PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO

42/2000
19 Oct/oct 2000 PCT Gazette - Section I - Gazette du PCT 15237
(51) 7 C07C 405/00, A61K 31/5575, A61P 9/00
(11) WO 00/61550 (13) A1
(21) PCT/JP00/02286
(22) 7 Apr/avr 2000 (07.04.2000)
(25) ja (26) ja
(30) 11/103323 9 Apr/avr 1999
(09.04.1999)
(43) 19 Oct/oct 2000 (19.10.2000)
(54) PROSTAGLANDIN E1 DERIVATIVES
DERIVES DE PROSTAGLANDINE E1
(71) TAISHO PHARMACEUTICAL CO.,
LTD. [JP/JP]; 24–1, Takata 3–chome, Toshima–ku,
Tokyo 170–8633 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(71, 72) SATO, Fumie [JP/JP]; 2–1–901, Kugenumahigashi,
251–0026 (JP).
Fujisawa–shi, Kanagawa
(72, 75) TANAMI, Tohru [JP/JP]; Taisho
Pharmaceutical Co., Ltd., 24–1, Takata
3–chome, Toshima–ku, Tokyo 170–8633
(JP). TANAKA, Hideo [JP/JP]; Taisho
Pharmaceutical Co., Ltd., 24–1, Takata
3–chome, Toshima–ku, Tokyo 170–8633
(JP). ONO, Naoya [JP/JP]; Taisho Pharmaceutical
Co., Ltd., 24–1, Takata 3–chome,
Toshima–ku, Tokyo 170–8633 (JP). YAGI,
Makoto [JP/JP]; Taisho Pharmaceutical Co.,
Ltd., 24–1, Takata 3–chome, Toshima–ku,
Tokyo 170–8633 (JP). HIRANO, Hitomi
[JP/JP]; Taisho Pharmaceutical Co., Ltd.,
24–1, Takata 3–chome, Toshima–ku, Tokyo
170–8633 (JP).
(74) KITAGAWA, Tomizo; Taisho Pharmaceutical
Co., Ltd. Patent Division, 24–1, Takata
3–chome, Toshima–ku, Tokyo 170–8633
(JP).
(81) AU CA CN JP KR US; EP (AT BE CH CY
DE DK ES FI FR GB GR IE IT LU MC NL
PT SE).
(51) 7 C07D
(11) WO 00/61551 (13) A2
(21) PCT/EP00/02746
(22) 29 Mar/mar 2000 (29.03.2000)
(25) de (26) de
(30) 199 16 719.2 13 Apr/avr 1999
(13.04.1999)
(30) 199 62 998.6 24 Dec/déc 1999
(24.12.1999)
JP
DE
DE
(43) 19 Oct/oct 2000 (19.10.2000)
(54) INTEGRIN RECEPTOR LIGANDS
LIGANDS
D’INTEGRINE
DE RECEPTEURS
(71) BASF AKTIENGESELLSCHAFT
[DE/DE]; D–67056 Ludwigshafen (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) ZECHEL, Johann–Christian
[DE/DE]; Schreiberweg 7, D–69226
Nußloch (DE). KLING, Andreas [DE/DE];
Riegeler Weg 14, D–68239 Mannheim
(DE). GENESTE, Hervé [FR/DE]; Rehbachstrasse
42, D–67141 Neuhofen (DE).
LANGE, Udo [DE/DE]; Königsstuhlstrasse
15, D–68163 Mannheim (DE). LAUTER-
BACH, Arnulf [DE/DE]; Innsbrucker Weg
7, D–67067 Ludwigshafen (DE). GRAEF,
Claudia, Isabella [DE/DE]; Tullastrasse 10,
D–68161 Mannheim (DE). SUBKOWSKI,
Thomas [DE/DE]; Wichernstrasse 13,
D–68526 Ladenburg (DE). SADOWSKI,
Jens [DE/DE]; Mainstrasse 2, D–67117
Limburgerhof (DE). HORNBERGER,
Wilfried [DE/DE]; Goldener Winkel 14,
D–67434 Neustadt (DE).
(74) BASF AKTIENGESELLSCHAFT;
D–67056 Ludwigshafen (DE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID
IL IN IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MA MD MG MK MN MW
MX NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ
VN YU ZA ZW; AP (GH GM KE LS MW
SD SL SZ TZ UG ZW); EA (AM AZ BY
KG KZ MD RU TJ TM); EP (AT BE CH
CY DE DK ES FI FR GB GR IE IT LU MC
NL PT SE); OA (BF BJ CF CG CI CM GA
GN GW ML MR NE SN TD TG).
(51) 7 C07D 207/09, 207/20, 295/14, 217/04,
211/26, A61K 31/40, 31/4453, 31/495,
31/5375, 31/445, A61P 37/06, 43/00
(11) WO 00/61552 (13) A1
(21) PCT/JP00/02267
(22) 7 Apr/avr 2000 (07.04.2000)
(25) ja (26) ja
(30) 11/100482 7 Apr/avr 1999
(07.04.1999)
(43) 19 Oct/oct 2000 (19.10.2000)
(54) N–SUBSTITUTED–N’–SUBSTITUTED
UREA DERIVATIVE AND USE THE-
REOF AS TNF– PRODUCTION
INHIBITOR
DERIVE D’UREE N–SUBSTITUE–N’–
SUBSTITUE, ET SON UTILISATION
COMME INHIBITEUR DE LA PRO-
DUCTION DE TNF–
(71) SANTEN PHARMACEUTICAL CO.,
LTD. [JP/JP]; 9–19, Shimoshinjo 3–chome,
Higashiyodogawa–ku, Osaka–shi, Osaka
533–6851 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) MITA, Shiro [JP/JP]; Santen Pharmaceutical
Co., Ltd., 9–19, Shimoshinjo
3–chome, Higashiyodogawa–ku, Osaka–shi,
Osaka 533–6851 (JP). HORIUCHI, Masato
[JP/JP]; Santen Pharmaceutical Co., Ltd.,
9–19, Shimoshinjo 3–chome, Higashiyodogawa–ku,
Osaka–shi, Osaka 533–6851 (JP).
BAN, Masakazu [JP/JP]; Santen Pharmaceutical
Co., Ltd., 9–19, Shimoshinjo
3–chome, Higashiyodogawa–ku, Osaka–shi,
Osaka 533–6851 (JP). SUHARA, Hiroshi
[JP/JP]; Santen Pharmaceutical Co., Ltd.,
9–19, Shimoshinjo 3–chome, Higashiyodogawa–ku,
Osaka–shi, Osaka 533–6851 (JP).
JP
(74) NAKAMURA, Minoru et al. / etc.; Room
646, Shin–Tokyo Bldg, 3–1, Marunouchi
3–chome, Chiyoda–ku, Tokyo 100–8355
(JP).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID
IL IN IS KE KG KP KR KZ LC LK LR LS
LT LU LV MA MD MG MK MN MW MX
NO NZ PL PT RO RU SD SE SG SI SK SL
TJ TM TR TT TZ UA UG US UZ VN YU
ZA ZW; AP (GH GM KE LS MW SD SL
SZ TZ UG ZW); EA (AM AZ BY KG KZ
MD RU TJ TM); EP (AT BE CH CY DE
DK ES FI FR GB GR IE IT LU MC NL PT
SE); OA (BF BJ CF CG CI CM GA GN GW
ML MR NE SN TD TG).
(51) 7 C07D 209/08, 209/30, A61K 31/40
(11) WO 00/61553 (13) A1
(21) PCT/FR00/00921
(22) 11 Apr/avr 2000 (11.04.2000)
(25) fr (26) fr
(30) 99/04576 13 Apr/avr 1999
(13.04.1999)
FR
(43) 19 Oct/oct 2000 (19.10.2000)
(54) 2–AMINOETHYL–INDOLE DERIVA-
TIVES, THEIR PREPARATION AND
THERAPEUTIC USE
DERIVES DE 2–AMINOETHYL–
INDOLE, LEUR PREPARATION ET
LEUR APPLICATION EN THERAPEU-
TIQUE
(71) SANOFI–SYNTHELABO [FR/FR]; 174,
avenue de France, F–75013 Paris (FR).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BOVY, Philippe, R. [BE/FR]; 13, rue
du 4 Septembre, F–78750 Mareil Marly
(FR). MOUGENOT, Patrick [FR/FR]; 2,
avenue Ossart, F–92500 Rueil Malmaison
(FR). PHILIPPO, Christophe [FR/FR]; 18,
place des Maitres Vignerons, F–92500 Rueil
Malmaison (FR).
(74) THOURET–LEMAITRE, Elisabeth;
Sanofi–Synthelabo, 174, avenue de France,
F–75013 Paris (FR).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID
IL IN IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MA MD MG MK MN MW
MX NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ
VN YU ZA ZW; AP (GH GM KE LS MW
SD SL SZ TZ UG ZW); EA (AM AZ BY
KG KZ MD RU TJ TM); EP (AT BE CH
CY DE DK ES FI FR GB GR IE IT LU MC
NL PT SE); OA (BF BJ CF CG CI CM GA
GN GW ML MR NE SN TD TG).
(51) 7 C07D 209/08, A61K 31/40, C07D 209/30,
A61P 43/00
(11) WO 00/61554 (13) A1
(21) PCT/FR00/00922
(22) 11 Apr/avr 2000 (11.04.2000)