PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO

42/2000
19 Oct/oct 2000 PCT Gazette - Section I - Gazette du PCT 15243
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID
IL IN IS JP KE KG KR KZ LC LK LR LS
LT LU LV MA MD MG MK MN MW MX
NO NZ PL PT RO RU SD SE SG SI SK SL
TJ TM TR TT UA UG US UZ VN YU ZA
ZW; AP (GH GM KE LS MW SD SL SZ
TZ UG ZW); EA (AM AZ BY KG KZ MD
RU TJ TM); EP (AT BE CH CY DE DK ES
FI FR GB GR IE IT LU MC NL PT SE);
OA (BF BJ CF CG CI CM GA GN GW ML
MR NE SN TD TG).
(51) 7 C07D 333/38, C07B 43/00
(11) WO 00/61574 (13) A2
(21) PCT/EP00/03018
(22) 5 Apr/avr 2000 (05.04.2000)
(25) de (26) de
(30) 199 15 930.0 9 Apr/avr 1999
(09.04.1999)
(30) 199 33 873.6 23 Jul/juil 1999
(23.07.1999)
(43) 19 Oct/oct 2000 (19.10.2000)
DE
DE
(54) METHOD
DINES
FOR PRODUCING AMI-
PROCEDE
D’AMIDINES
DE PRODUCTION
(71) BASF AKTIENGESELLSCHAFT
[DE/DE]; D–67056 Ludwigshafen (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) ZIERKE, Thomas [DE/DE]; Akazienstr.
12, D–67459 Böhl–Iggelheim (DE).
MACK, Helmut [DE/DE]; Neustadter Ring
80, D–67067 Ludwigshafen (DE).
(74) BASF AKTIENGESELLSCHAFT;
D–67056 Ludwigshafen (DE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID
IL IN IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MA MD MG MK MN MW
MX NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ
VN YU ZA ZW; AP (GH GM KE LS MW
SD SL SZ TZ UG ZW); EA (AM AZ BY
KG KZ MD RU TJ TM); EP (AT BE CH
CY DE DK ES FI FR GB GR IE IT LU MC
NL PT SE); OA (BF BJ CF CG CI CM GA
GN GW ML MR NE SN TD TG).
(51) 7 C07D 401/04, 211/58
(11) WO 00/61575 (13) A1
(21) PCT/JP00/02381
(22) 12 Apr/avr 2000 (12.04.2000)
(25) ja (26) ja
(30) 11/104084 12 Apr/avr 1999
(12.04.1999)
(30) 2000/73283 16 Mar/mar 2000
(16.03.2000)
(43) 19 Oct/oct 2000 (19.10.2000)
JP
JP
(54) PROCESS FOR THE PRODUCTION OF
INDOLE DERIVATIVES AND INTER-
MEDIATES THEREFOR
PRODUCTION DE DERIVES INDOLE
ET INTERMEDIAIRES A CET EFFET
(71) EISAI CO., LTD. [JP/JP]; 6–10, Koishikawa
4–chome, Bunkyo–ku, Tokyo
112–8088 (JP).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) SASHO, Manabu [JP/JP]; 4–22–2–506,
Matsushiro, Tsukuba–shi, Ibaraki 305–0035
(JP). KOMATSU, Yuki [JP/JP]; 4–5–62,
Ninomiya, Tsukuba–shi, Ibaraki 305–0051
(JP). MIYAZAWA, Mamoru [JP/JP];
Villa Shinryu #1–202, 1–3–38, Onohara,
Kamisu–machi, Kashima–gun, Ibaraki
314–0144 (JP). MATSUO, Kimihiro
[JP/JP]; F.Legend #303, 6–17–25, Shittechuo,
Kamisu–machi, Kashima–gun,
Ibaraki 314–0112 (JP). INOUE, Susumu
[JP/JP]; Garden Iris #23, 1–4–22, Onohara,
Kamisu–machi, Kashima–gun, Ibaraki
314–0144 (JP). UENO, Koshi [JP/JP];
668–49, Shimohirooka, Tsukuba–shi, Ibaraki
305–0042 (JP).
(74) FURUYA, Kaoru et al. / etc.; Hamacho–Hanacho
Building, 6th Floor, 2–17–8,
Nihonbashi–Hamacho, Chuo–ku, Tokyo
103–0007 (JP).
(81) US; EP (AT BE CH CY DE DK ES FI FR
GB GR IE IT LU MC NL PT SE).
(51) 7 C07D 401/04, 413/04, 405/14, A61K
31/4178, A61P 19/00
(11) WO 00/61576 (13) A1
(21) PCT/US00/09147
(22) 6 Apr/avr 2000 (06.04.2000)
(25) en (26) en
(30) 60/128,687 9 Apr/avr 1999
(09.04.1999)
(43) 19 Oct/oct 2000 (19.10.2000)
(54) TRIARYLIMIDAZOLES
TRIARYLIMIDAZOLES
US
(71) SMITHKLINE BEECHAM CORPORA-
TION [US/US]; One Franklin Plaza, Philadelphia,
PA 19103 (US).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BURGESS, Joelle, Lorraine [US/US];
1250 South Collegeville Road, Collegeville,
PA 19426–0989 (US). CALLAHAN,
James, Francis [US/US]; 1250 South Collegeville
Road, Collegeville, PA 19426–0989
(US).
(74) STEIN–FERNANDEZ, Nora et al. / etc.;
SmithKline Beecham Corporation, Corporate
Intellectual Property, UW2220, 709 Swedeland
Road, P.O. Box 1539, King of Prussia,
PA 19406–0939 (US).
(81) AE AL AU BA BB BG BR CA CN CZ DZ
EE GE GH GM HR HU ID IL IN IS JP KP
KR LC LK LR LT LV MA MG MK MN MX
NO NZ PL RO SG SI SK SL TR TT TZ UA
US UZ VN YU ZA; AP (GH GM KE LS
MW SD SL SZ TZ UG ZW); EA (AM AZ
BY KG KZ MD RU TJ TM); EP (AT BE
CH CY DE DK ES FI FR GB GR IE IT LU
MC NL PT SE); OA (BF BJ CF CG CI CM
GA GN GW ML MR NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 401/12, A61K 31/4427, A61P 7/02
(11) WO 00/61577 (13) A1
(21) PCT/EP00/03008
(22) 5 Apr/avr 2000 (05.04.2000)
(25) de (26) de
(30) 199 15 930.0 9 Apr/avr 1999
(09.04.1999)
(30) 100 06 799.9 15 Feb/fév 2000
(15.02.2000)
(43) 19 Oct/oct 2000 (19.10.2000)
DE
DE
(54) PRODRUGS
BITORS
OF THROMBIN INHI-
PROMEDICAMENTS D’INHIBITEURS
DE LA THROMBINE
(71) BASF AKTIENGESELLSCHAFT
[DE/DE]; D–67056 Ludwigshafen (DE).
(for all designated States except / pour tous
les États désignés sauf US)
(72, 75) BAUCKE, Dorit [DE/DE]; Bellenstr.
58, D–68163 Mannheim (DE). MACK,
Helmut [DE/DE]; Neustadter Ring 80,
D–67067 Ludwigshafen (DE). SEITZ,
Werner [DE/DE]; Bismarckstrasse 22b,
D–68723 Plankstadt (DE). HORNBER-
GER, Wilfried [DE/DE]; Goldener Winkel
14, D–67434 Neustadt (DE). BACKFISCH,
Gisela [DE/DE]; Talstr. 43, D–69221 Dossenheim
(DE). DELZER, Jürgen [DE/DE];
Franz–Stützel–Str. 78, D–67346 Speyer
(DE).
(74) BASF AKTIENGESELLSCHAFT;
D–67056 Ludwigshafen (DE).
(81) AE AG AL AM AT AU AZ BA BB BG BR
BY CA CH CN CR CU CZ DE DK DM DZ
EE ES FI GB GD GE GH GM HR HU ID
IL IN IS JP KE KG KP KR KZ LC LK LR
LS LT LU LV MA MD MG MK MN MW
MX NO NZ PL PT RO RU SD SE SG SI
SK SL TJ TM TR TT TZ UA UG US UZ
VN YU ZA ZW; AP (GH GM KE LS MW
SD SL SZ TZ UG ZW); EA (AM AZ BY
KG KZ MD RU TJ TM); EP (AT BE CH
CY DE DK ES FI FR GB GR IE IT LU MC
NL PT SE); OA (BF BJ CF CG CI CM GA
GN GW ML MR NE SN TD TG).
Published / Publiée :(c)
(51) 7 C07D 403/02, A61K 31/395, A61P 35/00
(11) WO 00/61578 (13) A1
(21) PCT/US00/09512
(22) 7 Apr/avr 2000 (07.04.2000)
(25) en (26) en