PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
Create successful ePaper yourself
Turn your PDF publications into a flip-book with our unique Google optimized e-Paper software.
<strong>42</strong>/<strong>2000</strong><br />
19 Oct/oct <strong>2000</strong> <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 15159<br />
(22) 6 Apr/avr <strong>2000</strong> (06.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 09/289,255 9 Apr/avr 1999<br />
(09.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
US<br />
(54) METHODS OF INDUCING CANCER<br />
CELL DEATH AND TUMOR REGRES-<br />
SION<br />
PROCEDES POUR L’INDUCTION DE<br />
LA MORT DE CELLULES CANCE-<br />
REUSES ET LA REGRESSION DE TU-<br />
MEURS<br />
(71) SCHERING CORPORATION [US/US];<br />
<strong>2000</strong> Galloping Hill Road, Kenilworth, NJ<br />
07033–0530 (US).<br />
(72) BISHOP, Walter, R.; 17 Hopper Avenue,<br />
Pompton Plains, NJ 07444 (US). BRAS-<br />
SARD, Diana, L.; 432 Tournament Drive,<br />
Apartment 10, Union, NJ 07083 (US). NA-<br />
GABHUSHAN, Tattanahalli, L.; 3 Sunset<br />
Lane, Parsippany, NJ 07054 (US).<br />
(74) GOULD, James, M. et al. / etc.; Schering–Plough<br />
Corporation, Patent Department,<br />
K–6–1 1990, <strong>2000</strong> Galloping Hill<br />
Road, Kenilworth, NJ 07033–0530 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CZ DE DK DM DZ EE<br />
ES FI GB GD GE HR HU ID IL IN IS JP<br />
KG KR KZ LC LK LR LT LU LV MA MD<br />
MG MK MN MX NO NZ PL PT RO RU<br />
SE SG SI SK SL TJ TM TR TT TZ UA UZ<br />
VN YU ZA; AP (GH GM KE LS MW SD<br />
SL SZ TZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY<br />
DE DK ES FI FR GB GR IE IT LU MC NL<br />
PT SE); OA (BF BJ CF CG CI CM GA GN<br />
GW ML MR NE SN TD TG).<br />
(51) 7 A61K 31/4738, 31/4745, C07D 491/22,<br />
491/14, 491/044, 471/04, 213/02<br />
(11) WO 00/61146 (13) A1<br />
(21) <strong>PCT</strong>/US00/09401<br />
(22) 7 Apr/avr <strong>2000</strong> (07.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 09/290,019 9 Apr/avr 1999<br />
(09.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
US<br />
(54) CAMPTOTHECIN ANALOGS AND<br />
METHODS OF PREPARATION THE-<br />
REOF<br />
ANALOGUES DE LA CAMPTOTHE-<br />
CINE ET PROCEDE DE PREPARATION<br />
ASSOCIES<br />
(71) UNIVERSITY OF PITTSBURGH<br />
[US/US]; Cathedral of Learning, Pittsburgh,<br />
PA 15260 (US). UNIVERSITY<br />
OF KENTUCKY RESEARCH FOUN-<br />
DATION [US/US]; 207 Administration<br />
Building, Lexington, KY 40506 (US).<br />
(72) CURRAN, Dennis, P.; 506 S. Linden Avenue,<br />
Pittsburgh, PA 15208 (US). BOM, David;<br />
885 Mirror Street, Pittsburgh, PA 15217<br />
(US). BURKE, Thomas, G.; 1227 Scoville<br />
Road, Lexington, KY 40502 (US).<br />
(74) BARTONY, Henry, E., Jr.; Bartony &<br />
Hare, Law & Finance Building, Suite 1801,<br />
<strong>42</strong>9 Fourth Avenue, Pittsburgh, PA 15219<br />
(US).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG UZ VN YU ZA ZW;<br />
AP (GH GM KE LS MW SD SL SZ TZ UG<br />
ZW); EA (AM AZ BY KG KZ MD RU TJ<br />
TM); EP (AT BE CH CY DE DK ES FI FR<br />
GB GR IE IT LU MC NL PT SE); OA (BF<br />
BJ CF CG CI CM GA GN GW ML MR NE<br />
SN TD TG).<br />
(51) 7 A61K 31/485, 9/16<br />
(11) WO 00/61147<br />
(21) <strong>PCT</strong>/US00/09438<br />
(13) A1<br />
(22) 8 Apr/avr <strong>2000</strong> (08.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 60/128,477 9 Apr/avr 1999<br />
(09.04.1999)<br />
US<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
(54) INJECTABLE NALTREXONE MI-<br />
CROSPHERE COMPOSITIONS AND<br />
THEIR USE IN REDUCING CON-<br />
SUMPTION<br />
ALCOHOL<br />
OF HEROIN AND<br />
COMPOSITIONS MICROSPHERIQUES<br />
INJECTABLES A BASE DE NAL-<br />
TREXONE ET LEUR UTILISATION<br />
DANS LA REDUCTION DE LA<br />
CONSOMMATION<br />
D’ALCOOL<br />
D’HEROINE ET<br />
(71) SOUTHERN RESEARCH INSTITUTE<br />
[US/US]; <strong>2000</strong> Ninth Avenue South, P.O.<br />
Box 55305, Birmingham, AL 35255–5305<br />
(US).<br />
(72) TICE, Thomas, R.; 1915 Forest River<br />
Court, Birmingham, AL 35244 (US).<br />
STAAS, Jay, K.; 101 Ashford Lane, Alabaster,<br />
AL 35007 (US). FERRELL, Teresa,<br />
M.; 608 Paden Drive, Vestavia Hills, AL<br />
35226 (US).<br />
(74) RAE–VENTER, Barbara et al. / etc.;<br />
Rae–Venter Law Group, Suite 440, 260<br />
Sheridan Ave., Palo Alto, CA 94306 (US).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID<br />
IL IN IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MA MD MG MK MN MW<br />
MX NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG UZ VN<br />
YU ZA ZW; AP (GH GM KE LS MW SD<br />
SL SZ TZ UG ZW); EA (AM AZ BY KG<br />
KZ MD RU TJ TM); EP (AT BE CH CY<br />
DE DK ES FI FR GB GR IE IT LU MC NL<br />
PT SE); OA (BF BJ CF CG CI CM GA GN<br />
GW ML MR NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 A61K 31/496, A61P 27/02 // C07D<br />
211/90<br />
(11) WO 00/61148 (13) A1<br />
(21) <strong>PCT</strong>/JP00/02348<br />
(22) 11 Apr/avr <strong>2000</strong> (11.04.<strong>2000</strong>)<br />
(25) ja (26) ja<br />
(30) 11/106<strong>42</strong>5 14 Apr/avr 1999<br />
(14.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
(54) INHIBITORS FOR OPTIC HYPO-<br />
FUNCTION CAUSED BY OPTIC<br />
NERVE CELL INJURY INDUCED BY<br />
FACTORS OTHER THAN OPTIC CIR-<br />
CULATORY DISORDER<br />
INHIBITEURS D’HYPOFONCTION<br />
OPTIQUE PROVOQUEE PAR UNE<br />
LESION D’UNE CELLULE DU NERF<br />
OPTIQUE INDUITE PAR DES FAC-<br />
TEURS AUTRES QUE LES TROUBLES<br />
CIRCULATOIRES OPTIQUES<br />
(71) SENJU PHARMACEUTICAL CO.,<br />
LTD. [JP/JP]; 5–8, Hiranomachi 2–chome,<br />
Chuo–ku, Osaka–shi, Osaka 541–0046 (JP).<br />
KYOTO PHARMACEUTICAL INDUS-<br />
TRIES, LTD. [JP/JP]; 38, Nishinokyo<br />
Tsukinowa–cho, Nakakyo–ku, Kyoto–shi,<br />
Kyoto 604–8444 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) AZUMA, Mitsuyoshi [JP/JP];<br />
4–13–102, Manchidani–cho, Nishinomiya–shi,<br />
Hyogo 662–0031 (JP). YO-<br />
SHIDA, Yukuo [JP/JP]; 6–3, Koyo–cho<br />
3–chome, Kita–ku, Kobe–shi, Hyogo<br />
651–1203 (JP). SAKAMOTO, Yuji [JP/JP];<br />
4–366–1–408, Minamibefu, Nishi–ku,<br />
Kobe–shi, Hyogo 651–2116 (JP).<br />
(74) TAKASHIMA, Hajime; Yuki Building,<br />
3–9, Hiranomachi 3–chome, Chuo–ku,<br />
Osaka–shi, Osaka 541–0046 (JP).<br />
(81) CA JP US; EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE).<br />
(51) 7 A61K 31/545, 47/12, A61P 31/04<br />
(11) WO 00/61149 (13) A1<br />
(21) <strong>PCT</strong>/JP00/02227<br />
(22) 6 Apr/avr <strong>2000</strong> (06.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 9907916.2 7 Apr/avr 1999<br />
(07.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
JP<br />
GB<br />
(54) LONG–ACTING<br />
COMPOSITION<br />
ANTIBACTERIAL<br />
COMPOSITION ANTIBACTERIENNE<br />
A ACTION PROLONGEE<br />
(71) TAKEDA CHEMICAL INDUSTRIES,<br />
LTD. [JP/JP]; 1–1, Doshomashi 4–chome,<br />
Chuo–ku, Osaka–shi, Osaka 541–0045 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) AWAI, Kazuhiro [JP/JP]; 23–15,<br />
Shakujiidai 3–chome, Nerima–ku, Tokyo<br />
177–0045 (JP). YAMAMOTO, Toru<br />
[JP/JP]; 5–11, Higashitokiwadai 3–chome,<br />
Toyono–cho, Toyono–gun, Osaka 563–0103<br />
(JP). DUFFY, Sean [GB/GB]; 57 Tullinavall<br />
Road, Cullyhanna, Newry, Co. Down BT35<br />
0PZ (GB).