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PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO

PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO

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<strong>42</strong>/<strong>2000</strong><br />

19 Oct/oct <strong>2000</strong> <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 15159<br />

(22) 6 Apr/avr <strong>2000</strong> (06.04.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 09/289,255 9 Apr/avr 1999<br />

(09.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

US<br />

(54) METHODS OF INDUCING CANCER<br />

CELL DEATH AND TUMOR REGRES-<br />

SION<br />

PROCEDES POUR L’INDUCTION DE<br />

LA MORT DE CELLULES CANCE-<br />

REUSES ET LA REGRESSION DE TU-<br />

MEURS<br />

(71) SCHERING CORPORATION [US/US];<br />

<strong>2000</strong> Galloping Hill Road, Kenilworth, NJ<br />

07033–0530 (US).<br />

(72) BISHOP, Walter, R.; 17 Hopper Avenue,<br />

Pompton Plains, NJ 07444 (US). BRAS-<br />

SARD, Diana, L.; 432 Tournament Drive,<br />

Apartment 10, Union, NJ 07083 (US). NA-<br />

GABHUSHAN, Tattanahalli, L.; 3 Sunset<br />

Lane, Parsippany, NJ 07054 (US).<br />

(74) GOULD, James, M. et al. / etc.; Schering–Plough<br />

Corporation, Patent Department,<br />

K–6–1 1990, <strong>2000</strong> Galloping Hill<br />

Road, Kenilworth, NJ 07033–0530 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CZ DE DK DM DZ EE<br />

ES FI GB GD GE HR HU ID IL IN IS JP<br />

KG KR KZ LC LK LR LT LU LV MA MD<br />

MG MK MN MX NO NZ PL PT RO RU<br />

SE SG SI SK SL TJ TM TR TT TZ UA UZ<br />

VN YU ZA; AP (GH GM KE LS MW SD<br />

SL SZ TZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY<br />

DE DK ES FI FR GB GR IE IT LU MC NL<br />

PT SE); OA (BF BJ CF CG CI CM GA GN<br />

GW ML MR NE SN TD TG).<br />

(51) 7 A61K 31/4738, 31/4745, C07D 491/22,<br />

491/14, 491/044, 471/04, 213/02<br />

(11) WO 00/61146 (13) A1<br />

(21) <strong>PCT</strong>/US00/09401<br />

(22) 7 Apr/avr <strong>2000</strong> (07.04.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 09/290,019 9 Apr/avr 1999<br />

(09.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

US<br />

(54) CAMPTOTHECIN ANALOGS AND<br />

METHODS OF PREPARATION THE-<br />

REOF<br />

ANALOGUES DE LA CAMPTOTHE-<br />

CINE ET PROCEDE DE PREPARATION<br />

ASSOCIES<br />

(71) UNIVERSITY OF PITTSBURGH<br />

[US/US]; Cathedral of Learning, Pittsburgh,<br />

PA 15260 (US). UNIVERSITY<br />

OF KENTUCKY RESEARCH FOUN-<br />

DATION [US/US]; 207 Administration<br />

Building, Lexington, KY 40506 (US).<br />

(72) CURRAN, Dennis, P.; 506 S. Linden Avenue,<br />

Pittsburgh, PA 15208 (US). BOM, David;<br />

885 Mirror Street, Pittsburgh, PA 15217<br />

(US). BURKE, Thomas, G.; 1227 Scoville<br />

Road, Lexington, KY 40502 (US).<br />

(74) BARTONY, Henry, E., Jr.; Bartony &<br />

Hare, Law & Finance Building, Suite 1801,<br />

<strong>42</strong>9 Fourth Avenue, Pittsburgh, PA 15219<br />

(US).<br />

(81) AE AL AM AT AU AZ BA BB BG BR BY<br />

CA CH CN CR CU CZ DE DK DM EE ES<br />

FI GB GD GE GH GM HR HU ID IL IN<br />

IS JP KE KG KP KR KZ LC LK LR LS LT<br />

LU LV MA MD MG MK MN MW MX NO<br />

NZ PL PT RO RU SD SE SG SI SK SL TJ<br />

TM TR TT TZ UA UG UZ VN YU ZA ZW;<br />

AP (GH GM KE LS MW SD SL SZ TZ UG<br />

ZW); EA (AM AZ BY KG KZ MD RU TJ<br />

TM); EP (AT BE CH CY DE DK ES FI FR<br />

GB GR IE IT LU MC NL PT SE); OA (BF<br />

BJ CF CG CI CM GA GN GW ML MR NE<br />

SN TD TG).<br />

(51) 7 A61K 31/485, 9/16<br />

(11) WO 00/61147<br />

(21) <strong>PCT</strong>/US00/09438<br />

(13) A1<br />

(22) 8 Apr/avr <strong>2000</strong> (08.04.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 60/128,477 9 Apr/avr 1999<br />

(09.04.1999)<br />

US<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

(54) INJECTABLE NALTREXONE MI-<br />

CROSPHERE COMPOSITIONS AND<br />

THEIR USE IN REDUCING CON-<br />

SUMPTION<br />

ALCOHOL<br />

OF HEROIN AND<br />

COMPOSITIONS MICROSPHERIQUES<br />

INJECTABLES A BASE DE NAL-<br />

TREXONE ET LEUR UTILISATION<br />

DANS LA REDUCTION DE LA<br />

CONSOMMATION<br />

D’ALCOOL<br />

D’HEROINE ET<br />

(71) SOUTHERN RESEARCH INSTITUTE<br />

[US/US]; <strong>2000</strong> Ninth Avenue South, P.O.<br />

Box 55305, Birmingham, AL 35255–5305<br />

(US).<br />

(72) TICE, Thomas, R.; 1915 Forest River<br />

Court, Birmingham, AL 35244 (US).<br />

STAAS, Jay, K.; 101 Ashford Lane, Alabaster,<br />

AL 35007 (US). FERRELL, Teresa,<br />

M.; 608 Paden Drive, Vestavia Hills, AL<br />

35226 (US).<br />

(74) RAE–VENTER, Barbara et al. / etc.;<br />

Rae–Venter Law Group, Suite 440, 260<br />

Sheridan Ave., Palo Alto, CA 94306 (US).<br />

(81) AE AG AL AM AT AU AZ BA BB BG BR<br />

BY CA CH CN CR CU CZ DE DK DM DZ<br />

EE ES FI GB GD GE GH GM HR HU ID<br />

IL IN IS JP KE KG KP KR KZ LC LK LR<br />

LS LT LU LV MA MD MG MK MN MW<br />

MX NO NZ PL PT RO RU SD SE SG SI<br />

SK SL TJ TM TR TT TZ UA UG UZ VN<br />

YU ZA ZW; AP (GH GM KE LS MW SD<br />

SL SZ TZ UG ZW); EA (AM AZ BY KG<br />

KZ MD RU TJ TM); EP (AT BE CH CY<br />

DE DK ES FI FR GB GR IE IT LU MC NL<br />

PT SE); OA (BF BJ CF CG CI CM GA GN<br />

GW ML MR NE SN TD TG).<br />

Published / Publiée :(c)<br />

(51) 7 A61K 31/496, A61P 27/02 // C07D<br />

211/90<br />

(11) WO 00/61148 (13) A1<br />

(21) <strong>PCT</strong>/JP00/02348<br />

(22) 11 Apr/avr <strong>2000</strong> (11.04.<strong>2000</strong>)<br />

(25) ja (26) ja<br />

(30) 11/106<strong>42</strong>5 14 Apr/avr 1999<br />

(14.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

(54) INHIBITORS FOR OPTIC HYPO-<br />

FUNCTION CAUSED BY OPTIC<br />

NERVE CELL INJURY INDUCED BY<br />

FACTORS OTHER THAN OPTIC CIR-<br />

CULATORY DISORDER<br />

INHIBITEURS D’HYPOFONCTION<br />

OPTIQUE PROVOQUEE PAR UNE<br />

LESION D’UNE CELLULE DU NERF<br />

OPTIQUE INDUITE PAR DES FAC-<br />

TEURS AUTRES QUE LES TROUBLES<br />

CIRCULATOIRES OPTIQUES<br />

(71) SENJU PHARMACEUTICAL CO.,<br />

LTD. [JP/JP]; 5–8, Hiranomachi 2–chome,<br />

Chuo–ku, Osaka–shi, Osaka 541–0046 (JP).<br />

KYOTO PHARMACEUTICAL INDUS-<br />

TRIES, LTD. [JP/JP]; 38, Nishinokyo<br />

Tsukinowa–cho, Nakakyo–ku, Kyoto–shi,<br />

Kyoto 604–8444 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) AZUMA, Mitsuyoshi [JP/JP];<br />

4–13–102, Manchidani–cho, Nishinomiya–shi,<br />

Hyogo 662–0031 (JP). YO-<br />

SHIDA, Yukuo [JP/JP]; 6–3, Koyo–cho<br />

3–chome, Kita–ku, Kobe–shi, Hyogo<br />

651–1203 (JP). SAKAMOTO, Yuji [JP/JP];<br />

4–366–1–408, Minamibefu, Nishi–ku,<br />

Kobe–shi, Hyogo 651–2116 (JP).<br />

(74) TAKASHIMA, Hajime; Yuki Building,<br />

3–9, Hiranomachi 3–chome, Chuo–ku,<br />

Osaka–shi, Osaka 541–0046 (JP).<br />

(81) CA JP US; EP (AT BE CH CY DE DK ES<br />

FI FR GB GR IE IT LU MC NL PT SE).<br />

(51) 7 A61K 31/545, 47/12, A61P 31/04<br />

(11) WO 00/61149 (13) A1<br />

(21) <strong>PCT</strong>/JP00/02227<br />

(22) 6 Apr/avr <strong>2000</strong> (06.04.<strong>2000</strong>)<br />

(25) en (26) en<br />

(30) 9907916.2 7 Apr/avr 1999<br />

(07.04.1999)<br />

(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />

JP<br />

GB<br />

(54) LONG–ACTING<br />

COMPOSITION<br />

ANTIBACTERIAL<br />

COMPOSITION ANTIBACTERIENNE<br />

A ACTION PROLONGEE<br />

(71) TAKEDA CHEMICAL INDUSTRIES,<br />

LTD. [JP/JP]; 1–1, Doshomashi 4–chome,<br />

Chuo–ku, Osaka–shi, Osaka 541–0045 (JP).<br />

(for all designated States except / pour tous<br />

les États désignés sauf US)<br />

(72, 75) AWAI, Kazuhiro [JP/JP]; 23–15,<br />

Shakujiidai 3–chome, Nerima–ku, Tokyo<br />

177–0045 (JP). YAMAMOTO, Toru<br />

[JP/JP]; 5–11, Higashitokiwadai 3–chome,<br />

Toyono–cho, Toyono–gun, Osaka 563–0103<br />

(JP). DUFFY, Sean [GB/GB]; 57 Tullinavall<br />

Road, Cullyhanna, Newry, Co. Down BT35<br />

0PZ (GB).

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