PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
PCT/2000/42 : PCT Gazette, Weekly Issue No. 42, 2000 - WIPO
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<strong>42</strong>/<strong>2000</strong><br />
15238 <strong>PCT</strong> <strong>Gazette</strong> - Section I - <strong>Gazette</strong> du <strong>PCT</strong> 19 Oct/oct <strong>2000</strong><br />
(25) fr (26) fr<br />
(30) 99/04577 13 Apr/avr 1999<br />
(13.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
FR<br />
(54) 1–AMINO ETHYLINDOLE DERIVA-<br />
TIVES FOR THE TREATMENT OF<br />
URINARY INCONTINENCE<br />
DERIVES DE 1–AMINO ETHY-<br />
LINDOLE POUR LE TRAITEMENT<br />
DE L’INCONTINENCE URINAIRE<br />
(71) SANOFI–SYNTHELABO [FR/FR]; 174,<br />
avenue de France, F–75013 Paris (FR).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) BOVY, Philippe, R. [BE/FR]; 13, rue<br />
du 4 Septembre, F–78750 Mareil Marly<br />
(FR). MOUGENOT, Patrick [FR/FR]; 2,<br />
avenue Ossart, F–92500 Rueil Malmaison<br />
(FR). PHILIPPO, Christophe [FR/FR]; 18,<br />
place des Maitres Vignerons, F–92500 Rueil<br />
Malmaison (FR).<br />
(74) THOURET–LEMAITRE, Elisabeth;<br />
Sanofi–Synthelabo, 174, avenue de France,<br />
F–75013 Paris (FR).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID<br />
IL IN IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MA MD MG MK MN MW<br />
MX NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ<br />
VN YU ZA ZW; AP (GH GM KE LS MW<br />
SD SL SZ TZ UG ZW); EA (AM AZ BY<br />
KG KZ MD RU TJ TM); EP (AT BE CH<br />
CY DE DK ES FI FR GB GR IE IT LU MC<br />
NL PT SE); OA (BF BJ CF CG CI CM GA<br />
GN GW ML MR NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 209/34, 209/40, A61K 31/404,<br />
A61P 35/00<br />
(11) WO 00/61555 (13) A1<br />
(21) <strong>PCT</strong>/EP00/03285<br />
(22) 12 Apr/avr <strong>2000</strong> (12.04.<strong>2000</strong>)<br />
(25) en (26) en<br />
(30) 99106207.6 12 Apr/avr 1999<br />
(12.04.1999)<br />
(30) 99107<strong>42</strong>9.5 27 Apr/avr 1999<br />
(27.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
EP<br />
EP<br />
(54) INDIGOID BISINDOLE DERIVATIVES<br />
DERIVES<br />
D’INDIGOIDES<br />
BISINDOLIQUES<br />
(71, 72) EISENBRAND, Gerhard [DE/DE];<br />
Gustav Kirchhoffstrasse 3, D–69120 Heidelberg<br />
(DE).<br />
(74) PERREY, Ralf; Müller–Boré & Partner,<br />
Grafinger Strasse 2, D–81671 München<br />
(DE).<br />
(81) AE AL AM AT AU AZ BA BB BG BR BY<br />
CA CH CN CR CU CZ DE DK DM EE ES<br />
FI GB GD GE GH GM HR HU ID IL IN<br />
IS JP KE KG KP KR KZ LC LK LR LS LT<br />
LU LV MA MD MG MK MN MW MX NO<br />
NZ PL PT RO RU SD SE SG SI SK SL TJ<br />
TM TR TT TZ UA UG US UZ VN YU ZA<br />
ZW; AP (GH GM KE LS MW SD SL SZ<br />
TZ UG ZW); EA (AM AZ BY KG KZ MD<br />
RU TJ TM); EP (AT BE CH CY DE DK ES<br />
FI FR GB GR IE IT LU MC NL PT SE);<br />
OA (BF BJ CF CG CI CM GA GN GW ML<br />
MR NE SN TD TG).<br />
Published / Publiée :(c)<br />
(51) 7 C07D 209/46, 213/81, 213/82, 217/22,<br />
237/30, 295/14, 307/22, 311/84, 333/20,<br />
335/14, 401/06, 401/12, 405/06, 405/12,<br />
405/14, 409/12, A61K 31/495, 31/496,<br />
31/502, A61P 43/00, 3/06, 9/10<br />
(11) WO 00/61556 (13) A1<br />
(21) <strong>PCT</strong>/JP00/02329<br />
(22) 10 Apr/avr <strong>2000</strong> (10.04.<strong>2000</strong>)<br />
(25) ja (26) ja<br />
(30) 11/102559 9 Apr/avr 1999<br />
(09.04.1999)<br />
(30) 11/118490 26 Apr/avr 1999<br />
(26.04.1999)<br />
(30) 11/119043 27 Apr/avr 1999<br />
(27.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
(54) NITROGEN–CONTAINING HETERO-<br />
CYCLIC COMPOUNDS AND BENA-<br />
MIDE COMPOUNDS AND DRUGS<br />
CONTAINING THE SAME<br />
COMPOSES HETEROCYCLIQUES<br />
CONTENANT DE L’AZOTE ET<br />
COMPOSES DE BENAMIDE ET<br />
MEDICAMENTS<br />
COMPOSES<br />
CONTENANT CES<br />
(71) MEIJI SEIKA KAISHA, LTD. [JP/JP];<br />
4–16, Kyobashi 2–chome, Chuo–ku, Tokyo<br />
104–8002 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) OHKURA, Naoto [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
HIRAIWA, Yukiko [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
MATSUSHIMA, Tetsuya [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
SASAKI, Kazue [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
YAMAMOTO, Takehiro [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
SHIOTANI, Masaharu [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
JP<br />
JP<br />
JP<br />
SUZUKI, Shigeki [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
NAKATANI, Yuuko [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
KURODA, Chizuko [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
NAGASAWA, Mieko [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha,<br />
Ltd., 760, Morooka–cho, Kouhoku–ku,<br />
Yokohama–shi, Kanagawa 222–8567 (JP).<br />
KATANO, Kiyoaki [JP/JP]; Pharmaceutical<br />
Research Center, Meiji Seika Kaisha, Ltd.,<br />
760, Morooka–cho, Kouhoku–ku, Yokohama–shi,<br />
Kanagawa 222–8567 (JP).<br />
(74) SATO, Kazuo et al. / etc.; Kyowa Patent &<br />
Law Office, Fuji Building, Room 323, 2–3,<br />
Marunouchi 3–chome, Chiyoda–ku, Tokyo<br />
100–0005 (JP).<br />
(81) AE AG AL AM AT AU AZ BA BB BG BR<br />
BY CA CH CN CR CU CZ DE DK DM DZ<br />
EE ES FI GB GD GE GH GM HR HU ID<br />
IL IN IS JP KE KG KP KR KZ LC LK LR<br />
LS LT LU LV MA MD MG MK MN MW<br />
MX NO NZ PL PT RO RU SD SE SG SI<br />
SK SL TJ TM TR TT TZ UA UG US UZ<br />
VN YU ZA ZW; AP (GH GM KE LS MW<br />
SD SL SZ TZ UG ZW); EA (AM AZ BY<br />
KG KZ MD RU TJ TM); EP (AT BE CH<br />
CY DE DK ES FI FR GB GR IE IT LU MC<br />
NL PT SE); OA (BF BJ CF CG CI CM GA<br />
GN GW ML MR NE SN TD TG).<br />
(51) 7 C07D 211/48, 405/06, 409/06, A61K<br />
31/445, 31/4525, 31/4535, A61P 9/06<br />
(11) WO 00/61557 (13) A1<br />
(21) <strong>PCT</strong>/JP00/02331<br />
(22) 10 Apr/avr <strong>2000</strong> (10.04.<strong>2000</strong>)<br />
(25) ja (26) ja<br />
(30) 11/103212 9 Apr/avr 1999<br />
(09.04.1999)<br />
(43) 19 Oct/oct <strong>2000</strong> (19.10.<strong>2000</strong>)<br />
(54) 4–HYDROXYPIPERIDINE DERIVA-<br />
TIVES HAVING ANTIARRHYTHMIC<br />
EFFECT<br />
DERIVES DE 4–<br />
HYDROXYPIPERIDINE AYANT UN<br />
EFFET ANTI–ARYTHMIQUE<br />
(71) MOCHIDA PHARMACEUTICAL CO.,<br />
LTD. [JP/JP]; 7, Yotsuya 1–chome, Shinjuku–ku,<br />
Tokyo 160–8515 (JP).<br />
(for all designated States except / pour tous<br />
les États désignés sauf US)<br />
(72, 75) YAMAMOTO, Ichiro [JP/JP]; Mochida<br />
Pharmaceutical Co., Ltd., 7, Yotsuya<br />
1–chome, Shinjuku–ku, Tokyo 160–8515<br />
(JP). ITOH, Manabu [JP/JP]; Mochida<br />
Pharmaceutical Co., Ltd., 7, Yotsuya<br />
1–chome, Shinjuku–ku, Tokyo 160–8515<br />
(JP). YAMASAKI, Fumiaki [JP/JP]; Mochida<br />
Pharmaceutical Co., Ltd., 7, Yotsuya<br />
1–chome, Shinjuku–ku, Tokyo 160–8515<br />
(JP). MIYAZAKI, Yutaka [JP/JP]; Mochida<br />
Pharmaceutical Co., Ltd., 7, Yotsuya<br />
1–chome, Shinjuku–ku, Tokyo 160–8515<br />
JP