) BHAGWAT, Shripad, S.; 30055 N. Waukegan<br />

Road, Lake Bluff, IL 60044 (US). LEE, Chih–<br />

Hung; 966 Dunhill Road, Grayslake, IL 60030<br />

(US). PERNER, Richard, J.; 1655 Pinetree<br />

Drive, Gurnee, IL 60031 (US). GU, Yu–Gui; 312<br />

Cambridge Drive, Grayslake, IL 60030 (US).<br />

(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />

D377/AP6D, 100 Abbott Park Road, Abbott Park,<br />

IL 60064–3500 (US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM<br />

GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MD MG MK MN MW MX NO<br />

NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />

TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/46604<br />

(21) PCT/US98/07201<br />

(13) A1<br />

(22) 13 Apr/avr 1998 (13.04.1998)<br />

(25) en (26) en<br />

(31) 08/843,484 (32) 16 Apr/avr 1997<br />

(16.04.1997)<br />

(33) US<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 C07D 471/04, A61K 31/505<br />

(54) • 5,6,7–TRISUBSTITUTED–4–<br />

AMINOPYRIDOL[2,3–D]PYRIMIDINE<br />

COMPOUNDS<br />

• COMPOSES DE 4–AMINOPYRIDOL[2,3–<br />

D]PYRIMIDINE A TRISUBSTITUTION 5,6,7<br />

(71) ABBOTT LABORATORIES [US/US];<br />

CHAD–0377/AP6D–2, 100 Abbott Park Road,<br />

Abbott Park, IL 60064–3500 (US).<br />

(72) BHAGWAT, Shripad, S.; 1310 Kristin Drive,<br />

Libertyville, IL 60048 (US). PERNER, Richard,<br />

J.; 704 Penny Lake, Gurnee, IL 60031 (US). GU,<br />

Yu, Gui; 312 Cambridge Drive, Grayslake, IL<br />

60030 (US).<br />

(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />

CHAD 0377/AP6D–2, 100 Abbott Park Road,<br />

Abbott Park, IL 60064–3500 (US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM<br />

GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MD MG MK MN MW MX NO<br />

NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />

TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

Published / Publiée : (c)<br />

(11) WO 98/46605 (13) A1<br />

(21) PCT/US98/07207<br />

(22) 14 Apr/avr 1998 (14.04.1998)<br />

(25) en (26) en<br />

(31) 08/838,216 (32) 16 Apr/avr 1997<br />

(16.04.1997)<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 C07D 471/04, A61K 31/495<br />

(33) US<br />

(54) • 5,7–DISUBSTITUTED 4–<br />

AMINOPYRIDO[2,3–D]PYRIMIDINE<br />

COMPOUNDS AND THEIR USE AS<br />

ADENOSINE KINASE INHIBITORS<br />

• COMPOSES DE 4–AMINOPYRIDO[2,3–<br />

D]PYRIMIDINE 5,7–DISUBSTITUES ET<br />

LEUR UTILISATION COMME INHIBITEURS<br />

DE L’ADENOSINE KINASE<br />

(71) ABBOTT LABORATORIES [US/US]; CHAD<br />

0377/AP6D–2, 100 Abbott Park Road, Abbott<br />

Park, IL 60064–3500 (US).<br />

(72) BHAGWAT, Shripad, S.; 30055 N. Waukegan<br />

Road, Lake Bluff, IL 60044 (US). LEE, Chih–<br />

Hung; 966 Dunhill Road, Grayslake, IL 60030<br />

(US). COWART, Marlon, D.; 43 E. Dahlia Lane,<br />

Round Lake Beach, IL 60073 (US). MCKIE,<br />

Jeffrey; Apartment 211, 716 Water’s Edge Drive,<br />

Lake Villa, IL 60046 (US). GRILLOT, Anne,<br />

Laure; Apartment 2, 99 Hammond Street, Cambridge,<br />

MA 02138 (US).<br />

(74) YANG, Frank, Z. et al. / etc.; Abbott Laboratories,<br />

CHAD 0377/AP6D–2, 100 Abbott Park Road,<br />

Abbott Park, IL 60064–3500 (US).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM<br />

GW HU ID IL IS JP KE KG KP KR KZ LC LK<br />

LR LS LT LU LV MD MG MK MN MW MX NO<br />

NZ PL PT RO RU SD SE SG SI SK SL TJ TM<br />

TR TT UA UG UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).<br />

(11) WO 98/46606 (13) A1<br />

(21) PCT/SE98/00640<br />

(22) 7 Apr/avr 1998 (07.04.1998)<br />

(25) en (26) en<br />

(31) 9701398–1 (32) 15 Apr/avr 1997 (33) SE<br />

(15.04.1997)<br />

(43) 22 Oct/oct 1998 (22.10.1998)<br />

(51) 6 C07D 487/04, A61K 31/505, 31/415 // (C07D<br />

487/04, 239:00, 231:00)<br />

(54) • NOVEL COMPOUNDS<br />

• NOUVEAUX COMPOSES<br />

(71) ASTRA PHARMACEUTICALS LTD. [GB/GB];<br />

Home Park, Kings Langley, Herts WD4 8DH (GB).<br />

(for all designated States except / pour tous les États<br />

désignés sauf US)<br />

(71) ASTRA AKTIEBOLAG [SE/SE]; S–151 85<br />

Södertälje (SE).<br />

(only for / seulement pour MG)<br />

(72, 75) CHESHIRE, David [GB/GB]; Astra Charnwood,<br />

Bakewell Road, Loughborough, Leics.<br />

LE11 5RH (GB). COOPER, Martin [GB/GB];<br />

Astra Charnwood, Bakewell Road, Loughborough,<br />

Leics. LE11 5RH (GB). DONALD, David<br />

[GB/GB]; Astra Charnwood, Bakewell<br />

Road, Loughborough, Leics. LE11 5RH (GB).<br />

THORNE, Philip [GB/GB]; Astra Charnwood,<br />

Bakewell Road, Loughborough, Leics. LE11 5RH<br />

(GB).<br />

(74) ASTRA AKTIEBOLAG; Patent Dept., S–151 85<br />

Södertälje (SE).<br />

(81) AL AM AT AU AZ BA BB BG BR BY CA CH<br />

CN CU CZ DE DK EE ES FI GB GE GH GM GW<br />

HU ID IL IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MD MG MK MN MW MX NO NZ<br />

PL PT RO RU SD SE SG SI SK SL TJ TM TR<br />

TT UA UG US UZ VN YU ZW; AP (GH GM KE<br />

LS MW SD SZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY DE DK<br />

ES FI FR GB GR IE IT LU MC NL PT SE); OA<br />

(BF BJ CF CG CI CM GA GN ML MR NE SN<br />

TD TG).

Hooray! Your file is uploaded and ready to be published.

Saved successfully!

Ooh no, something went wrong!